Sedative-Hypnotics Flashcards
Alprazolam
Benzodiazepines
shortest acting
Chlordiazepoxide
Benzodiazepines
Clonazepam
Benzodiazepines
second line for absence seizures
Clorazepate
Benzodiazepines
Diazepam
Benzodiazepines
Estazolam
Benzodiazepines
Flurazepam
Benzodiazepines
longest acting
Lorazepam
Benzodiazepines
conjugated and excreted via kidney(LOT)
Midazolam
Benzodiazepines
45 min. anterograde amnesia
Oxazepam
Benzodiazepines
conjugated and excreted via kidney(LOT)
Quazepam
Benzodiazepines
Temazepam
Benzodiazepines
conjugated and excreted via kidney(LOT)
maintains sleep
Triazolam
Benzodiazepines
puts you to sleep
Flumazenil
Benzodiazepine Antagonist
Amobarbital
Barbiturates (most hepatic metabolism)
Mephobarbital
Barbiturates
Phenobarbital
Barbiturates
urine alkalization can increase elimination rate
Pentobarbital
Barbiturates
Secobarbital
Barbiturates
Eszopiclone (Lunesta)
Sedative-Hypnotic Drug
good for sleep aid (CYP3A4) increase sleep time
Buspirone
Sedative-Hypnotic Drug
Chloral hydrate
Sedative-Hypnotic Drug
Zaleplon
Sedative-Hypnotic Drug
good for sleep aid (CYP3A4)
Zolpidem (Ambien)
Sedative-Hypnotic Drug
sleep driving, and others
good for sleep aid (CYP3A4)