CYP45 Inhibitors and Inducers Flashcards
(32 cards)
1
Q
Sodium Valproate
A
CYP450 inhibitor
2
Q
Isonizaid
A
CYP450 inhibitor
3
Q
Cimetidine
A
CYP450 inhibitor
4
Q
Ketoconazole
A
CYP450 inhibitor
5
Q
Fluconazole
A
CYP450 inhibitor
6
Q
Alcohol
A
CYP450 inhibitor
7
Q
Ciprofloxacin
A
CYP450 inhibitor
8
Q
Erythromycin/ Clarithromycin
A
CYP450 inhibitor
9
Q
Sulfonamide
A
CYP450 inhibitor
10
Q
Cranberry juice
A
CYP450 inhibitor
11
Q
Metronidazole
A
CYP450 inhibitor
12
Q
Grapefruit
A
CYP450 inhibitor
13
Q
Amiodaron
A
CYP450 inhibitor
14
Q
Verapamil
A
CYP450 inhibitor
15
Q
Itraconazole
A
CYP450 inhibitor
16
Q
Diltiazem
A
CYP450 inhibitor
17
Q
Barbituates
A
CYP450 inducer
18
Q
St. Johns Wart
A
CYP450 inducer
19
Q
Carbamazepine
A
CYP450 inducer
20
Q
Rifampicin
A
CYP450 inducer
21
Q
Alcohol
A
CYP450 inducer
22
Q
Phenytoin
A
CYP450 inducer
23
Q
Griseofulvin
A
CYP450 inducer
24
Q
Phenobarbital
A
CYP450 inducer
25
Sulfonylureas
CYP450 **inducer**
26
Warfarin
CYP450 **substrate**
27
Corticosteroids
CYP450 **substrate**
28
Oral contraceptives
CYP450 **substrate**
29
Aminophylline/ Theophylline
CYP450 **substrate**
30
31
Statins
CYP450 **substrate**
32
Tricyclic Antidepressants
CYP450 **substrate**