Adrenergic Receptors Flashcards
(6 cards)
Alpha-1
1) blood vessels - vasoconstriction2) Pupillary dilator muscle - contraction (DILATES)3) Pilomotor smooth muscle - contraction (hairs)4) Prostate - contraction (alpha-1-A)5) Heart - increases force of contraction
Alpha-2
1) POST synaptic adrenoceptors - decreases SNS outflow (alpha-2-A)2) Platelets - aggregation3) PRE synaptic adrenergic & cholinergic nerve terminals - inhibition of transmitter release (alpha-2-A)4) Blood vessels - vasoconstriction (alpha-2-B)
Beta-1
1) Heart - increases HR, contractility, AV node conduction2) Kidney - increases renin release
Beta-2
1) Respiratory, uterine, blood vessels - relaxation (vasodilation)2) Skeletal muscle - potassium uptake3) Human liver - glycogenolysis (increases glucose)4) Heart - increases HR, contractility, AV node conduction
Beta-3
Fat cells - lipolysis
DA-1
Smooth muscle - dilates renal blood vessels