Enzyme Inducers/inhibitors Flashcards
(45 cards)
Carbamazepine
Induces Pgp, CYP 1A2/2C/3A, UGTs
Phenytoin
Induces Pgp, CYP 1A2/2C/3A, UGTs
Rifampin
Induces Pgp, CYP 1A2/2C/3A, UGTs
St. John’s Wort
Induces Pgp, CYP 3A
Ritonavir
Induces Pgp
Inhibits CYP 2D6/3A4
Tipanavir
Induces Pgp
Avasimbe
Induces Pgp
Phenobarbital
Induces CYP 1A2/2C/3A, UGTs
Felbamate
Induces CYP3A
Topiramate
Induces CYP3A
Oxcarbazepine
Induces CYP3A, UGTs
Griseofulvin
Induces CYP3A
Nevirapine
Induces CYP3A
Smoking
Induces CYP1A2
Alcohol
Induces CYP2E1
Lamotrigine
Induces UGTs
Oral contraceptives
Induces UGTs
Cyclosporin
Inhibits Pgp
Quinidine
Inhibits Pgp, CYP2D6
Verapamil
Inhibits Pgp
Amiodarone
Inhibits Pgp, CYP 1A2/2C9/2D6/3A4
Erythromycin
Inhibits Pgp, CYP3A4
Clarithromycin
Inhibits Pgp, CYP3A4
Azithromycin
Inhibits Pgp