drugs Flashcards

1
Q

RAAS-ACE INHIBITORS

A

END IN PRIL
SIDE EFFECTS-COUGH, ANGIOEDEMA, HYPERKALEMIA
BECAUSE YOU ARENT MAKING ANGIOTENSIN 2 SO ITS NOT MAKING ALDOSTERONE SO YOU LOSE NA+ AND H20 THEREFORE RETAINING K+

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2
Q

ANGIOTENSIN 2 BLOCKER-SARTANS

A

DOESNT INTERFERE WITH PRODUCTION OF ANGIOTENSIN, JUST BLOCKS THE RECEPTOR.
USE IF PT CANT TAKE ACEI BECAUSE OF ACE COUGH OR ANGIOEDEMA (STILL RISK)
CAUSES HYPERKALEMIA

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3
Q

ALDOSTERONE ANTAGONIST

A

SPIRONOLACTONE/ EPPLERANONE

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4
Q

ALDOSTERONE ANTAGONIST

A

SPIRONOLACTONE/ EPPLERANONE
BLOCKS ALDOSTERONE RECEPTORS
ELIMINATES VOLUME EXPANSION (ESPECIALLY FOR HYPER ALDOSTERONISM)
HORMONAL SIDE EFFECTS LIKE GYNECOMASTIA, DEEPENING OF VOICE
CAUSES HYPERKALEMIA

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5
Q

ALPHA 2 AGONISTS

A

CLONADINE

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6
Q

ALPHA 2 AGONISTS

A

CLONADINE
BLOCKS NOR EPI
NOR EPI CONTINUES TO BUILD
CAUSES REBOUND HTN IF ABRUPTLY STOPPED, DROWSINESS, XEROSTOMIA

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7
Q

RESERPINE

A

DIMINISHES SYNTHESIS OF NOR EPI

S/E IS DEPRESSION

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8
Q

BETA BLOCKER

A

LOL
ATENALOL, METATROPROLOL
DECREASES HEART RATE AND CONTRACTIITY

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9
Q

ALPHA AND BETA BLOCKER

A

CARVETALOL AND LABETALOL

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10
Q

ALPHA 1 ANTAGONIST (SIN)

A

ALPHA 1 RECEPTORS ARE ON ARTERIES AND VEINS
SIN DRUGS DIALATE ARTERIES AND VEINS
SIDE EFFECT- 1ST DOSE RESPONSE
TAMSALOSIN, DOXAZASIN

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11
Q

DIHYDROPYRIDINE CALCIUM CHANNEL BLOCKERS

A
SUBSTANTIAL AFTERLOAD REDUCERS
NIFEDIPINE
PROFOUND BLOCKADE OF CALCIUM CHANNELS IN ARTERIES
NO EFFECT ON HEART
CAN TRIGGER BARORECEPTORS
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12
Q

DIHYDROPYRIDINE CALCIUM CHANNEL BLOCKERS- S/E

A
DIZZINESS
HA
**PERIPHERAL EDEMA
GINGIVAL HYPERPLASIA
REFLEX TACH
FAST ACTING NIFEDIPINE LINKED TO INCREASED MORTALITY
IF TAKEN IN EXCESS, IT LOSES SELECTIVITY
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13
Q

NONDIHYDROPYRIDINE CHANNEL BLOCKERS

A

BLOCK CALCIUM CHANNELS ON ARTERIES AND ON THE HEART

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14
Q

NONDIHYDROPYRIDINE CHANNEL BLOCKERS

A
VERAPAMIL
ANTI-ARRHYTHMIA 
ACTS LIKE A BETA BLOCKER ON HEART
DECREASES AFTERLOAD, REDUCES CO
THERAPEUTIC USE- ANGINA
CAUSES BAD CONSTIPATION!
CP450 INHIBITOR
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15
Q

NONDIHYDROPYRIDINE CHANNEL BLOCKERS

A

DILTIAZEM AND VERAPIMIL

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16
Q

NONDIHYDROPYRIDINE CHANNEL BLOCKERS

CARDIAC GLYCOSIDES

A
DILTIAZEM
TREATS CHF
ANTI-ARRHYTHMIA 
ACTS LIKE A BETA BLOCKER ON HEART
DECREASES AFTERLOAD, REDUCES CO
THERAPEUTIC USE- ANGINA
CAUSES LESS CONSTIPATION THAN VERAPIMIL
CP450 INHIBITOR!
IANTROPIC DRUG
17
Q

DIURETICS

A

LOOP- FUROSAMIDE-DECREASE CA+

THIAZIDE HCTZ- INCREASE CA+

18
Q

MOST COMMON DIURETIC FOR HTN

A

THIAZIDE

19
Q

ACE INHIBITORS

A

USED FOR DM PTS TO HELP PROTECT KIDNEYS

20
Q

sympatholytics

A

beta blockers-lol
alpha 1 blockers-sin
alpha/beta blockers- labetalol/carvetalol
central acting alpha 2 agonists- clonidine/methyldopa
adrenergic neuron blocker-reserpine/guanadrel/guanethidine

21
Q

reserpine

A

adrenergic neuron blocker