antibiyotikler Flashcards

1
Q

RNA
RR

A

Rifampin
rifabutin

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2
Q

DNA
KM

A

Kinolonlar
metronidazol(anaerobolarda etkili)

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3
Q

30S
ATO

A

AMİNOGLİKOZİT
TETRACYCLİNES
OXAZOLİDİN

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4
Q

50S
KSKM

A

KLORAMFENİKOL
STREPTOMİSİN
KLİNDAMİSİN
MACROLİD

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5
Q

Antibiyotiklerin etki mek

A

hücre duvarını bozma
protein sentezi inh
nükleik asit sentezi
antimetobolik

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6
Q

Betalaktamlar
PSSKMB

A

PENİSİLİNLER
SEFOLOSPORİN
SEFAMİSİNLER
KARPANEMLER
MONOBAKTAM
B LAKTMAZ İNH

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7
Q

BETA LAKTAMAZ İNH
SKTA

A

SULBAKTAM
KLAVULONİK ASİT
TAZOBAKTAM
AVİBAKTAM

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8
Q

PENİSİLİNAZ DİRENÇLİ PENİSİLİN
mndko

A

METİSİLİN
NAFSİLİN
DİKLOkSASİLİN
KLOKSASİLİN
OKSASİLİN

-STAFİLOKOKLARA ETKİLİLER

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9
Q

GENİŞ SPEKTRUMLU
AKÜ

A

AMİNOPENİSİLİN (amoksisilin ampisilin)
Karboksipenislin(karbenislin tikarsilin)
üreideopenisilin(piperasilin)
-gr- çomaklar

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10
Q

sefamisinler

A

b laktamazlardan etkilenmez
potansiyeli en yüksek sefalosporin
sefotetan
sefoksitin

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11
Q

Karbapenemler
ime

A

imipenem
meropenem
ertapenem
-metisilin dirençli stafilokoklara etkili

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12
Q

Monobaktam

A

aztreonam
en dar spekli b.laktam
h.influenza

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13
Q

Glikopeptitler
VT

A

VANKOMİSİN
TEİKOPLANİN
-g+ etkili
-d alanin d alanine bağlanır

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14
Q

Lipopeptitler
DF

A

DAPTOMİSİN
-İrreversibl olarak stoplazmik membrana bağlanır
-metisilin dirençli stafilokok + streptokok
-vankomisin dirençli enterokok
FOSFOMİSİN
-NAMA sentezi engeller
-MRSA + VRE etki spektrumu

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15
Q

Polipeptitler
BP

A

BASİTRASİN
-Toxit sebeplerden ötürü topikal uygulanır
-stafilokok +gas deri enf
Polimiksinler
-hücre geçirgenliğini artır lipopolisakkaritler ve fosfolipitlere etkileşerek
-acibetobakteriler asye etkili

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16
Q

Protein sentezini inh edenler
AKTOLS

A

AMİNOGLİKOZİTLER(AMİKASİN GENTAMİSİN TOBRAMİSİN)
KLORAMFENİKOL
TETRASİKLİNLER
OKZALİDİNON
LİNKOZAMİDLER(KLİNDAMİSİN LİNKOMİSİN)
STREPROGRAMİNLER

17
Q

spektrumu dar antistafilokoklar

A

mupirosin
fusidik asit

18
Q

nükleik asit sentezini inh edenler
K
RR
N
NN

A

Kilononlar
-DNA giraz + topoizomeraz 4
RİFAMİSİN RİFAMPİNLER
-DNA bağımlı RNA pollimeraz
Novobiyosin
-DNA giraz enzim fonksiyonu engelleme
NİTROFURANLAR NİTROİMİDAZOLLER
- DNA iplikçiğinde kırılma
-protein sentez inh
-nitrit radikal olusumu

19
Q

Antimetabolitler
ST
DP

A

Sülfonamidler ve trimetoprim
-tetrahidropteroik asit esentetaz ing
-dihidrofolik asit sentataz inh(mikobakteri lepra cüzzam hastalığI)
Dapson ve Paraaminosalisilik asit