analgesicos Flashcards

(33 cards)

1
Q

acido acetasilico

A

AINES que producce acidossi metabolica o respiratoria

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2
Q

AINES que producce acidossi metabolica o respiratoria

A

acido acetasilico

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3
Q

AINES que produce agranulocitosis

A

Dipirona

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4
Q

AINES analgesico y antitermico (2)

A

paracetamol y dipirona

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5
Q

Mecanismo periferico de los aines

A

bloqueo de la producccion de prostaglandina tromboxanos y prostaciclinas

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6
Q

Que sintomas renales provocan los aines

A

disminuye FG (retencion agua) dsiminuye flujo sanguineo en IRC

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6
Q

Que sintomas hematologicos provocan los aines

A

anemia trombocitopenia (agranulocitosis la dipirona)

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6
Q

Que provocan los aines al inhibir cox

A

inhiben la produccion de prosttaglandinas y tromboxano

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6
Q

Acciones aines

A

analgesica (inhibicion de COX ) antitermica (evita pirogenos) antiinflamatorios

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7
Q

Que sintomas gastrointestinales provocan los aines

A

inhiben las prostaglandinas que son las encargadas de estimular la produccion de moco por l oqie producen lesiones de intensidad variable

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7
Q

A que niveles provocan los aines efectos adversos

A

gastrointestinales
renaleles
anticogulante (inhibicion de tromboxano A)
hipersensibilidad
reacciones hematologicas

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8
Q

ketofreno

A

AINES

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9
Q

DICLOFENAC

A

AINES

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10
Q

HAPROXENO

A

AINES

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11
Q

Opioides endógenos

A

encefalina
dinorfina
endorfina

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12
Q

endorfina

A

opioide endogeno

13
Q

dinorfina

A

opioide endogeno

14
Q

encefalina

A

opioide endogeno

15
Q

Enzimas degradadoras de los opioides

A

heprilisina y aminopepetidas N

16
Q

morfina

A

opioide agonista puro (mu)

17
Q

metadona

A

opioide agonista puro (mu)

18
Q

oxicodona

A

opioide agonista puro (mu)

19
Q

fentalnilo

A

opioide agonista puro (mu)

20
Q

codeina

A

opioide agonista puro (mu) , dolor leve moderado

21
Buprenorfina
Agonitas de K (lamda) y antagonistas-agonista de u (mu)
22
pentazocina
Agonitas de K (lamda) y antagonistas-agonista de u ( mu)
23
Naltrexona
opiaceo antagonis puro (u>>>delta=K)
24
Naloxona
opiaceo antagonis puro (u>>>delta=K)
25
Naloxona uso
opiaceo antagonis puro tto intoxicacion por opiaceos
26
Naltrexona y metadona uso
tto adiccion a opioides por vida media larga
27
tramadol
agonista opiaceo con actividad monoaminergica
28
tapentadol
agonista opiaceo con actividad monoaminergica
29
La pregabalina es un analgesico?
Si