Final Review Blocks 1-3 Flashcards

(344 cards)

1
Q

Norepinephrine

A

Mixed Agonist (Adrenergic)

  • A1, A2, and B1
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2
Q

Epinephrine

A

Mixed Agonist (Adrenergic)

  • A1, A2, B1, B2
  • low doses = B1 and B2, high doses = A1
  • treat acute anaphylaxis or cardiac arrest
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3
Q

Cocaine

A

NET, DAT, SERT Inhibitor (Adrenergic)

  • vasoconstriction, MI, stroke, death
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4
Q

Methylphenidate

A

NET, DAT Inhibitor (Adrenergic)

  • ADHD and narcolepsy tx
  • anorexia, jitters, poor growth, priapism
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5
Q

Atomoxetine

A

NET Inhibitor (Adrenergic)

  • ADHD tx
  • low abuse potential because non-stimulant
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6
Q

Ephedrine / Pseudoephedrine

A

Indirect Sympathomimetic (Adrenergic)

  • increase BP and HR
  • don’t use with MAOi
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7
Q

Amphetamine / Methamphetamine

A

Indirect Sympathomimetic (Adrenergic)

  • 1st line for ADHD in low doses
  • jitters, poor growth, anorexia, addictive
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8
Q

Phenylephrine

A

A1 Agonist (Adrenergic)

  • vasoconstriction
  • used for decongestant, hemorrhoids, mydriasis
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9
Q

Clonidine

A

A2 Agonist (Adrenergic)

  • treat HTN, ADHD, neuropathic pain
  • causes hypotension, sedation, dry mouth
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10
Q

Phenoxybenzamine

A

Nonselective Alpha Antagonist (Adrenergic)

  • non-competitive and irreversible
  • A1 and A2 antagonist
  • pheochromocytoma tx
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11
Q

Phentolamine

A

Nonselective Alpha Antagonist (Adrenergic)

  • competitive and reversible
  • A1 and A2 antagonist
  • pheochromocytoma tx
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12
Q

Prazosin

A

A1 Antagonist (Adrenergic)

  • decreases peripheral vascular resistance
  • treats HTN, BPH, Raynaud’s
  • “first dose phenomenon” = hypotension and syncope with first dose
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13
Q

Tamsulosin

A

A1 Antagonist (Adrenergic)

  • decreases peripheral vascular resistance, more selective for prostatic urethra
  • treats BPH primarily
  • “first dose phenomenon” = hypotension and syncope with first dose
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14
Q

Dobutamine

A

B1 Agonist (Adrenergic)

  • cardiac stimulation and renin release
  • used for cardiac failure
  • dysrhythmias
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15
Q

Albuterol

A

B2 Agonist (Adrenergic)

  • Short acting
  • Asthma and COPD tx
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16
Q

Terbutaline

A

B2 Agonist (Adrenergic)

  • Short acting
  • Asthma and COPD tx
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17
Q

Salmeterol

A

B2 Agonist (Adrenergic)

  • long acting
  • persistent asthma and COPD
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18
Q

Mirabegron

A

B3 Agonist (Adrenergic)

  • OAB tx
  • slow onset, can cause HTN
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19
Q

Esmolol

A

B1 Selective Antagonist (Adrenergic)

  • tx for HTN, angina, arrhythmia, ischemia
  • also used for intraoperative HTN
  • rebound HTN = taper dose
  • bronchoconstriction, bradycardia, CNS effects
  • short half life
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20
Q

Metoprolol

A

B1 Selective Antagonist (Adrenergic)

  • tx for HTN, angina, arrhythmia, ischemia
  • also used for intraoperative HTN
  • rebound HTN = taper dose
  • bronchoconstriction, bradycardia, CNS effects
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21
Q

Propanolol

A

B1/B2 Nonselective Antagonist (Adrenergic)

  • tx for HTN, angina, arrhythmia, ischemia
  • migraine prophylaxis
  • caution with asthma due to B2 effects
  • rebound HTN = taper dose
  • bronchoconstriction, bradycardia, CNS effects
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22
Q

Timolol

A

B1/B2 Nonselective Antagonist (Adrenergic)

  • decreases aqueous humor production and reduces intraocular pressure
  • bronchoconstriction, bradycardia, CNS effects
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23
Q

Labetalol

A

A/B Nonselective Antagonist (Adrenergic)

  • Mostly B1 and B2 antagonism with some A1
  • HTN tx and for Hypertensive Emergency
  • rebound HTN = taper dose
  • bronchoconstriction, bradycardia, CNS effects
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24
Q

Carvedilol

A

A/B Nonselective Antagonist (Adrenergic)

  • 10:1 B1 and B2 to A1 antagonism
  • HTN, HF
  • rebound HTN = taper dose
  • bronchoconstriction, bradycardia, CNS effects
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25
Methacholine
Muscarinic Agonist (Cholinergic)
26
Pilocarpine
Muscarinic Agonist (Cholinergic) - open angle glaucoma tx - DUMBBELS - sweating
27
Bethanecol
Muscarinic Agonist (Cholinergic) - GI stimulation / inactive bowel - urinary retention tx - DUMBBELS and sweating
28
Atropine
Muscarinic Antagonist (Cholinergic) - mydriasis tx - antidote for muscarinic toxicity, can cross BBB - DUMBBELS and sweating
29
Scopolamine
Muscarinic Antagonist (Cholinergic) - motion sickness tx
30
Ipratropium
Muscarinic Antagonist (Cholinergic) - asthma and COPD tx
31
Glycopyrrolate
Muscarinic Antagonist (Cholinergic) - used prep to decrease secretions and gastric acidity
32
Darifenacin
Muscarinic Antagonist (Cholinergic) - M3 selective antagonist - treats OAB
33
Benztropine
Muscarinic Antagonist (Cholinergic) - PSNS symptoms, including confusion - AVOID IN ELDERLY AND COGNITIVELY IMPAIRED - can treat Parkinson's and extrapyramidal symptoms
34
Nicotine
Nicotinic Agent (Cholinergic) - used for smoking cessation - can develop tolerance or dependence
35
Varenicline
Nicotinic Agent (Cholinergic) - partial agonist for smoking cessation - can cause depression and suicidal ideation
36
Rocuronium
Nicotinic NMJ Antagonist (Cholinergic) - skeletal muscle relaxer, useful in intubation - prolonged paralysis can occur
37
Succinylcholine
Depolarizing NMJ Blockade (Cholinergic) - activates nicotinic receptor before blocking it - skeletal muscle relaxation during anesthesia, useful for intubation - muscle soreness (potential hyperkalemia), malignant hypothermia
38
Donepezil
Acetylcholinesterase Inhibitor (Cholinergic) - used for Alzheimer's, improves cognition
39
Pyridostigmine
Acetylcholinesterase Inhibitor (Cholinergic) - reversible carbamate substrate - does NOT cross BBB
40
Neostigmine
Acetylcholinesterase Inhibitor (Cholinergic) - reversible carbamate substrate - does NOT cross BBB - causes contraction of denervated skeletal muscle
41
Physostigmine
Acetylcholinesterase Inhibitor (Cholinergic) - Readily crosses the BBB - DUMBBELS side effects - can treat atropine overdose
42
Edrophonium
Acetylcholinesterase Inhibitor (Cholinergic) - reversible substrate - very short acting, used for myasthenia gravis
43
Pralidoxome (2-PAM)
Acetylcholinesterase Poisoning Antidote (Cholinergic) - does not cross BBB - treats organophosphate toxicity, reverses NMJ blockade paralysis
44
Atropine
Acetylcholinesterase Poisoning Antidote (Cholinergic) - Crosses BBB - treats organophosphate toxicity, reverses NMJ blockade paralysis
45
Sarin
Toxic Organophosphate (Cholinergic) - nerve gas - DUMBBELS
46
Malathion
Toxic Organophosphate (Cholinergic) - insecticide - DUMBBELS
47
Amitriptyline
Tricyclic Antidepressant - NET / SERT inhibitor - also blocks muscarinic, A1, A2 - Causes coma, cardio toxicity, convulsions (3 Cs) - sexual dysfunction, serotonin syndrome with MAOi
48
Nortriptyline
Tricyclic Antidepressant - Primarily NET inhibitor - also blocks muscarinic, A1, A2 - Causes coma, cardio toxicity, convulsions (3 Cs) - sexual dysfunction, serotonin syndrome with MAOi
49
Imipramine
Tricyclic Antidepressant - NET / SERT inhibitor - also blocks muscarinic, A1, A2 - Causes coma, cardio toxicity, convulsions (3 Cs) - sexual dysfunction, serotonin syndrome with MAOi
50
Sertraline
SSRI - can cause GI issues, CNS issues, sexual dysfunction - can precipitate mania in bipolar pt - SSRI withdrawal: FLUSH - risk of serotonin syndrome with MAOi
51
Citalopram
SSRI - can cause GI issues, CNS issues, sexual dysfunction - can precipitate mania in bipolar pt - SSRI withdrawal: FLUSH - risk of serotonin syndrome with MAOi
52
Fluoxetine
SSRI - can cause GI issues, CNS issues, sexual dysfunction - can precipitate mania in bipolar pt - SSRI withdrawal: FLUSH - risk of serotonin syndrome with MAOi
53
Paroxetine
SSRI - can cause GI issues, CNS issues, sexual dysfunction - can precipitate mania in bipolar pt - SSRI withdrawal: FLUSH - risk of serotonin syndrome with MAOi
54
Escitalopram
SSRI - can cause GI issues, CNS issues, sexual dysfunction - can precipitate mania in bipolar pt - SSRI withdrawal: FLUSH - risk of serotonin syndrome with MAOi
55
Venlafaxine
SNRI (Serotonin-Norepinephrine) - dose dependent inhibition, same side effects as SSRI - Low: SERT - Mid: SERT/NET - High: SERT/NET/DAT
56
Duloxetine
SNRI (Serotonin-Norepinephrine) - selective NET/SERT inhibition, same side effects as SSRI
57
Bupropion
Atypical Antidepressant - weak inhibition of NET/DAT/SERT - nicotinic antagonist - NO SEXUAL DYSFUNCTION
58
Mirtazapine
Atypical Antidepressant - block A adrenergic and serotonin - increased appetite and weight gain = GOOD FOR ELDERLY - NO SEXUAL DYSFUNCTION
59
Trazodone
Serotonin Modulator - weak SERT inhibition - NO SEXUAL DYSFUNCTION - off label treatment for insomnia
60
Vilazodone
Serotonin Modulator - partial serotonin agonist - insomnia side effect - causes sexual dysfunction
61
St. John's Wart
Herbal Supplement (Antidepressant) - Hypericin --> MAO inhibitor - Hyperforin --> NET/DAT/SERT inhibitor
62
Lithium
Mood Stabilizer (Bipolar / Antipsychotic) - not safe in pregnancy - needs regular renal and thyroid monitoring
63
Valproic Acid
Antiepileptic - Mood Stabilizer (Bipolar / Antipsychotic) - prolongs Na channel inactivation and suppresses Ca influx - increases GABA - hepatotoxic - contraindicated in pregnancy
64
Lamotrigine
Antiepileptic - Mood Stabilizer (Bipolar / Antipsychotic) - inhibit glutamate release - CAUSES STEVEN-JOHNSON RASH - SAFE IN PREGNANCY
65
Haloperidol
High Potency Typical Antipsychotic (Bipolar / Antipsychotic) - blocks D2 receptors - frequent extrapyramidal effects, high risk of tardive dyskinesia - prolongs QT interval
66
Chlorpromazine
Low Potency Typical Antipsychotic (Bipolar / Antipsychotic) - also blocks muscarinic, histamine, A adrenergic receptors - rare extrapyrimidal effects, low risk of tardive dyskinesia
67
Clozapine
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - rare extrapyramidal effects
68
Aripiprazole
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - rare extrapyramidal effects - low incidence of weight gain
69
Olanzapine
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - rare extrapyramidal effects - SIGNIFICANT WEIGHT GAIN and sedation
70
Ziprasidone
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - rare extrapyramidal effects - PROLONGED QT INTERVAL
71
Quetiapine
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - rare extrapyramidal effects - weight gain and tachycardia - ABUSE POTENTIAL
72
Risperidone
Atypical Antipsychotic (Bipolar / Antipsychotic) - 1st line class for schizophrenia - block D2 and 5HT receptors - HIGHER extrapyramidal risk - PROLONGED QT INTERVAL - INCREASED PROLACTIN AND GYNECOMASTIA IN MALES
73
Midazolam
Short Acting Benzodiazepine (Anxiolytic) - positive allosteric modulator at GABAa - respiratory depression, impaired memory and cognitive function
74
Triazolam
Short Acting Benzodiazepine (Anxiolytic) - positive allosteric modulator at GABAa - respiratory depression, impaired memory and cognitive function
75
Alprazolam
Intermediate Acting Benzodiazepine (Anxiolytic) - positive allosteric modulator at GABAa - respiratory depression, impaired memory and cognitive function
76
Lorazepam
Intermediate Acting Benzodiazepine (Anxiolytic) - positive allosteric modulator at GABAa - respiratory depression, impaired memory and cognitive function
77
Clonazepam
Long Acting Benzodiazepine (Anxiolytic) - respiratory depression, impaired memory and cognitive function
78
Diazepam
Long Acting Benzodiazepine (Anxiolytic) - respiratory depression, impaired memory and cognitive function - treat alcohol withdrawal and bento withdrawal
79
Buspirone
Non-GABA Anxiolytic - serotonin partial agonist, D2 antagonist
80
Flumazenil
Non-GABA Anxiolytic - GABAa antagonist - CAN INDUCE BENZO WITHDRAWAL OR SEIZURE - USED FOR BENZO REVERSAL
81
Zolpidem
Z-Drug (Anxiolytic) - GABAa agonist - for insomnia
82
Zaleplon
Z-Drug (Anxiolytic) - GABAa positive allosteric modulator - for insomnia - causes aggression and hallucination so NO IN ELEDERLY
83
Eszoplicone
Z-Drug (Anxiolytic) - GABAa agonist - for insomnia, CAN BE USED LONG TERM
84
Suvorexant
Sleep Drug (Anxiolytic) - orexin antagonist
85
Doxepin
Sleep Drug (Anxiolytic) - selective H1 antagonist at low doses, 5HT and D2 at higher doses - don't use with MAOi --> serotonin syndrome
86
Ramelteon
Sleep Drug (Anxiolytic) - melatonin agonist
87
Trazodone
Sleep Drug / Atypical Antidepressant (Anxiolytic) - increase serotonin, decrease histamine
88
Mirtazapine
Sleep Drug / Atypical Antidepressant (Anxiolytic) - increase serotonin, decrease histamine - good for elderly, hyperphagia and weight gain
89
Diphenhydramine
Sleep Drug / Atypical Antidepressant (Anxiolytic) - increase serotonin, decrease histamine - concern in elderly
90
Phenobarbital
Barbiturates (Anxiolytic) - long acting GABAa agonist - respiratory depression - high concentration doesn't require GABA binding
91
Pentobarbital
Barbiturates (Anxiolytic) - short acting GABAa agonist - respiratory depression - high concentration doesn't require GABA binding
92
Propofol
GABA Associated Anxiolytic - GABAa agonist - anesthetic
93
Baclofen
GABA Associated Anxiolytic - ONLY GABAb agonist
94
Chloral Hydrate
GABA Associated Anxiolytic - sedative, alleviates insomnia - incapacitates individuals in prison
95
Phenytoin
Na+ Channel Anti-Epileptic - arrhythmia - teratogenic
96
Carbamazepine
Na+ Channel Anti-Epileptic - bone marrow suppression - neural tube defects in pregnancy
97
Lacosamide
Na+ Channel Anti-Epileptic - well tolerated
98
Lamotrigine
Na+ Channel Anti-Epileptic - epilepsy, bipolar, or depression - inhibits glutamate as well - CAUSES STEVENS-JOHNSON RASH - SAFE IN PREGNANCY
99
Topiramate
Na+ Channel Anti-Epileptic - CAUSES WEIGHT LOSS - metabolic acidosis and cleft palate (teratogenic)
100
Ethosuximide
Ca2+ Channel Inhibitor Anti-Epileptic - very safe and effective
101
Valproic Acid
Ca2+ Channel Inhibitor Anti-Epileptic - hair loss, bruising, liver injury - TERATOGENIC - SPINA BIFIDA
102
Gabapentin
Ca2+ Channel Anti-Epileptic - inhibits glutamate - weight gain - can cause respiratory depression, especially with opioids or benzos
103
Diazepam Lorazepam
Benzodiazepines / Anti-Epileptics - positive allosteric modulators at GABAa - for acute seizure attacks - can develop tolerance
104
Phenobarbital
Barbiturate / Anti-Epileptic - GABA agonist at high doses - 1st line for neonatal seizures
105
Levetiracetam
SV2A Modulator (Anti-Epileptic) - well tolerated broad spectrum anti-epileptic
106
Carbidopa / Levodopa
Dopamine Precursors (Parkinson's) - L-dopa passes BBB to increase DA - Carbidopa reduces conversion of L-Dopa to DA - used for basically all Parkinson's pts
107
Sinemet
Dopamine Precursors (Parkinson's) - brand name for carbidopa / levodopa
108
Entacapone
L-Dopa/DA Degradation Inhibitor (Parkinson's) - COMT inhibitor - causes orthostatic hypotension
109
Rasagiline
L-Dopa/DA Degradation Inhibitor (Parkinson's) - MAO-B inhibitor - may be NEUROPROTECTIVE
110
Stalevo
L-Dopa/DA Degradation Inhibitor (Parkinson's) - Entacapone + Carbidopa / Levodopa
111
Pramipexole
DA Receptor Agonist (Parkinson's) - for younger pt, hallucinations in older pt
112
Rotigotine
DA Receptor Agonist (Parkinson's) - once daily patch - can cause hyperhidrosis
113
Bromocriptine
DA Receptor Agonist (Parkinson's) - also 5HT inhibitor and glutamate inhibitor - exacerbates/causes heart disease
114
Benztropine
Anticholinergic - ACh Inhibitor (Parkinson's) - inhibits DAT and ACh (an excitatory NT) - can cause tachycardia or psychosis
115
Lidocaine
Local Anesthetic - Amine - degraded by cytochrome P450 - hepatotoxic
116
Bupivacaine
Local Anesthetic - Amine - degraded by cytochrome P450 - hepatotoxic
117
Benzocaine
Local Anesthetic - Ester - degraded by plasma esterases - more likely to cause allergic reactions
118
Cocaine
Local Anesthetic - Ester - degraded by plasma esterases - more likely to cause allergic reactions
119
Propofol
General Anesthetic - enhances GABAa receptor - induction and maintenance - antiemetic
120
Ketamine
General Anesthetic - NMDA receptor antagonist - AWAKE AMNESIA - bronchodilator that can cause bronchospasm
121
Midazolam
General Anesthetic - positive allosteric modulator at GABAa - shortest half life
122
Methohexital
General Anesthetic - positive allosteric modulator at GABAa
123
Etomidate
General Anesthetic - enhances GABAa - CARDIOSTABLE, USE IN PT AT RISK FOR HYPOTENSION - significant nausea and vomiting
124
Flumazenil
Used to shorten recovery from anesthesia with benzodiazepines
125
Isoflurane
General Anesthetic - Inhaled (Volatile) - pungent odor - tachycardia and malignant hypothermia
126
Sevoflurane
General Anesthetic - Inhaled (Volatile) - induction and maintenance - NOT IRRITATING TO AIRWAYS - malignant hypothermia
127
Desflurane
General Anesthetic - Inhaled (Volatile) - used to maintain anesthesia - NO INDUCTION DUE TO AIRWAY IRRITATION - tachycardia and malignant hypothermia
128
Nitrous Oxide
General Anesthetic - Inhaled (Volatile) - weak anesthetic, used as adjunct - can cause diffusion hypoxia, need to give 100% O2 at end of procedure - IMPOTENT --> MAC = 105%
129
Morphine
Opioid - Mu agonist - can cause respiratory depression and constipation
130
Hydromorphine
Morphine-Like Opioid - Mu agonist - can cause respiratory depression and constipation - preferred in renal pt
131
Fentanyl
Morphine-Like Opioid - Mu agonist - can cause respiratory depression and constipation - no histamine release
132
Heroin
Morphine-Like Opioid - Mu agonist - can cause respiratory depression and constipation
133
Codeine
Opioid - Mu agonist - can cause respiratory depression and constipation - metabolized by CYP2D6 - no patients <18 years old
134
Oxycodone
Codeine-Like Opioid - Mu agonist - can cause respiratory depression and constipation - COMBINED WITH ACETAMINOPHEN = POSSIBLE ACETAMINOPHEN TOXICITY
135
Hydrocodone
Codeine-Like Opioid - Mu agonist - can cause respiratory depression and constipation - COMBINED WITH ACETAMINOPHEN = POSSIBLE ACETAMINOPHEN TOXICITY
136
Tramadol
Opioid - Mu agonist - NET/SERT inhibitor - LOW RISK of respiratory depression, constipation, or abuse - can cause serotonin syndrome
137
Pentazocine
Opioid - Kappa agonist, Mu antagonist - causes dysphoria, increase HR and BP
138
Methadone
Opioid - Mu agonist, NMDA antagonist, NET/DAT/SERT inhibitor - risk of overdose - prolonged QT interval and arrhythmia
139
Buprenorphine
Opioid
140
Naloxone
Opioid Receptor Antagonist - IV admin - causes respiratory depression - can cause opioid relapses in higher doses
141
Naltrexone
Opioid Receptor Antagonist - oral admin - treats chronic alcoholism
142
Methylnaltrexone
Opioid Receptor Antagonist - doesn't cross the BBB
143
Pregabalin
Anticonvulsant / Pain Management
144
Gabapentin
Anticonvulsant / Pain Management
145
Acyclovir
Anti-Herpes Virus (Antiviral)
146
Ganciclovir
Anti-Herpes Virus (Antiviral)
147
Valacyclovir
Anti-Herpes Virus (Antiviral)
148
Foscarnet
Anti-Herpes Virus (Antiviral)
149
Oseltamivir
Anti-Influenza (Antiviral)
150
Zanamivir
Anti-Influenza (Antiviral)
151
Sofosbuvir
Anti-Hep C (Antiviral)
152
Velpatasvir
Anti-Hep C (Antiviral)
153
Remdesivir
Anti-Sars-CoV-2 (Antiviral)
154
Nirmatrelvir / Ritonavir
Anti-Sars-CoV-2 (Antiviral)
155
Zidovudine (AZT)
Anti-Retroviral (NRTI) [Antiviral]
156
Abacavir (ABC)
Anti-Retroviral (NRTI) [Antiviral]
157
Tenofovir (TDF)
Anti-Retroviral (NRTI) [Antiviral]
158
Nevirapine
Anti-Retroviral (NNRTI) [Antiviral]
159
Rifampicin
Anti-Retroviral (NNRTI) [Antiviral]
160
Darunavir (DRV) + Ritonavir
Anti-Retroviral (Protease Inhibitor) [Antiviral]
161
Dolutegravir
Anti-Retroviral (Integrase Inhibitor) [Antiviral]
162
Penicillin G / V
Beta Lactam (Antibiotic)
163
Amoxicillin
Beta Lactam (Antibiotic)
164
Amoxicillin / Clavulanic Acid
Beta Lactam (Antibiotic)
165
Cephalexin
Beta Lactam - Cephalosporin (Antibiotic)
166
Cefazolin
Beta Lactam - Cephalosporin (Antibiotic)
167
Ceftriaxone
Beta Lactam - Cephalosporin (Antibiotic)
168
Cefotaxime
Beta Lactam - Cephalosporin (Antibiotic)
169
Ceftazidime
Beta Lactam - Cephalosporin (Antibiotic)
170
Trimethoprim / Sulfamethoxazole (TMP/SMX)
Antifolate (Antibiotic) and Antifungal
171
Nitrofurantoin
UTI Drug (Antibiotic)
172
Ciprofloxacin
Fluoroquinolone (Antibiotic)
173
Levofloxacin
Fluoroquinolone (Antibiotic)
174
Chloramphenicol
Protein Synthesis Inhibitor (Antibiotic)
175
Clindamycin
Protein Synthesis Inhibitor (Antibiotic)
176
Azithromycin
Macrolide (Antibiotic)
177
Erythromycin
Macrolide (Antibiotic)
178
Doxycycline
Tetracycline (Antibiotic)
179
Gentamycin
Aminoglycoside (Antibiotic)
180
Metronidazole
Treatment Resistant (Antibiotic)
181
Vancomycin
Treatment Resistant (Antibiotic)
182
Linezolid
Treatment Resistant (Antibiotic)
183
Polymyxin B & E
Treatment Resistant (Antibiotic)
184
Isoniazid
Treatment Resistant (Antibiotic)
185
Rifampin
Treatment Resistant (Antibiotic)
186
Amphotericin B
Antifungal
187
Terbinafine
Antifungal
188
Fluconazole
Antifungal
189
Itraconazole
Antifungal
190
Medtronidazole
Anti-Parasitic
191
Chloroquine
Anti-Parasitic
192
Artemether-Lemefantrine
Anti-Parasitic
193
Artesunate
Anti-Parasitic
194
Sulfadiazine + Pyrimethamine
Anti-Parasitic
195
Sodium Stibogluconate
Anti-Parasitic
196
Nifurtimox
Anti-Parasitic
197
Mebendazole
Anti-Parasitic
198
Albendazole
Anti-Parasitic
199
Praziquantel
Anti-Parasitic
200
Amphetamine / Methamphetamine
Stimulant
201
Stimulant treatments
Benzodiazepines Haloperidol
202
Depressants
Benzodiazepines GHB Opioids Alcohol
203
Alcohol overuse treatment
Naltrexone
204
Depressant overdose treatments
Flumazenil (avoid in benzos) Naloxone Naltrexone (alcohol)
205
LSD
Hallucinogen - benzos for agitation, atypical antipsychotics for hallucination
206
PCP
Hallucinogen - benzos for agitation, atypical antipsychotics for hallucination
207
Ketamine
Hallucinogen - benzos for agitation, atypical antipsychotics for hallucination
208
Marijuana
Hallucinogen
209
Synthetic Cannabinoids (K2/Spice)
Hallucinogen - treat agitation or seizure with benzos
210
Addiction treatments
Methadone (long acting agonist) Buprenorphine (partial agonist to reduce withdrawal symptoms)
211
Quinidine
Sodium Channel Blocker (Antiarrhythmic) - Class 1A Antiarrhythmic
212
Procainamide
Sodium Channel Blocker (Antiarrhythmic) - Class 1A Antiarrhythmic
213
Lidocaine
Sodium Channel Blocker (Antiarrhythmic) - Class 1B Antiarrhythmic
214
Flecainide
Sodium Channel Blocker (Antiarrhythmic) - Class 1C Antiarrhythmic
215
Propanolol
Beta Blocker (Antiarrhythmic) - Class II Antiarrhythmic
216
Esmolol
Beta Blocker (Antiarrhythmic) - Class II Antiarrhythmic
217
Metoprolol
Beta Blocker (Antiarrhythmic) - Class II Antiarrhythmic Vasodilator
218
Carvedilol
Beta Blocker (Antiarrhythmic) - Class II Antiarrhythmic Vasodilator
219
Amiodarone
Potassium Channel Blocker (Antiarrhythmic) - Class III Antiarrhythmic
220
Verapamil
Calcium Channel Blocker (Antiarrhythmic) - Class IV Antiarrhythmic (Vasodilator and HTN) - Non-dihydropyridine
221
Diltiazem
Calcium Channel Blocker (Antiarrhythmic) - Class IV Antiarrhythmic (Vasodilator and HTN) - Non-dihydropyridine
222
Amlodipine
Calcium Channel Blocker (Vasodilator) - Dihydropyridine
223
Nifedipine
Calcium Channel Blocker (Vasodilator) (HTN) - Dihydropyridine
224
Adenosine
Class V Antiarrhythmic
225
Nitroglycerine
Nitrate (Vasodilator)
226
Isosorbide Dinitrate
Nitrate (Vasodilator)
227
Sildenafil
PDE Type 5 Inhibitor (Vasodilator)
228
Acetazolamide
Carbonic Anhydrase Inhibitor (Diuretic)
229
Furosemide
Loop Diuretic
230
Hydrochlorothiazide
Distal Tubule Diuretic
231
Amiloride
Sodium Channel Inhibitor (Potassium-Sparing Diuretic)
232
Spirinolactone
Aldosterone Receptor Antagonist (Potassium-Sparing Diuretic)
233
Digoxin
Digitalis Glycoside (Ionotropic) [Heart Failure]
234
Dobutamine
Sympathomimetic Amine (Ionotropic) [Heart Failure] - for acute heart failure
235
Milrinone
Phosphodiesterase-3 Inhibitor (Ionotropic) [Heart Failure] - for acute heart failure
236
Captopril
ACE Inhibitor (Heart Failure / HTN)
237
Lisinopril
ACE Inhibitor (Heart Failure / HTN)
238
Losartan
ARB (Heart Failure / HTN)
239
Sacubitril / Valsartan
ARNI (Heart Failure)
240
Other Drugs for Heart Failure
Beta blockers - Metoprolol - Bisoprolol - Carvedilol Aldosterone Receptor Antagonist - Spirinolactone
241
Aspirin
COX Inhibitor (Antiplatelet and NSAID)
242
Dipyridamole
cAMP-Altering Antiplatelet
243
Clopidogrel
ADP Receptor Inhibitor (Antiplatelet)
244
Prasugrel
ADP Receptor Inhibitor (Antiplatelet)
245
Ticagrelor
ADP Receptor Inhibitor (Antiplatelet)
246
Eptifibatide
Glycoprotein IIb/IIIa Receptor Inhibitor (Antiplatelet)
247
Vorapaxar
Protease-Activated Receptor Antagonist (Antiplatelet)
248
Heparin
Clotting Factor Inhibitor (Anticoagulant)
249
Protamine Sulfate
Heparin Antidote
250
Enoxparin
Clotting Factor Inhibitor (Anticoagulant) - low molecular weight heparin
251
Fondaparinox
Clotting Factor Inhibitor (Anticoagulant)
252
Rivaroxaban
Direct Factor X Inhibitor (Anticoagulant)
253
Apixaban
Direct Factor X Inhibitor (Anticoagulant)
254
Andexanet Alfa
Direct Factor X Inhibitor antidote
255
Warfarin
Coumarin (Anticoagulant)
256
Vitamin K
Warfarin antidote
257
Prothrombin complex concentrates
Warfarin antidote
258
Dabigatran
Direct Thrombin Inhibitor (Anticoagulant and Antiplatelet)
259
Idarucizumab
Dabigatran (Direct Thrombin Inhibitor) antidote
260
Alteplase
Tissue Plasminogen Activator (Fibrinolytic)
261
Tenecteplase
Tissue Plasminogen Activator (Fibrinolytic)
262
Aminocaproic Acid
Tissue Plasminogen Activator (Fibrinolytic)
263
Lovastatin
HMG-CoA Inhibitor / Statin
264
Atorvastatin
HMG-CoA Inhibitor / Statin
265
Rosuvastatin
HMG-CoA Inhibitor / Statin
266
Cholestyramine
Bile Acid Resin (Lipid Lowering)
267
Alirocumab
PCSK9 Inhibitor (Lipid Lowering)
268
Ezetimibe
Cholesterol Absorption Inhibitor
269
Niacin
Nicotinic Acid (Lipid Lowering)
270
Gemfibrozil
Fibrate (Lipid Lowering)
271
Fenofibrate
Fibrate (Lipid Lowering)
272
Icosapent Ethyl (Eicosapentaenoic Acid)
Omega-3 Fatty Acid (Lipid Lowering)
273
First Line Hypertension Drugs
Diuretics - HCTZ - Chlorthalidone ACE Inhibitor - Captopril ARB - Losartan Ca Channel Blocker - Verapimil - Diltiazem - Nifedipine
274
Hydralazine
Direct Vasodilator (HTN)
275
Nitroprusside
Direct Vasodilator (HTN)
276
Aliskiren
Renin Inhibitor (HTN)
277
Secondary HTN agents
Beta Blockers - Propanolol - Metoprolol - Labetalol A2 Agonist - Clonidine Direct Vasodilators - Hydralazine - Nitroprusside Renin Inhibitor - Aliskiren
278
Clomiphene
Estrogen Receptor Antagonist (Fertility)
279
Gonadorelin
GnRH (Fertility)
280
Menotropin
Gonadotropin (Fertility)
281
Urofollitropin
Gonadotropin (Fertility)
282
hCG
Gonadotropin (Fertility)
283
Estradiol
Estrogen Contraceptive
284
Estrone
Estrogen Contraceptive
285
Ethinyl Estradiol
Estrogen Contraceptive Estrogen HRT
286
Mestranol
Estrogen Contraceptive Estrogen HRT
287
Medroxyprogesterone
Progestin Contraceptive Progestin HRT
288
Norethindrone
Progestin Contraceptive
289
Drospirenone
Progestin Contraceptive
290
Norgestrel
Progestin Contraceptive
291
Levonorgestrel
Progestin Contraceptive Progestin HRT
292
Levonorgestrel + ethinyl estradiol
Post Coital Contraceptive
293
Mifepristone + Misoprostol
Elective Abortion
294
Conjugated Estrogens
Estrogen HRT
295
Tamoxifen
Selective Estrogen Receptor Modulator (SERM) [HRT and Breast Cancer]
296
Raloxifene
Selective Estrogen Receptor Modulator (SERM) [HRT and Breast Cancer]
297
Anastrozole
Aromatase Inhibitor (HRT and Breast Cancer)
298
Letrozole
Aromatase Inhibitor (HRT and Breast Cancer)
299
Testosterone
Androgen
300
Dihydrotestosterone
Androgen
301
Oxandrolone
Androgen
302
Danazol
Androgen
303
Finasteride
5a- Reductase Inhibitor (BPH)
304
Leuprolide
GnRH Agonist (Prostate Cancer)
305
Degarelix
GnRH Antagonist (Prostate Cancer)
306
Flutamide
Androgen Receptor Antagonist (Prostate Cancer)
307
Bicalutamide
Androgen Receptor Antagonist (Prostate Cancer)
308
Lispro
Rapid Acting Insulin (Diabetes)
309
Aspart
Rapid Acting Insulin (Diabetes)
310
Glulisine
Rapid Acting Insulin (Diabetes)
311
Regular Insulin
Short Acting Insulin (Diabetes)
312
NPH
Intermediate Acting Insulin (Diabetes)
313
Glargine
Long Acting Insulin (Diabetes)
314
Detemir
Long Acting Insulin (Diabetes)
315
Degludec
Long Acting Insulin (Diabetes)
316
Glyburide
Sulfonylurea (Diabetes)
317
Glimepiride
Sulfonylurea (Diabetes)
318
Glipizide
Sulfonylurea (Diabetes)
319
Metformin
Biguanide (Diabetes)
320
Pioglitazone
Thizolidinediones (TZD) [Diabetes]
321
Repaglinide
Meglitinide (Diabetes)
322
Exenatide
GLP-1 Agonist (Diabetes)
323
Sitagliptin
DPP-4 Inhibitor (Diabetes)
324
Canagliflozin
SGLT2 Inhibitor (Diabetes)
325
Acarbose
a-Glucosidase Inhibitor (Diabetes)
326
Plamlintide
Amylin Mimetic (Diabetes)
327
Colesevelem
Bile Acid Sequestrant (Diabetes)
328
Glucagon
Increases blood glucose levels
329
Levothyroxine (T4)
Hypothyroid Drug
330
Propylthiouracil
Hyperthyroid Drug
331
Methimazole
Hyperthyroid Drug
332
Potassium Iodide
Hyperthyroid Drug
333
Radioiodine
Hyperthyroid Drug
334
Adjunct Thyroid Treatments
1. Propanolol 2. Diltiazem 3. Rituximab
335
Calcitonin
Anti-Catabolic (Osteoporosis
336
Alendronate
Bisphosphonate (Anti-Catabolic) [Osteoporosis]
337
Zolendronate
Bisphosphonate (Anti-Catabolic) [Osteoporosis]
338
Denosumab
RANK Ligand Inhibitor (Anti-Catabolic) [Osteoporosis]
339
Raloxifene
SERM (Anti-Catabolic) [Osteoporosis]
340
Teriparatide (Recombinant Parathyroid Hormone)
Anabolic Therapy (Osteoporosis)
341
Cinacalcet
Antihypercalcemic Therapy
342
Calcitriol
Antihypocalcemic Therapy
343
Calcium Gluconate
Antihypocalcemic Therapy - IV admin
344
Calcium Citrate
Antihypocalcemic Therapy - Oral admin