Gabapentinoides Flashcards

(14 cards)

1
Q

MoA de acción de gabapentinoides

A

Inh ca de Ca tipo P/Q

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
2
Q

Efectos de gabapentinoides

A

Reduce glutamato
Anticonvulsivo
Analgésico

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
3
Q

Gabapentinoides

A

Gabapentina
Pregabalina

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
4
Q

Indicas de gabapentinoides

A

1º Dolor neuropático
Convulsiones focales
T. de ansiedad

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
5
Q

¿Los gabapentinoides actuan con los R GABA?

A

NO

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
6
Q

Gabapentinoide + potente

A

Pregabalina

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
7
Q

Absorción de gabapentina

A

Dependiente de transp. intestinales

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
8
Q

Inicio de acción de pregabalina

A

Rápido

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
9
Q

Inicio de acción de gabapentina

A

Lento

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
10
Q

Indicas off-label de gabapentinoides

A

Fibromialgia
Sx. de piernas inquietas
Dolor post-qx cron

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
11
Q

EA de gabapentinoides

A

Depresión resp
- EPOC
- Opioides
Sedación
Ataxia
Edema perif.

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
12
Q

Contraindicas de gabapentinoides

A

Insuf renal

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
13
Q

Absorción de pregabalina

A

Lineal

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
14
Q

Indicas específicas de pregabalina

A

Fibromialgia
Ansiedad generalizada

How well did you know this?
1
Not at all
2
3
4
5
Perfectly