Drug list to know Flashcards
(78 cards)
1
Q
Phenothiazine tranquilizers
A
- Acepromazine - Chlorpromazine - Propionylpromazine - Promethazine
2
Q
Butyrophenone tranquilizers
A
- Azaperone
- Droperidol
- Fluanisone
3
Q
Alpha-2- agonists
A
- Xylazine
- Detomidine (Eq)
- Medetomidine (Small animals)
- Dexmedetomidine (Small animals)
- Romfidine (Eq)
4
Q
Alfa-2-antagonist
A
- Atipamezole
- Yohimbine
5
Q
Benzodiazepines
A
- Diazepam - Midazolam - Zolazepam - Alprazolam - Lorzepam
6
Q
Barbiturates
A
- Phenobarbital - Pentobarbital - Thiopental - Methohexital
7
Q
Antidepressants
A
- TCAs, SRIs, MAOIs, Lithimu
- TCAs:
- Amitriptyline, Clomipramine
- SRIs:
- Fluoxetine, Flavuoxamine, Sertraline
MAOs:
- Selegiline
8
Q
Parasympathomimetics
A
Direct Parasympathomimetics:
- Choline esters:
- Acetylcholine
- Carbachol,
- Bethanechol,
- Pilocarpine
Indirect parasympathomimetics:
- Cholinesteraseinhibitors
- Reversible inhibitors: Phyostigmine, Neostigmine, Edrophonium, Pyridostigmine
- Non-reversible: Organophosphates
9
Q
Parasympatholytics
A
- Atropin - Glycopyrrolate - Ipratropium - Homatropine - Tropicamide - Benzetimide
10
Q
Sympathomimetics
A
Non-specific sympathomimetics:
- Epinephrine
- Norepinephrine
- Dopamine -
Specific sympathomimetics:
- B-1 agonist: Dobutamine
- B-2 agonist: Clenbuterol, Salbuterol, Terbutaline, Salmeterol
- A-1 agonist:
- Local use: Phenylephrine, Xylometazoline, Oxymetazoline
- Systemic use: Phenylephrine, Phenylpropanolamine
- A-2 agonist: Xylazine, Detomidine, Medetomidine, Romfidine
11
Q
Sympatholytics
A
A- Adrenoceptor antagonists:
- Non-specific: Phenoxybenzamine, Phentolamine, Tolazoline
- A1-antagonist: Prazosine, Doxasozine
- A2-antagonist: Atipamezole, Yohimbine
B-adrenoreceptor antagonists:
- Non-specific: Propranolole, Timolole
- B1- antagonists: Metoprolole, Atenolole
12
Q
Xanthine derivates and CNS stimulants
A
- Caffeine - Theophylline - Theobromine - Aminophylline - Propenthophylline - Doxapram
13
Q
Opioids
A
- Morphine - Codeine - Methadone - Fentanyl - Sufentanil - Alfentanil - Remifentanil - Tramadol - Hydrocodone - Oxycodone - Butorphanol - Buprenorphine - Naloxone
14
Q
Antiepileptics
A
- Phenobarbital - Potassium bromide - Levetiracetam - Imepitoin - Gabapentin
15
Q
Injectable Anesthetics
A
- Pentobarbital - Thiopental - Methohexital - Propofol - Etomidate - Ketamine - Tiletamine - Alfaxalone - Alfadolone
16
Q
Inhalational anesthetics
A
- Halothane - Isoflurane - Sevoflurane - Desflurane - dinitrogen oxide
17
Q
Peripheral muscle relaxants
A
- Tubocurarine - Vecuronium - Atracurium - Rocuronium
18
Q
Local anesthetics
A
- Procaine - Oxybuprocaine - Tetracaine - Lidocaine - Bupivacaine - Ropivacaine - Prilocaine - Articaine
19
Q
NSAIDs
A
- Salicylates:
- Acetylsalicylic acid, Sodium salicylate, Sulfasalazine, Mesalazine
- Arilpropionic acids:
- Ketoprofen - Carprofen - Vedaprofen
- Heteroaryl acetic acids:
- Diclofenac, Etodolac (COX-2)
- Anthranilic acids:
- Flunixin meglumine, Tolfenamic acids
- Oxicams:
- Piroxicam, tenoxicam
- Meloxicam (COX-2)
- Anilin derivatives:
- Paracetamol (COX-3)
- Pyrazoles:
- Metamizole sodium (COX-3)
- Coxibs:
- Fibrocoxib - Robenacoxib - Deracoxib - Cimicoxib - Mavacoxib
20
Q
Glucocorticoids
A
- Cortisol: Short effect
- Prednisolone: Medium effect
- Methylprednisolone : Medium effect
- Triamcinolone: Medium effect
- Dexamethasone: Long effect
- Betamethasone: Long effect
- Fluticasone: Local
- Beclomethasone: Local
- Budesonide: Oral
21
Q
Mineralocorticoids
A
Fludrocortisone
22
Q
Antihistamines
A
1st generation:
- Hydroxyzine, Diphenhydramine, Dimenhydrinate
- Chlorpheniramine, Dimetindene, Cyproheptadine, Promethazine
2nd generation:
- Cetirizine, Levocetirizine, Loratadine
23
Q
JAK inhibitors
A
- Oclacitinib
24
Q
Monoclonal antibodies
A
- Lokivetmab
25
Immunosuppressant agents
_1. Antimetabolites:_
- Purine analogues:
* Azathioprine, Mycophenolate mofetil
- Pyrimidine analogues:
* Leflunomide
- Folic acid antagonist:
* Methotrexate
_2. Alkalyting agents:_
* Cyclophosphamide
_3. Cytokine gene expression inhibitors_
- Calcineurin-inhibitors
* Cyclosporin
* Tacrolimus, Pimecrolimus
26
Antiarrhytmic drugs
- Quinidine - Procainamide - Lidocaine - Mexiletine - Propranolol - Metoprolol - Sotalol - Amiodarone - Diltiazem - Verapamil - Digoxin
27
Drugs acting on the cardiovascular system
- Pimobendan - Enalapril - Benazepril - Ramipril - Lizinopril - Losartan - Valsartan - Telmisartan - Amlodipin - Nitroglycerin - Hydralazine
28
Diuretics
- Spironolactone - Furosemide - Torasemide - Hydrochlorothiazide - Chlorothiazide - Acetazolamide - Dorzolamide - Brinzolamide - Mannitol
29
Antitussives
- Codein - Dihydrocodein - Butorphanol - Tramadol - Dextromethorphan
30
Mucolytics and expectorants
- Acetylcysteine - Carbocysteine - Bromhexine - Dembrexine - Ambroxol - Guaifenesin - Ammonium chloride - Volatile oils
31
Bronchodilators
- Clenbuterol - Salbutamol - Terbutalin - Salmeterol - Formoterol - Ephedrine - Theophylline - Aminophylline - Propentophylline - Ipratropium
32
Emetics and antiemetics
- Xylazine - Apomorphine - Acepromazine - chlorpromapzine - Thiethylperazine - Metoclopramide - Domperidone - Ondasetron - Dolasetron - Maropitant - Diphenhydramine
33
Prokinetic agents
- Metoclopramide - Domperidone - Cisapride - Prucalopride - Tegaserod
34
Antacids and coating agents
- Magnesium oxide - Magnesium hydroxide - Aluminium hydroxide - Sucralfat
35
Acid secretion inhibitors
- Famotidine - Ranitidine - Omeprazole - Pantoprazole - Lansoprazole
36
Laxatives and coating agents
- Magnesium sulfate - Sodium sulfate - Sodium hydrogenphosphate - Potassium citrate - Lactulose - Phenolphthalein - Bisacodyl - Docusate - Liquid paraffin
37
Absorbents and Adstringents
- Activated charcoal - Kaolin - Montmorillonite - Attapulgite - Bismuth salts - Tannic acid
38
Hormones of the hypothalamus and the pituitary gland
_1. Releasing nad Inhibitory hormones (RHs and IHs)_
From hypothalamus --\> Adenohypophysis
* Gonadotropin-releasing hormone (GnRH)
* Corticotropin-releasing hormone (CRH)
_2. Hormones of the pituitary gland_
- Adenohypophysis:
* Somatotropin (STH, GH)
* Adrenocorticotropic hormone (Corticotropin, ACTH)
- Neurohypophysis:
* Antidiuretic hormone (ADH, Vasopressin)
* Oxytocin
- Non-hypophyseal gonadotropins:
* Human Chorionic gonadotropin (hCG)
* Pregnant mares serum gonadotropin (PMSG, eCG)
- Buserelin - Fertirelin - Gonadorelin - Deslorein - ECG - HCG - Oxytocin - Desmopressin
39
Hormones of the Adenohypophysis
_1. Somatotropin inj., Somatrem inj. (GH, STH, ST)_
- Released by: GHRH
- Inhibited by: GHIH and Ghrelin
GH-inhibition (Somatostatin)
- Synthetic analogues:
* Octreotide (SC)
* Lanreotide (SC, IM)
- Dopamine agents:
* Cabergoline (PO)
- GH receptor antagonist, IGF-I synthesis inhibition:
* Pegvisomant
_2. Corticotropin_
- Natural form: ACTH
- Synthetic: Tetracosactide (IV, IM9
_3 Thyrotropin, THS, Thyrotropin alfa_
_4. Gonadotropin, FSH, LH_
40
Hormones of Neurohypophysis:
1. _ADH, Vasopressin_,
- Preparations:
* Desmopressin (IV, SC, IM, PO, Nasal)
* Vasopressin (natural): nasal spray
* Chlorpropamide (PO)
- Overproduction of ADH (SIADH) preparations:
* Conivaptan (IV)
* Tolvaptan and Lixivaptan (PO)
* Non-specific drugs: Demelocycline, tetracyclines, lithium
_2. Oxytocin_
41
Adrenal hormones, drugs for treatment of Cushings and Addisons disease
Treatment of Hypoadrenocorticism (Addisons):
- Aldosterone: for research use only
- Desoxycortisone pivalate (DOCP) (SC)
- Fludrocortisone acetate (PO, SC)
Treatment of Hyperadrenocorticism:
- Pituitary dependent:
* Bromocriptine, Cyproheptadine
- Pituitary and/or adrenal-dependent:
* Ketoconazole
* Mitostane, Trilostane
42
Pharmacology of sexual functions (GnRH, gonadotropins, prostaglandins)
- GnRH: FSH, LH
* Gonadorelin: Eq, Bo, sus, rabbit
* Buserelin: Eq, Bo, Rabbit
* Fertirelin: Bo
* Lecirelin: Bo
* Deslorelin: dog
- Non-pituitary gonadotropins:
* PMSG: Werfaser, Gonadophyl, Suidan
* hCG: Werfachor, Suidan, Prolan, Nymphalon, P.G
- Prostaglandins:
* Alfaprostol
* Dinoprost
* Cloprostenol
* Luprostiol
* Etiproston
43
Androgens
Andriol, Retandrol, Sesoral
44
Progestogens
- Flurogeston - Norgestomet - Altrenogest - Medroxyprogesteron acetate - Proligeston - Megestrol acetate
Antiprostagenes:
- Aglepristone, Bromocripitne, Cabergoline
45
Prostaglandins
Alfaprostol, Dinoprost, cloprostenol, Luprostiol, Etiproston
46
Oestrogens
- Oestriol , Oestradiol benzoate, Oestradiol cypionate
47
Progesteron antagonists
- Aglepriston
48
Dopamine agonists
- Cabergolin - Bromocriptin
49
Insulin and other antidiabetics
_Classification of insulin products by:_
- 1. orgin: natural or biosynthetic
- 2. Purity:
* Regular insulin: 4-8hr
* Insulin Zinc suspension (Caninsulin): 12-24ht
* Protamine Zinc insulin: 24-36ht
* Isophane insulin
_Orally actuve hypoglycaemic drugs:_
- 1. Sulphonylurea substances
* Tolbutamide: short action
* chorpropamide: long action
* Metahexamide
* Glibenclamide
* Glipizide
- 2. Acarbose, PO
- 3. Biguanides
* Fenifam, Buformine, Methformine
- 4. Thiazollidine diones
* Troglitazone, Draglitazone
50
Thyroid hormones, drugs for treatment of hypo-hyperthyroidism
- Calcitonin (Salcatonin: for treatment of hypercalcemia
- Preparations for hypothyroidism:
* L-thyroxine/Levothyroxine: PO, dog, cat, horse
* L-thyroxine-Na: IV, SC
* L-triiodothyronine: PO
- Preparations ofr hyperthyroidsim:
* Iodine
* I131 isotope
* Thiouracils: Thiouracil, Propylthiouracil, Thiamizole
51
Other hormones, hormone antagonists
- Insuline - Glipizide - Acarbose - Fludrocortisone - Trilostane - Mitotane - Levothyroxine - Methimazole - Carbimazole
52
Anthelmintichs
_Benzimidazoles:_
- Mebendazole, Albendazole, Fenbendazole, Flubendazole, Triclabendazole, Oxfendazole
_Probenzimidazoles (Prodrugs)_
- Febantel, Netobimin
_Imidazothiazoles_
- Levamisole
_Tetrahydropyrimidines_
- Pyrantel
_Isoquinolin and Benzazepin derivatives_
- Epsiprantel
_Other endoparasiticides:_
- Emodepside
- Monepantel
- Clorsulon
_Salicylanilides and Substituted phenols:_
- Niclosamide
- Oxyclozanide
_Monocyclic lactones_
- Avermectin: Ivermectin, Doramectin, Selamectin, Eprinomectin
- Milbemycins: Moxidectin, Milbemycin oxime
53
Ectoparasiticides
_Organophosphates:_
- Diazinon, Phoxim, Coumaphos
_Carbamates:_
- Propoxur
_Pyrethroids:_
- Permethrin
- Deltamethrin
- Tetramethrin
_Amitraz_
_Fipronil_
_Pyriprol_
_Neonicotinoid insecticides_
- Imidacloprid
- Nitenpyram
- Dinotefuran
_Isoxazolines_
- Fluralaner
- Afocolaner
- Sarolaner
- Lotilaner
_IGRs_
- Juvenile hormone analogues: Methoprene, Pyriproxyfen
- Chitin synhtesis inhibitors: Lufenuron
54
Antineoplastic drugs
- Methotrexate
- Mitoxantrone
- Carboplatin
- Cyclophosphamide
- Chlorambucil
- Lomustine
- Doxorubicin
- Vincristine
- Vinblastine
- Toceranib
- Mastinib
- Asparaginase
55
Antifungal drugs
- Terbinafin
- Naftifine
- Natmycin
- Nystatin
- Clotrimazole
- Enilconazole
- Miconazole
- Bifonazole
- Ketoconazole
- Posaconazole
- Itraconazole
- Fluconazole
- Voriconazole
- Griseofulvin
- Amphotericin B
56
Antiprotozoal agents
- Monensin
- Salinomycin
- Narasin
- Lasalocid
- Maduramycin
- Semduramycin
- Diclazuril
- Toltrazuril
- Ponazuril
- Clazuril
- Clopidol
- Robenidine
- Paromomycin
- Decoquinate
- Metronidazole
- Tinidazole
- Imidocarb
- Miltefosine
- Allopurinol
- Sodium stibogluconate
57
Antiviral drugs
- Acyclovir
- Ganciclovir
- Famciclovir
- Idocuridine
- Trifluridine
- Interferon-alfa and omega
- Zidovudin
- Amantadine
- Oseltamivir
- Vidarabine
58
Beta-lactame antibiotics
- penicillin
_Narrow spectrum penicillins:_
- Benzylpenicillin Na, K
- Procaine-, Benzathine benzylpenicillin
- Phenoxymethylpenicillin
_Penicillinase resistant penicillins:_
- oxacillin, cloxacillin, dicloxacillin, flucloxacillin
_Broad spectrum antibiotics:_
- Amoxicillin, Ampicillin
_Antipseudomonal penicillins:_
- Ticarcillin, Piperacillin
59
Beta-lactame antibiotics
- Beta-lactamase inhibitors:
- clavulanic acid
- sulbactam
- tazobactam
60
Beta-lactame antibiotics
- Cefalosporins
_1st. generation:_
- Cefazolin, Cefapirin, Cefadroxil, Cefalexin
_2nd. generation:_
- Cefuroxime
_3rd. generation:_
- Ceftiofur, Cefovecin, Ceftriaxone, Cefotaxime, Ceftazidim, Cefoperazon
_4th. generation:_
- Cefquinome
61
Beta-lactame antibiotics
- Carbapenems and Monobactams
_Carbapenems:_
- Imipenem, Meropenem
_Monobactams:_
- Aztreonam, Tigemonam
62
Aminoglycosides
- Streptomycin
- Neomycin
- Kanamycin
- Gentamycin
- Tobramycin
- Amikacin
- Apramycin
- Spectinomycin
63
Tetracyclines
Naturally-occuring:
* Oxytetracycline, Chlortetracycline
Semisyntehtic:
* Doxycyline, Minocycline
Short acting:
* tetracycline, ocytetracycline, chlorotetracycline
Intermediate acting:
* Demetetracycline
Long acting:
* Doxycycline, Minocycline
64
Macrolides
- Erythromycin
- Azithromycin
- Clarithromycin
- Spiramycin
- Tylosin
- Tylvalosin
- Tilmicosin
- Tulathromycin
- Gamitrhomycin
- Tildipirosin
65
Lincosamides
- Lincomycin
- Clindamycin
66
Pleuromutilins
- Tiamulin
- Valnemulin
67
Phenicols
- Chloramfenikol
- Florfenicol
- Thiamphenicol
68
Peptide ab
_Polypeptide ab_
- Bacitracin, Polymyxin B
_Glycopeptide ab_
- Vancomycin, Teicoplanin
69
Rifamiycins, Mupirocin, Fosfomycin
_Rifamiycins_
- Rifampin (rifampicin)
_Mupirocin_
- Mupirocin
_Fosfomycin_
- Fosfomycin
70
Sulphonamides
- Sulfadimidine
- Sulfadiazine
- Sulfachlorpyridazine
- Sulfachlorpyrazine
- Sulfamethoxazole
- Sulfadoxine
- Sulfaquinoxaline
- Sulfasalazine
71
Diaminopyrimidines
- Trimethoprim, Diaveridine, Pirimethamine, Omethropin, Aditoprim, Baquiloprim
72
Fluoroquinolones
_1st. generation:_
- Nalidixic acid
_2nd. generation:_
- Flumequine, Norfloxacin, Ciprofloxacin, Enrofloxacin, Danofloxacin, Difloxacin, Marbofloxacin
_3rd. generation:_
- Levofloxacin, Sparfloxacin
_4th. generation:_
- Pradofloxacin, Moxifloxacin
73
Nitrofuranes
- Nitrofurantoin
- Furazolidone
74
Nitroimidazoles
- Metronidazole
- Ronidazole
- Tinidazole
75
Uterus stimulants
- Oxytocin
* Carbetocin
- Ergot alkaloids
* Ergotoxin
* ERgotamine
* Ergometrine
- Prostaglandins
* Etiproston
* Luprostiol
* Dinoprost
76
Uterus relaxants
- B2-adrenoceptor agonsts
* Isoxuprine: B2-agonist, A1-antagonist
* Clenbuterol
* Terbutaline
* Vetrabutin
- Antispasmodics
- Phenotiazines
* Praquamezine
- Anticholinergics
* Denaverine
77
Pharmacology of anemia
- Erythropotein
* Epotein-alpha
* Derbepoetin
- Irondeficiency anemia
* Iron supplement PO
* Iron supplement IM: Iron Dextrane
78