Diabetes Flashcards

1
Q

Metformina acción:

A
  • Disminuye gluconeogénesis
  • Aumenta sensibilidad a insulina
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2
Q

Metformina características:

A
  • Mejor en obesidad
  • 1ra linea DM2
  • No se metaboliza= Excreción sin cambios
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3
Q

EA metformina

A

Nausea vomito, diarrea, flatulencia

Pérdida de peso, anorexia

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4
Q

Como actúan las tiazolidinedoinas:

A

Pioglitazona y rosiglitazona

  • Aumentan sensibilidad a insulina
  • Aumentan GLUT4
  • Mejoran perfil lipídico en px con dislipidemias
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5
Q

EA de rosiglistazona:

A

disminuye densidad ósea
riesgo cardio

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6
Q

Cómo actúan las sulfanilureas?

A

inhiben canales de K+

  • Aumnetan insulina
  • Disminuyen glucagon
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7
Q

1er fármaco que se agrega a metformina:

A

Glibenclamida

Sulfonilurea

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8
Q

Cuando se recomiendas las glinidas?

A

Repaglinida

  • Px con horarios de comida NO fijos
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9
Q

Miméticos de incretinas:

A

Exenatida
Lireglutida
Lixisenatida

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10
Q

Efectos terapéuticos de miméticos incretinas

A
  • Aumenta insulina
  • Disminuye glucagon
  • Reduce apetito
  • Retrasa vaciamiento gástrico
  • Mejora efecto de metformina
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11
Q

Inhibidores de la DPP4:

A

Aumentan vida de GLP-1

  • Sitagliptina
  • Saxagliptina
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12
Q

Mecanismo de acción acarbosa

A

Inhibe alpha glucosidosa

Disminuye absorción de glucosa

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13
Q

Inhibidores de reabsorción renal de glucosa:

A

Glifozinas:

  • Canaglifozina
  • Empaglifozina
  • Dapaglifozina
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