Semester 1 drug list Flashcards

1
Q

A1. Pharmacodynamics I

A

(no specific drugs to be known)

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2
Q

A2. Pharmacodynamics II

A

(no specific drugs to be known)

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3
Q

A3. Drug absorption, distribution and bioavailability. Membrane transport mechanisms.

A

(no specific drugs to be known)

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4
Q

A4. Drug biotransformation and excretion, linear and non-linear kinetics. Enzyme inhibitors and enzyme inducers. Clearance, half life, loading and maintenance dose. Pharmacokinetic drug interactions.

A

(no specific drugs to be known)

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5
Q

A5. Drugs acting on gastrointestinal and urogenital smooth muscles. Drugs influencing uterine function

A

papaverine, drotaverine, butylscopolamine, misoprostol, oxytocin, ergotamine, terbutaline, atosiban, Magnesium, ethanol, solifenacin, oxybutinine, tamsulosin

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6
Q

A6. Histamine and antihistamines

A

promethazine, diphenhydramine, (levo)cetirizine, (des)loratadine, dimetinden, fexofenadin

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7
Q

A7. Glucocorticoids for oral and parenteral use

A

hydrocortisone, prednisolone, methylprednisolone, dexamethasone, triamcinolone

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8
Q

A8. Mineralocorticoids. Topically applied glucocorticoids. Adrenocortical antagonists, inhibitors of corticosteroid synthesis

A

fludrocortisone, fluocinolone, mometazone, budesonide, fluticasone, metyrapone

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9
Q

A9. Androgens, anabolic steroids, antiandrogens. Agents affecting the sexual activity

A

testosterone-undecanoate, bicalutamide, finasteride, goserelin, degarelix, sildenafil, nandrolone

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10
Q

A10. Estrogens and antiestrogens

A

ethinylestradiol, estradiol, clomifen, tamoxifen, raloxifen, anastrozole, goserelin, degarelix

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11
Q

A11. Progestins and antiprogestins

A

medroxyprogesterone-acetate, drospirenone, norethisterone, levonorgestrel, desogestrel, cyproterone-acetate, mifepristone, ulipristal acetate

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12
Q

A12. Contraceptives

A

ethinyestradiol + levonorgestrel, medroxyprogesterone-acetate, levonorgestrel, desogestrel

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13
Q

A13. Thyroid and antithyroid drugs. Pituitary hormones. Hypothalamic hormones, hormone analogues and antagonists

A

levothyroxin, thiamazole (methimazole), propylthiouracil, iodine, octreotide, bromocriptine, desmopressin, oxytocin

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14
Q

A14. Pancreatic hormones and parenterally applied antidiabetic drugs

A

regular insulin, lispro insulin, aspart insulin, glargine insulin, isophan (NPH) insulin, liraglutide

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15
Q

A15. Oral antidiabetics

A

glipizide, glimepiride, repaglinide, metformin, vildagliptin, dapagliflozin, acarbose

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16
Q

A16. Agents affecting bone mineral homeostasis

A

cholecalciferol (vitamin D), teriparatide, raloxifen, zoledronate, alendronate, denosumab

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17
Q

A17. Drugs influencing blood coagulation I: Antiplatelet drugs

A

acetylsalicylic acid (aspirin), clopidogrel, prasugrel, ticagrelor, abciximab

18
Q

A18. Drugs influencing blood coagulation II: Anticoagulant drugs

A

heparin, dalteparin, bivalirudin, warfarin, dabigatran-etexilate, rivaroxaban, fondaparinux

19
Q

A19. Drugs influencing blood coagulation III: Fibrinolytic drugs. Drugs inhibiting bleeding

A

alteplase, reteplase, epsilon-amino-caproic-acid, vitamin K, epinephrine, fibrin foam

20
Q

A20. Agents used in anemia

A

iron hydroxide polymaltose, folic acid, vitamin B12, epoetin-alpha, filgrastim

21
Q

B1. Cholinergic transmission and its presynaptic modification

A

(no specific drugs to be known)

22
Q

B2. Adrenergic transmission and its presynaptic modification

A

(no specific drugs to be known)

23
Q

B3. Cholinomimetics

A

carbachol, pilocarpine, neostigmine, pyridostigmine, rivastigmine, edrophonium

24
Q

B4. Muscarinic receptor blocking drugs

A

atropine, scopolamine, butyl-scopolamine, ipratropium, procyclidine, solifenacin, cyclopentolate, tiotropium, oxybutinin

25
B5. catecholamines
epinephrine, norepinephrine, dopamine, isoprenaline, dobutamine
26
B6. Indirect sympathomimetics. Selective alpha-1 and alpha 2 agonists and drugs acting on the imidazoline receptors
ephedrine, phenylephrine, clonidine, rilmenidine, methyldopa, oxymetazoline
27
B7. alpha receptor antagonists
prazosin, doxazosin, tamsulozin, urapidil, carvedilol, phentolamine
28
B8. Beta receptor antagonists
propranolol, pindolol, carvedilol, timolol, sotalol, metoprolol, bisoprolol, nebivolol, esmolol
29
B9. Centrally acting skeletal muscle relaxants (spasmolytics). Dantrolene. Botulinum toxin
baclofen, tolperisone, diazepam, tizanidine, dantrolene, botulinum toxin
30
B10. Skeletal muscle relaxants acting on the neuromuscular junction
(cis)atracurium, mivacurium, pipecuronium, rocuronium, succynylcholine (suxamethonium)
31
B11. Selective-Beta-2 stimulants and other bronchodilators
salbutamol, terbutaline, fenoterol, salmeterol, formoterol, ipratropium, tiotropium, theophylline
32
B12. Antiinflammatory agents inhibiting bronchial inflammatory processes. Antitussive agents and expectorants
prednisolone, methylprednisolone, fluticasone, budesonide, montelukast, omalizumab, codein, butamirate, prenoxdiazine, acetylcysteine, bromhexine
33
B13. Positive inotropic drugs
digoxin, digitoxin, milrinone, levosimendan, dobutamine
34
B14. Drugs influencing cardiac electrophysiology
lidocaine, propafenone, esmolol, amiodarone, sotalol, verapamil, adenosine, digoxin, Magnesium
35
B15. Drugs acting on the renin-angiotensin-aldosterone system (RAAS)
enalapril, perindopril, ramipril, losartan, valsartan, valsartan-sacubitril, irbesartan, spironolactone, eplerenone, captopril
36
B16. Calcium channel blockers and other vasodilators
amlodipine, felodipine, nifedipine, nimodipine, verapamil, dihydralazine, bozentan, sildenafil
37
B17. Drugs influencing the oxygen demand and oxygen supply of the heart
nitroglycerin, isosorbid-mononitrate, trimetazidine, ivabradine, propranolol, pindolol, carvedilol, timolol, sotalol, metoprolol, bisoprolol, nebivolol, esmolol, amlodipine, felodipine, nifedipine, nimodipine, verapamil, dihydralazine
38
B18. Drugs improving microcirculation
vinpocetin, nicergoline, cilostazol, pentoxifylline, Calcium-dobesilate, sumatriptan, galcanezumab, cinnarazine, propranolol, verapamil, carbamazepine, valproate, imipramine
39
B19. Drugs affecting lipid metabolism
simvastatin, atorvastatin, rosuvastatin, ezetimib, fenofibrate, colesevelam
40
B20. Potassium excreting (wasting) diuretics
acetazolomide, hydrochlorothiazide, indapamide, furosemide, etacrynic acid
41
B21. Potassium sparing diuretics, ADH antagonists, osmotic diuretics
spironolactone, eplerenone, amiloride, tolvaptan, mannitol, glycerol