Autonomic Pharmacology Flashcards
(53 cards)
Hemicholinium
Inhibitor of choline uptake
Botulin toxin
By brevin prevent Ach release in post synaptic
Edrophonium
Reversible AchE inhibitor
Physostigmine
Reversible AchE inhibitor
Neostigmine
Reversible AchE inhibitor
Malathion
Irreversible AchE inhibitor - indirect acting cholinomimetics
Parathion
Irreversible AchE inhibitor - indirect acting cholinomimetics
Betanechol
Muscarinic Agonist; lieus and urinary retention
Methacoline
Muscarinic Agonist; bronquial hyper reactivity
Pilocarpine
Muscarinic Agonist; xerostomia - glaucoma
Endrophonium
Acetylcholinesterase inhibitor; miastenia gravis
Physostigmine
Acetylcholinesterase inhibitor; glaucoma- atropine over dose
Neostigmine
Acetylcholinesterase inhibitor; ileus- urinary retention- miastenia gravis
Pyridostigmine
Acetylcholinesterase inhibitor; ileus - urinary retention- miastenia gravis
Donepezil
Acetylcholinesterase inhibitor; Alzheimer
Rivastigmine
Acetylcholinesterase inhibitor; Alzheimer
Organophosphates
Acetylcholinesterase inhibitor; insecticide- nerve gas ( sarin)
Atropine
Muscarinic receptor antagonist - antispasmodic, antisecretory, AchE inhibitor OD, ophthalmology
Tropicamide
Muscarinic receptor antagonist; ophthalmology
Ipratropium
Muscarinic receptor antagonist; asthma and COPD
Scopolamine
Muscarinic receptor antagonist; used in motion sickness
Benztropine
Muscarinic receptor antagonist; lipid soluble (CNS entry) used in Párkinsonism and acute extrapyramidal symptoms by antipsychotics
Oxybutynin
Muscarinic receptor antagonist; overactive bladder (urge incontinence)
Hexamethonium
Nicotine Receptor Antagonist; Ganglion blocking agents;