AINES Flashcards

1
Q

Historia

A

Leroux, Sauce blanco o salix alba, salicina

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2
Q

Clasificacion

A
Salicilatos
Pirazolonas
Anilina
Ac propionico
Fenamato (antranilico)
Ac acetico
Coxibes
Otros
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3
Q

Clasificacion salicilatos

A

Ac salicilico

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4
Q

Clasificacion pirazolonas

A

Dipirona o metamizol

Butazonas

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5
Q

Clasificacion anilinas

A

Acetaminofen

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6
Q

Clasificacion ac propionico

A

Naproxeno

Iburoprofen

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7
Q

Clasificacion fenamatos (antranilico)

A

Ac mefenamico

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8
Q

Clasificacion ac acetico

A
Diclofenaco
Indometacina
Piroxicam
Meloxicam
Ketorolaco
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9
Q

Clasificacion coxibes

A

Celecoxib

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10
Q

Clasificacion otros

A

Nimesulide

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11
Q

Vm corta menor 4 hr

A
Paracetamol
Diclofenaco
Iburoprofeno
Metamizol o Dipirona
Tolmetina
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12
Q

Via parenteral

A

IV: metamizol
IM: metamizol, diclofenaco

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13
Q

Distribucion

A

Proteinas 90%

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14
Q

Biotransformacion

A
Oxidacion
Hidrolisis
Glucoronico
Glicina
Sulfato
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15
Q

Excrecion

A

Renal

Biliar

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16
Q

Acciones salicilatos

A
Analgesico
Antii
Antipiretico
Antirreuma
Antiagregante
17
Q

Analgesicos

A
Salicilatos
Pirazolonas
Anilina
Fenamato
Coxibes
Nimesulide
18
Q

Antipireticos

A
Salicilatos
Pirazolona
Anilina
Propionico
Nimesulide
19
Q

Antiagregantes

A

Salicilatos

20
Q

Antirreumaticos

A
Salicilatos
Butazona
Propionico
Ac acetico
Coxibes
21
Q

Analgesicos antipireticos y antiinflamatorios

A

Nimesulida y salicilatos

22
Q

Para el cierre del ductus arterioso

A

Ac acetico (indometacina)

23
Q

Formacion de ac araquidonico a partr de

A

Fosfolipidos de membrana por fosfolipasa

24
Q

COX que es

A

Prostaglandin sintetasa

25
COX 2 selectivos
Celecoxib, meloxicam, nimesulide
26
Propiedad antipiretica
Metamizol sudor y vasodilatación | Acetaminofen centro termorregulador hipotalamo
27
Uricosuricos y antigotosos
Butazonas | Ac acetico
28
Acciones tromboxanos
Vasoconstricción | Agregante
29
Acciones prostaglandinas
Vasodilatador | Antiagregante
30
Antiespasmodicos
Pirazolona metamizol | Fenamato
31
Amenaza de parto prematuro
Ac acetico indometacina
32
Dosis Acetaminofen
40 mg/kg/ dia | Repartido en 3
33
Presentacion Acetaminofen
Gotas 100 Jarabe 120/5ml Suposit 300 Tabs 500 y 750
34
Salicilismo
``` Suicidio Sudoracion Hipernea Hipertermia Alucinaciones Convulsiones Coma ```
35
Tx salicilismo
``` Lavado Temperatura Liquidos Vit k Control Acido base Transfusion Dialisis ```