antibioticos Flashcards

(70 cards)

1
Q

amikacina

A

aminoglucosido
síntesis proteica (30 y 50S)
bactericida

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2
Q

gentamicina

A

aminoglucosido
síntesis proteica (30 y 50S)
bactericida

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3
Q

trobamicina

A

aminoglucosido
síntesis proteica (30 y 50S)
bactericida
Pseudomonas

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4
Q

estreptomicina

A

aminoglucosido
síntesis proteica (30S)
bactericida

Mecanismo: impide apareamiento aa-tRNA y mRNA)

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5
Q

neomicina

A

aminoglucosido
síntesis proteica (30 y 50S)
bactericida

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6
Q

paromicina

A

aminoglucosido
síntesis proteica (30 y 50S)
bactericida

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7
Q

meticilina

A

b lactamico (penicilina)
pared celular (transpeptidacion)
bactericida
No se puede VO

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8
Q

cloxacilina

A

b lactamico (penicilina)
pared celular (transpeptidacion)
bactericida

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9
Q

ampicilina

A

b lactamico (penicilina)
pared celular (transpeptidacion)
bactericida
Tto elección meningitis infantil

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10
Q

amoxicilina

A

b lactamico (penicilina)
pared celular (transpeptidacion)
bactericida

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11
Q

piperacilina

A

b lactamico (penicilina)
pared celular (transpeptidacion)
bactericida

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12
Q

imipenem

A

b lactamico (carbapenem)
pared celular (transpeptidacion)
bactericida

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13
Q

meropenem

A

b lactamico (carbapenem)
pared celular (transpeptidacion)
bactericida

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14
Q

ertapenem

A

b lactamico (carbapenem)
pared celular (transpeptidacion)
bactericida

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15
Q

clavulanico

A

b lactamico (inhibidor)
pared celular (transpeptidacion)
bactericida

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16
Q

clavulanico

A

b lactamico (inhibidor)
pared celular (transpeptidacion)
bactericida

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17
Q

avibactam

A

b lactamico (inhibidor)
pared celular (transpeptidacion)
bactericida

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18
Q

avibactam

A

b lactamico (inhibidor)
pared celular (transpeptidacion)
bactericida

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19
Q

varbovactam

A

b lactamico SIN ANILLO (inh)
pared celular (transpeptidacion)
bactericida

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20
Q

aztreonam

A

b lactamico (monobactama)
pared celular (transpeptidacion)
bactericida
Importante en metalolactamasas y alergicos

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21
Q

vancomicina

A

glicopeptido
pared celular (union NAG-NAM)
bactericida

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22
Q

teicomicina

A

glicopeptido
pared celular (union NAG-NAM)
bactericida

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23
Q

fosfomicina

A

sin grupo
pared celular (formación NAM)
bactericida

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24
Q

bacitracina

A

sin grupo
pared celular (bactoprenol)
bactericida

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25
daptomicina
sin grupo (lipopeptido) membrana plasmatica (despolarización dpte de Ca) bactericida
26
colistina
polimixina membrana plasmatica (unen lipopolisac, detergente) bactericida Inhalatorio para pseudomonas-FQ
27
ácido nalixicido
quinolonas (1gen) ANs (topoisomerasas) bactericida
28
norfloxacino
quinolonas (2gen) ANs (topoisomerasas) bactericida
29
ciprofloxacino
quinolonas (2gen) ANs (topoisomerasas) bactericida Y pestis y Shigella
30
oflofloxacino
quinolonas (3gen) ANs (topoisomerasas) bactericida
31
levofloxacino
quinolonas (3gen) ANs (topoisomerasas) bactericida
32
moxifloxacino
quinolonas (4gen) ANs (topoisomerasas) bactericida
33
metronidazol
imidazol ANs bactericida
34
Cefoxitina
b lactamico (cefamicina, cefalosporina 2) pared celular (transpeptidacion) bactericida
35
cefepima
b lactamico (cefalosporina 4) pared celular (transpeptidacion) bactericida
36
ceftazidima
b lactamico (cefalosporina 3) pared celular (transpeptidacion) bactericida Pseudomonas
37
trimetoprim
Sin grupo, similar a sulfonamidas metabolismo (ac folico) bacteriostatico
38
sulfametoxazol
sulfonamida metabolismo (ac folico) bacteriostatico
39
cotrimoxazol
SULFAMETOXAZOL+TRIMETOPRIM metabolismo (ac folico) Bactericida !!!!
40
claritromicina
macrolido (14c) proteínas (translocacion) bacteriostatico
41
claritromicina
macrolido (14c) proteínas (translocacion) bacteriostatico
42
eritromicina
macrolido (14c) proteínas (translocacion) bacteriostatico
43
azitromicina
macrolido (15) proteínas (translocacion) bacteriostatico
44
espiramicina
macrolido (16c) proteínas (translocacion) bacteriostatico
45
cloranfenicol
anfenicoles proteínas (50S) bacteriostatico Mecanismo: inhibidor competitivo del 23S
46
doxiciclina
tetraciclina (Vd larga) proteínas (30S, bloqueando sitio A) bacteriostatico
47
minociclina
tetraciclina (Vd larga) proteínas (30S) bacteriostatico
48
clindamicina
lincosamida proteínas (50s) bacteriostatico
49
linezolid
sin grupo proteínas (50s) bacteriostatico
50
ácido fusidico
sin grupo proteínas (50s, elongación) bacteriostatico
51
ketolidos
derivados de macrolidos proteínas (50s) bacteriostatico
52
espectinomicina
sin grupo proteínas (50s) bacteriostatico
53
isoniazida
antituberculoso síntesis micolicos
54
isoniazida
antituberculoso síntesis micolicos
55
pirazinamida
antituberculoso síntesis micolicos
56
rifampicina
antituberculoso ARNpol
57
etambutol
antituberculoso síntesis pared celular
58
etambutol
antituberculoso síntesis pared celular
59
dapsona
antileproso ácido folico
60
dapsona
antileproso ácido folico
61
clofazimina
antileproso ANs micobact
62
Cefoperazona
b lactamico (cefalosporina 3) pared celular (transpeptidacion) bactericida Antipseudomonas
63
Ceftarolina
b lactamico (cefalosporina 5) pared celular (transpeptidacion) bactericida SARM
64
Ceftriaxona
b lactamico (cefalosporina 3) pared celular (transpeptidacion) bactericida T whipplei, N gonorrea, H ducreyi Cualquier meningitis salvo listeria
65
Cefotaxmina
b lactamico (cefalosporina 3) pared celular (transpeptidacion) bactericida Meningitis grave H influenziae Meningococo
66
Tobramicina
aminoglucosido síntesis proteica (30 y 50S) bactericida
67
Fidaxomicina
Macrólido síntesis proteica (50S, translocación) bactericida C difficile
68
Cefmetazol
b lactamico (cefamicina, cefalosporina 2) pared celular (transpeptidacion) bactericida
69
Cefa—
b lactamico (cefalosporina 1) pared celular (transpeptidacion) bactericida
70
Puromicina
Sin grupo Proteínas (analogo de aa-tRNA)