Autcoids Flashcards
Highly sedative anti histaminics
PRO METHA ZINE,
DI PHEN HYDRA MINE,
HYDROXY ZINE,
DOXE PIN,
DOXYL AMINE
Anti histaminic with transdermal patch
Diphenhydramine
Anti histaminics ,used in
Motion sickness,
Drug induced parkinson’s disease
Pronethazine,
Diphenhydramine
Anti histaminics which can also be used as local anaesthetic
Promethazine,
Diphenhydramine
Anti histaminics with maximum anti pruritic effect
Hydroxyzine
Anti histaminic which is also a tricyclic antidepressants
Doxepin
Antihistamine
DOC in morning sickness
Doxylamine
Moderately sedative antihistamine
Cycli zine,
Mecli zine,
Cinnari zine,
Cypro heptadine,
Pheni ramine
Antihistamine good in sea sickness
Cycli zine,
Mecli zine,
Cinnari zine
Antihistamine + anti serotonin
Cypro heptadine
Least sedative antihistamine
CHLOR pheni ramine,
Clemastine,
Tirolidine
DOC in Anaphylaxis
I/m adrenaline 0.5 ml of 1:1000
2nd gen antihistamine
Fexo fenadine,
Cetrizine,
Levo cetrizine,
Loratidine,
Rupatidine,
Banned 2nd gen antihistamine
Terfinadine,
Astemizole
2nd gen antihistamine also PAF inhibitor
Rupatidine
Topical 2nd gen antihistamine
ALOKA
A- Aze lastine
L- levo car bastine
O- Olopa tidine
K- Keto tifen
A- Alcaf tadine
H2 blockers
Cime tidine,
Rani tidine,
Famo tidine,
Roxa tidine,
Niza tidine,
Lafu tidine,
H2 blockers which causes
Gynecomastia,
Menstrual irregulation
Cime tidine
H2 blockers which can cause
Galactorrhoea
Cime tidine
H2 blockers - max. CYP inhibitor
Cime tidine
Only drug for H3 receptor
Tipro lisant (pito lisant)
H3 INVERSE ANTAGONIST
INC. HISTAMINIC RELEASE
Tipro lisant can be used to treat
Narcolepsy
DOC in narcolepsy
Moda finil
No. Of receptors of serotonin
7,
5HT1-5HT7