GABAERGIC SYNAPSE Flashcards
1
Q
GABA-A
(Ion Channeling)
Activating Drugs
A
Benzodiazepines
Barbiturates
Alcohol
Neurosteroids
2
Q
GABA-A
(Ion Channeling)
Inhibiting Drugs
A
B-Carbolines (Inverse Agonist)
Bicuculline
PTZ
3
Q
GABA-B
(GPCR)
Activating Drugs
A
Baclofen (Agonist)
4
Q
GABA-B
(GPCR)
Inhibiting Drugs
A
Phaclofen (Antagonist)
5
Q
GABA-Transporter
(Presynaptic)
Inhibiting Drugs
(Block GABA transporter- increase GABA in synapse)
A
Tiagabine
Nipecotic Acid
6
Q
GABA-T
(Transaminase)
Inhibitor
(Indirectly acting agonist- increase GABA)
A
Vigabatrin