Drug Group 3 Flashcards
(28 cards)
CLASS:
BRONCHODILATOR
MOA:
- RELAXATION OF BRONCHIAL TREE AND PERIPHERAL VASCULATURE WITH MINIMAL CARDIAC EFFECTS.
INDICATIONS:
- BRONCHIAL ASTHMA, BRONCHOSPASM ASSOCIATED WITH EXERCISE.
DOSAGE:
.25MG SC
TERBUTALINE SULFATE (BRETHINE)
CLASS:
SYMPATHOMIMETIC
MOA:
- POSITIVE INOTROPIC (CONTRACTILITY), CHRONOTROPIC (RATE), AND DROMOTROPIC (NODE CONDUCTION) EFFECTS
INDICATIONS:
- ANAPHYLAXIS
- ASTHMA
CONTRAINDICATIONS:
- HYPERTENSION
- HYPOTHERMIA
- PULMONARY EDEMA
- MYOCARDIAL ISCHEMIA
- CARDIAC DISEASES
DOSAGE:
1: 1000 ADULT .3Mg - .5Mg SC/IM (ANAPHYLAXIS)
1: 10,000 1Mg q 3-5 MINS IV/IO (CARDIAC)
ADVERSE REACTIONS:
- NERVOUSNESS
- RESTLESSNESS
- HEADACHE
- TREMOR
EPINEPHRINE (ADRENALIN)
(PROVENIL, VENTOLIN)
ALBUTEROL
CLASS:
- SYMPATHOMIMETIC
INDICATIONS:
- BRONCHIAL ASTHMA
- PREVENTION OF BRONCHOSPASM
- CROUP
EPINEPHRINE RACEMIC (MICRONEFRIN)
CLASS:
ANTICHOLERGENIC, BRONCHODILATOR
INDICATIONS:
PERSISTENT BRONCHOSPASMS, COPD EXACERBATION.
CONTRAINDICATIONS:
HYPERSENSITIVITY TO IPRATROPIUM, ATROPINE, ALKALOIDS, PEANUTS.
DOSAGE:
250 - 500 MCG NEBULIZED EVERY 20 MINUTES, MAX 3 TREATMENTS
IPRATOPIUM (ATROVENT)
CLASS:
SYMPATHOMIMETIC, BRONCHODILATOR
MOA:
- BETA 2 SELECTIVE
- RESULTS IN SMOOTH-MUSCLE RELAXATION IN THE BRONCHIAL TREE
DOSAGE:
2.5 MG (REPEAT AS NEEDED)
CONSIDERATIONS:
- MAY PRECIPITATE ANGINA PECTORIS AND TACHYCARDIC DYSRHYTHMIAS.
- EFFECTS MAY BE DIMINISHED WITH BETA-BLOCKERS.
ALBUTEROL (PROVENIL, VENTOLIN)
(BRETHINE)
TERBUTALINE SULFATE
(ATROVENT)
IPRATOPIUM
(NEO-SYNEPHRINE)
PHENYLEPHRINE
(PITRESSIN)
VASOPRESSIN
(ADRENALIN)
EPINEPHRINE
CLASS:
SYMPATHOMIMETIC BRONCHODILATOR
LEVALBUTEROL (XOPENEX)
CLASS:
- SYMPATHOMIMETIC
ISOETHRINE (BRONCHOSOL, BRONKOMETER)
(ALUPENT)
METAPROPERENOL SULFATE
(LEVOPHED)
NOREPINEPHRINE BITARTRATE
CLASS:
- SYMPATHOMIMETIC VASOPRESSOR
MOA:
- POTENT ALPHA-AGONIST RESULTING IN INTENSE PERIPHERAL VASOCONSTRICTION
INDICATIONS:
- CARDIOGENIC SHOCK
- UNRESPONSIVE TO FLUID RESUSCITATION
NOREPINEPHRINE BITARTRATE (LEVOPHED)
(ZICAM)
OXYMETAZOLINE
CLASS:
VASOCONSTRICTOR
OXYMETAZOLINE (ZICAM)
CLASS:
BRONCHODILATOR
MOA:
ACTS DIRECTLY ON BRONCHIAL SMOOTH MUSCLE CAUSING RELAXATION.
INDICATIONS:
BRONCHIAL ASTHMA, COPD
METAPROPERENOL SULFATE (ALUPENT)
CLASS:
VASOPRESSOR (ADRENERGIC, ALPHA AGONIST)
PHENYLEPHRINE (NEO-SYNEPHRINE)
(XOPENEX)
LEVALBUTEROL
(BRONCHOSOL, BRONKOMETER)
ISOETHARINE
(MICRONEFRIN)
EPINEPHRINE RACEMIC
CLASS:
- VASOPRESSOR
MOA:
- STIMULATION OF SMOOTH MUSCLE RECEPTORS
- ADH (ANTI-DIURETIC HORMONE)
INDICATIONS:
- CAN BE USED IN THE PLACE OF EPINEPHRINE IN CARDIAC ARREST, VASODILATORY SHOCK.
VASOPRESSIN (PITRESSIN)