Farmacologia vies catecolaminèrgiques: antidepressius, psicoestimulants i al·lucinògens Flashcards

1
Q

Imipramina

A

Antidepressiu tricíclic

Amina primària/secundària

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2
Q

Amitriptilina

A

Antidepressiu tricíclic

Amina primària/secundària

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3
Q

Desipramina

A

Antidepressiu tricíclic

Amina secundària/terciària

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4
Q

Nortriptilina

A

Antidepressiu tricíclic

Amina secundària/terciària

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5
Q

Fluoxetina (prozac)

A

Antidepressiu ISRS

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6
Q

Paroxetina

A

Antidepressiu ISRS

Efecte 2i d’estrenyiment

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7
Q

Sertralina

A

Antidepressiu ISRS

Efecte 2i d’estrenyiment

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8
Q

Fluvoxamina

A

Antidepressiu ISRS

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9
Q

Citalopram

A

Antidepressiu ISRS

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10
Q

Escitalopram

A

Antidepressiu ISRS

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11
Q

Reboxetina

A

Inhibidor selectiu recaptació NA

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12
Q

Venlafaxina

A

Antidepressiu dual

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13
Q

Desvenlafaxina

A

Antidepressiu dual

Metabòlit de venlafaxina

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14
Q

Duloxetina

A

Antidepressiu dual

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15
Q

Tranilcipromina

A

Antidepressiu IMAO
No selectiva de MAO, irreversible
Obsolets per efectes 2s forts

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16
Q

Moclobemida

A

Antidepressiu IMAO
Selectiva MAO-A, reversible
Obsolets per efectes 2s forts

17
Q

Bupropiona

A

Antidepressiu atípic
Augmenta Ser i DA (útil depre atípica)
Baixa llindar convulsiu

18
Q

Mirtazapina

A

Antidepressiu atípic
Bloq Ralfa2
Augmenta alliberació Ser i NA
Ansiolític, hipnòtic i orexigen

19
Q

Trazodona

A

Antidepressiu atípic
Agonista 5-HT (2A/2C)
Bon sedant

20
Q

Propranolol

A

Pot causar depressió

Betabloquejant

21
Q

L-DA, ago DA, isoniazida i corticoides

A

Fàrmacs que poden causar mania

22
Q

Liti

A

Pot causar trastorn bipolar (és un eutimitzant, estabilitzador estat d’ànim)
Efecte 2i: insuficiència renal

23
Q

Valproat, carbamazepina, lamotrigina i gabapentina

A

Anticonvulsius que poden causar trastorn bipolar

24
Q

Dextroamfetamina

A

Estimulant SNC

Alliberen NA, DA i poca Ser en SNC

25
Q

Metamfetamina

A

Estimulant SNC

Alliberen NA, DA i poca Ser en SNC

26
Q

Metilfenidat

A

Estimulant SNC

Alliberen NA, DA i poca Ser en SNC