opiod analgesics Flashcards
1
Q
Opiod receptor subtypes
A
Mu receptors:
-Mu 1, Mu 2 receptors
Kappa receptors:
-Kappa 1, Kappa 3 receptors
Delta receptors:
-Delta 1, Delta 2 receptors
2
Q
Endogenous Opioids
A
Pro-opiomelanocortin peptides:
-B-endorphin
Pro-enkephalin peptides:
-Met-enkephalin and leu-enkephalin
Prodynorphin peptides:
-Dyn-A, Dyn-B, and alpha neo-endorphin
Endomorphins:
-Endomorphin-1; Endomorphin-2
3
Q
Opiod receptors, endogenous ligands, and function
A
Mu receptors:
Mu1: B-endorphin