Adrenergic receptors Flashcards
(9 cards)
adrenergic receptor location
ANS effector organs
Noradrenaline
endogenous transmitter released from synapses
adrenaline
hormone from adrenal medulla
dopamine
NA precursor but endogenous transmitter in CNS
Alpha 1 adrenergic receptor
Gq linked
-Constricts SM except for Gastrointestinal tract
-causes glycogen-lysis (increase metabolism)
Alpha 2 adrenergic receptor
Gi linked
- relax gastrointestinal tract
-depresses further adrenergic and cholinergic releases
Beta 1 adrenergic receptor
Gs linked
-Has strong effect on increasing heart rate and contraction
Beta 2 adrenergic receptor
Gs linked
-relaxes most SM
-causes tremor and muscle mass/ contraction force
-inhibits histamine release
-stimulates further adrenergic release
Beta 3 adrenergic receptor
Gs linked
-relaxes bladder
-increase anabolic metabolism