Nicotinic receptor Flashcards
(31 cards)
Trimethaphan
Antagonist Nn receptor
Hexamethonium
Antagonist Nn receptor
Mecamylamine
Antagonist Nr receptor
Tubocurarine
Antagonists Nm Receptor
Atracurium
Antagonists Nm Receptor
Carbachol (CCh)
Nm Agonist receptor.
Suxamethonium
Nm Receptor Agonist.
Acetylcholine
Direct Acting Receptor Agonist (Muscarinic)
Bethanechol
Direct Acting Receptor Agonist (Muscarinic)
Carbachol
Direct Acting Receptor Agonist (Muscarinic)
Pilocarpine
Direct Acting Receptor Agonist (Muscarinic)
Nicotine
Nicotinic Agonist
Varenicline
Nicotinic Agonist
Physostigmine (Natural)
Indirect-acting (Cholinesterase inhibitors)
Neostigmine
Indirect-acting (Cholinesterase inhibitors)
Pyridostigmine
Indirect-acting (Cholinesterase inhibitors)
Donepezil
Indirect-acting (Cholinesterase inhibitors)
Rivastigmine
Indirect-acting (Cholinesterase inhibitors)
Edrophonium
Indirect-acting (Cholinesterase inhibitors) use in Tensilon Test
Organophosphorus _
Echothiophate, Parathion, Malathion (Insecticide and Pesticides)
Irreversible Anticholinesterases inhibitor
Tabun Nerve gas in war
Indirect-acting (Cholinesterase inhibitors) Irreversible
Sarin Nerve gas in war
Indirect-acting (Cholinesterase inhibitors) Irreversible
Soman Nerve Gas in war
Indirect-acting (Cholinesterase inhibitors) Irreversible
Carbamate Esters:
Carbaryl and Propoxur
Indirect-acting (Cholinesterase inhibitors) Irreversible