Exact Classes of Drugs Flashcards

(159 cards)

1
Q

Trimethphan

A

Peripheral vasodilator and ganglionic blocker

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2
Q

Sodium Nitroprusside

A

Direct peripheral arterial vasodilator

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3
Q

Nitroglycerine

A

Organic nitrate vasodilator

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4
Q

HYDRALAZINE

A

VASODILATOR

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5
Q

MILRINONE

A

BYPYRIDINE INOTROPIC VASODILATOR WITH PHOPHODIESTERASE INHIB ACTIVITY

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6
Q

CLONIDINE

A

ALPHA 2 ADRENERGIC AGONIST VASODILATOR

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7
Q

KETAMINE

A

NON BARBITUATE INDUCTION, LIKE PCP

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8
Q

ETOMIDATE

A

NON BARBITUATE INDUCTION (IMIDAZOLE DERIVATIVE)

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9
Q

PROPOFOL

A

2, 6 DI ISO PROPOPHENYL; NON BARB INDUCTION

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10
Q

PRECEDEX

A

SELECTIVE ALPHA 2 AGONIST

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11
Q

KETEROLAC

A

NSAID

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12
Q

ESMOLOL

A

SELECTIVE BETA 1 ANTAGONIST

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13
Q

METOPROLOL

A

SELECTIVE BETA 1 ANTAGONIST

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14
Q

LABETOLOL

A

NON SELECTIVE BETA AND ALPHA 1 ANTAGONIST

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15
Q

PROPANOLOL

A

NON SELECTIVE BETA ANTAGONIST BETA 1 & 2

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16
Q

Prazosin

A

alpha 1 adrenergic antagonist

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17
Q

PHENOXYBENZAMINE

A

NON SELECTIVE ALPHA ADRENERGIC ANTAGONIST

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18
Q

PHENTOLAMINE

A

NON SELECTIVE ALPHA ADRENERGIC ANTAGONIST

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19
Q

HYDROCORTISONE

A

CORTICOSTEROID

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20
Q

METHYLPREDNISOLONE

A

CORTICOSTEROID

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21
Q

DEXAMETHASONE

A

CORTICOSTEROID

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22
Q

AMPICILLIN

A

ANTIMICROBIAL, BETA LACTUM, 2ND GEN. PCN, BROAD SPECTRUM, (GI/GU/DENTAL)

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23
Q

CEFAZOLIN

A

ANTIMICROBIAL, BETA LACTUM, 1ST GENERATION, BROAD SPECTRUM

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24
Q

GENTAMYCIN

A

ANTIMICROBIAL, AMINOGLYCOSIDE, BROAD SPECTRUM

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25
CLINDAMYCIN
ANTIMICROBIAL, LINCOSAMIDE, NARROW SPECTRUM, TREAT PCN RESIST STAPH AND BACTEROIDES
26
VANCOMYCIN
ANTIMICROBIAL, GLYCOPEPTIDES, BROAD SPECTRUM
27
METRONIDAZOLE
ANTIMICROBIAL, ANTI PROTOAZAN, ANAEROBIC
28
CIPROFLOXACIN
ANTIMICROBIAL, FLUORO QUINOLONE, BROAD SPECTRUM
29
DANTROLENE
DIRECT, CENTRALLY ACTING MUSCLE RELAXANT (TX: MH AND SKELETAL MUSCLE SPASTICITY)
30
REGLAN
ANTI NAUSEA/ANTI EMETIC, DOPAmine ANTAGONIST
31
DROPERIDOL
ANTI NAUSEA/ANTI EMETIC, DOPAmine ANTAGONIST
32
ONDASETRON/ZOFRAN
ANTI NAUSEA/ANT EMETIC, 5HT-3 INHIBITOR SERATONIN ANTAGONIST
33
PROMETHAZINE/PHENERGAN
ANTI NAUSEA/ANTI EMTIC, H1 ANTAGONIST PHENOTHIAZINE
34
OMEPRAZOLE/PRILOSEC
ANTI NAUSEA/ ANTI EMETIC, SUBSTITUTED BENZIMIDAZOLE (PPI)
35
SODIUM CITRATE BICTIRA
ANTI NAUSEA/ ANTI EMETIC, NON PARTICULATE ANTACID
36
ATROPINE
ANTICHOLINERGIC, TERTIARY AMINE, CROSSES BBB
37
GLYCOPYROLATE
ANTICHOLINERGIC, SYNTHETIC QUARTENARY AMMONIUM, DOES NOT CROSS BBB
38
SCOPALAMINE
ANTICHOLINERGIC, TERTIARY AMINE, CROSSES BBB AND PLACENTA
39
PYRIDOSTIGMINE
ANTICHOLINESTERASE INHIBITOR, QUARTENARY AMMONIUM, DOES NOT CROSS BBB
40
EDROPHONIUM
ANTICHOLINESTERASE INHIBITOR, QUARTENARY AMMONIUM, DOES NOT CROSS BBB
41
NEOSTIGMINE
ANTICHOLINESTERASES INHIBITOR, QUARTENARY AMMONIUM, DOES NOT CROSS BBB
42
PHYSOSTIGMINE
ANTICHOLINESTERASE, TERTIARY AMINE, CROSSES BBB, (TX: ATROPINE TOX, MG, GLAUCOMA)
43
EPINEPHRINE
ENDOGENOUS CATECHOLAMINE, NONSELECTIVE ADRENERGIV AGONIST
44
NOREPINEPHRINE (LEVOPHED)
DIRECT ACTING ENDOGENOUS CATECHOLAMINE AND ADRENERGIC AGONIST
45
DOPAMINE
ENDOGENOUS CATECHOLAMINE SYMPATHETIC AMINE ADN ADRENERGIV AGONIST
46
DOBUTAMINE
SYMPATHOMIMETIC, SYNTHETIC CATECHOLAMINE, B1 SELECTIVE AGONIST
47
VASOPRESSIN
EXOGENOUS ANTIDIURETIC PEPTIDE AND VASOPRESSOR
48
ISOPRETERONOL
SYNTHETIC CATECHOLAMINE, B1 >B2, MINIMAL ALPHA
49
EPHEDRINE
SYNTHETIC NON-CATECHOLAMINE, DIRECT AND INDIRECT ADRENERGIC AGONIST
50
PHENLYEPHRINE
SYNTHETIC NON CATECHOLAMINE DIRECT AND INDIRECT ACTING, SELECTIVE ALPHA 1
51
PHENYTOIN
ANTICONVULSANT, ANTIARRHYTHMIC CLASS 1B
52
PHENOBARBITOL
OXYBARBITUATE USED AS AN ANTICONVULSANT
53
TPL (THIOBARBITUATE)
BARBITUATE
54
METHOHEXITOL (OXYBARBITUATE)
BARBITUATE
55
CIMETIDINE
H2 BLOCKER
56
FAMOTIDINE
H2 BLOCKER
57
RANITIDINE
H2 BLOCKER
58
BENADRYL
H1 ANTAGONIST, 1ST GENERATION, CROSSES BBB
59
HEPARIN
ANTICOAGULANT, DVT PROPHYLAXIS, PE tx,
60
PROTAMINE
HEPARIN ANTIDOTE, LMW PROTEIN DERIVED FROM SALMON SEAMEN
61
INSULIN
PANCREATIC HORMONE STRUCTURALLY IDENTICAL TO ENDOGENOUS INSULIN
62
GLUCAGON
SYNTHETIC ANALOG OF ENDOGENOUS GLUCAGON, SECRETED IN RESPONSE TO HYPOGLYCEMIA, USED FOR SPHINCTER OF ODDI SPASM AND BB OD
63
OCTREOTIDE
SOMOSTATIN ANALOG, INHIBITS PRODUCTION AND RELEASE OF INSULIN AND GLUCAGON
64
OXYTOCIN
ENDOGENOUS POST PIT HORMONE
65
RAPID ACTING INSULIN CLASS NAMES
LISOPRO (HUMALOG) ASPART (NOVALOG) GLULISINE (APIDRA)
66
RAPID ACTING INSULIN MOA
MONOMORPH FORM - IMMEDIATELY AVAILABLE - MIMICS REGULAR MEAL RELEASE
67
SHORT ACTING INSULIN CLASS NAMES
REGULAR (HUMULIN R, NOVOLIN R)
68
SHORT ACTING INSULIN MOA
HEXOMER FORM, TAKES TIME TO BREAK DOWN TO MONOMORPH FORM
69
INTERMEDIATE ACTING INSULIN CLASS NAMES
NPH (HUMULIN N, NOVOLIN N)
70
INTERMEDIATE ACTING INSULIN MOA
N= NEUTRAL, P=PROTAMINE OFTEN COMBINED IWTH REGULAR INSULIN OR RAPID ACTING INSULIN
71
LONG ACTING INSULIN CLASS NAMES
GLARGINE (LANTUS) DETEMIR (LEVEMIR) ULTRALENTE
72
LONG ACTING INSULIN MOA
VERY PHYSIOLOGIC - NO PEAK, MIMICS BASAL INSULIN SECREITON CAN GIVE RAPID ACTING TO COVER EACH MEAL
73
GLULISINE (APIDRA)
RAPID ACTING INSULIN
74
ASPART (NOVALOG)
RAPID ACTING INSULIN
75
LISOPRO (HUMALOG)
RAPID ACTING INSULIN
76
GLARGINE (LANTUS)
LONG ACTING INSULIN
77
DETEMIR (LEVEMIR)
LONG ACTING INSULIN
78
ULTRALENTE
LONG ACTING INSULIN
79
NPH (HUMULIN N, NOVOLIN N)
INTERMEDIATE ACTING INSULIN
80
REGULAR (HUMULIN R, NOVOLIN R)
SHORT ACTING INSULIN
81
TOLBUTAMIDE/ CHLOROPROPAMIDE
ORAL ANTIDIABETIC MED, SULFONYLUREA 1ST GENERATION
82
GLIPIZIDE (GLUCATROL) GLYBURIDE (DIABETA) GLIMEPIRIDE
ORAL ANTIDIABETIC MED, SULFONYLUREA 2ND GENERATION
83
CHOLORPROPAMIDE
ORAL ANTIDIABETIC MED, SULFONYLUREA 1ST GENERATION
84
GLYBURIDE
ORAL ANTIDIABETIC MED, SULFONYLUREA 2ND GEN
85
GLIMEPIRIDE
ORAL ANTIDIABETIC MED, SULFONYLUREA 2ND GEN
86
METFORMIN (GLUCOPHAGE)
ORAL ANTIDIABETIC MED, BIGUANIDES
87
PIOGLITAZONE (ACTOS) | ROSIGLITAZONE (AVANDIA)
ORAL ANTIDIABETIC MEDS , THIAZOLIDINEDIONES (TZDs)
88
ACARBOSE (PRECOSE) | MIGLITOL (GLYSET)
ORAL ANTIDIABETIC MED, ALPHA GLUCOSIDASE INHIB
89
ROSIGLITAZONE (AVANDIA)
ORAL ANTIDIABETIC MED, TZD
90
ACARBOSE (PRECOSE)
ORAL ANTIDIABETIC MED, ALPHA GLUCOSIDASE INHIB
91
MIGLITOL (GLYSET)
ORAL ANTIDIABETIC MED, ALPHA GLUCOSIDASE INHIB
92
REPAGLINIDIE (PRANDIN)
ORAL ANTIDIABETIC MED, MEGLITINIDES
93
NATEGLINIDE (STARLIX)
ORAL ANTIDIABETIC MED, MEGLITINIDES
94
SITAGLIPTAN (JANUVIA)
ORAL ANTIDIABETIC MED, GLP-1 MIMETIC AND AGONIST
95
EXENATIDE (BYETTA)
ORAL ANTIDIABETIC MED, GLP-1 MIMETIC AND AGONIST
96
ORAL ANTIDIABETIC MED, meGLITINIDES
repaGLINIDE (PRANDIN) | nateGLINIDE (STARLIX)
97
oral antidiabetic med, GLP-1 MIMETIC and AGONIST
sitagliptan (januvia) | exenatide (byetta)
98
Morphine
OPIOID, natural opioid agonst
99
MEPERIDINE
OPIOID, PHENYL PIPERIDINE SYNTHETIC OPIOID AGONIST
100
FENTANYL
OPIOID, PHENYL PIPERIDINE SYNTHETIC OPIOID AGONIST
101
SUFENTANYL
OPIOID, PHENYL PIPERIDINE SYNTHETIC OPIOID AGONIST
102
ALFENTANYL
OPIOID, TETRAZOLE FENTANYL DERIVATIVE, SYNTHETIC OPIOID AGONIST
103
REMIFENTANYL
OPIOID, PHENYL PIPERDINE SYNTHETIC OPIOID AGONIST WITH ESTER LINK
104
Succhinylcholine
DEPOLARIZING NEUROMUSCULAR BLOCKER
105
ATRACURIUM (TRACURIUM)
NEUROMUSCULAR BLOCKER, INTERMEDIATE ACTING BISQUATERNARY BENZYLISOQUINOLINE
106
CISATRACURIUM (NIMBEX)
NEUROMUSCULAR BLOCKER, INTERMEDIATE ACTING BENZYLISOQUINOLINE STEREOISOMER OF ATRICURIUM
107
ROCURONIUM (ZEMURON)
NEUROMUSCULAR BLOCKER, SHORT-INTERMEDIATE ACTING STERIOD TYPE
108
VECURONIUM (NORCURON)
NEUROMUSCULAR BLOCKER, INTERMEDIATE ACTING STEROID TYPE MONOQUATERNARY AMINOSTERIOD
109
PANCURONIUM (PAVULON)
NEUROMUSCULAR BLOCKER, LONG ACTING STERIOD TYPE BISQUATERNARY AMINOSTEROID
110
MIVACURIUM (MIVACRON)
NEUROMUSCULAR BLOCKER, SHORT ACTING BENZYLISOQUINOLINE
111
D-TUBOCURARINE (CURARE)
NEUROMUSCULAR BLOCKER, LONG ACTING BENZYLISOQUINOLINE
112
DOXACURIUM (NEUROMAX)
LONG ACTING BENZYLISOQUINILINE
113
PIPERCURONIUM (ARDUAN)
LONG ACTING STEROID TYPE
114
NALBUPHINE
OPIOID AGONIST-ANTAGONIST (MU ANTAGONIST AND FULL OR PARTIAL AGONIST AT KAPPA)
115
BUTORPHANOL
OPIOID AGONIST - ANTAGONIST (NASAL SPRAY FOR MIGRANES)
116
DIAZEPAM (VALIUM)
BENZODIAZEPINE
117
MIDAZOLAM (VERSED)
BENZODIAZEPINE WITH AN IMIDAZOLE RING
118
LORAZEPAM (ATIVAN)
BENZODIAZEPINE
119
FLUMAZENIL
BENZO RECEPTOR ANTAGONIST, IMIDAZOBENZODIAZEPINE DERIVATIVE
120
NITROUS
INHALATION AGENT, INORGANIC, COLORLESS, SWEET GAS AT ROOM TEMP, MAC: 105 BG: 0.47 VP: 38770
121
HALOTHANE
INHALATION AGENT; HALOGENATED ALKALINE DERIVATIVE WITH BROMIDE SUBSTITUTION (SWEET, PUNGENT, CONTAINS THYMOL) MAC: 0.74 BG: 2.4 VP: 244
122
ENFLURANE
INHALATION AGENT, HALOGENATED METHYL ETHYL ETHER (MILD, SWEET, ISOMER OF ISO) MAC: 1.7 BG: 1.8 VPP: 175
123
ISOFLURANE
INHALATION AGENT, HALOGENATED METHYL ETHYL ETHER (ISOMER OF ENFLURANE, PUNGENT) MAC: 1.15 BG: 1.4 VP: 240
124
DESFLURANE
INHALATION AGENT, FLUORINATED METHYL ETHYL ETHER (SIMILAR STRUCTURE TO ISO, PUNGENT, TEC 6, FAST ON/OFF) MAC: 6 BG: 0.42 VP: 669
125
SEVOFLURANE
INHALATION AGENT, FLUORINATED METHYL ISOPROPYL ETHER (IDEAL FOR PEDS, NON PUNGENT, SWEET, EXPENSIVE) MAC: 2.05 BG: 0.69 VP: 157
126
PROCAINE
``` LOCAL ANESTHETIC: ESTER PKA: 8.9, LS: 1, PB: 5 DOSE: 7MG/KG SPINAL: 100-200MG DOA: ~60MIN PNB: 100-400MG DOA~30 MINUTES ```
127
AMIODARONE
ANTI-ARRHYTHMIC, CLASS 3, ALSO HAS CLASS 1,2,4 PROPERITES
128
ADENOSINE
ANTI-ARRHYTHMIC, ENDOGENOUS NUCLEOTIDE
129
DIGOXIN
ANTI-ARRHYTHMIC, CARDIAC GLYCOSIDE, MANDAGE AFIB/AFLUTTER
130
QUINIDINE
ANTI-ARRHYTMIC, CLASS 1, MANAGE SVT/AFIB
131
PROCAINAMIDE
ANTI-ARRYTHMIC, CLASS 1A, ANALOGUE OF PROCAINE (TX: AFIB/VTACH)
132
DILTIZEM
CALCIUM CHANNEL BLOCKER CLASS 4 ANTI-ARRHYTHMIC, NON DIHYDROPYRIDINE
133
VERAPAMIL
CALCIUM CHANNEL BLOCKER, CLASS 4 ANTI-ARRHYTHMIC, NON DIHYDROPYRIDINE
134
NIFEDIPINE
CALCIUM CHANNEL BLOCKER, CLASS 4 ANTI-ARRHYTHMIC, DIHYDROPYRIDINE
135
PROTON PUMP INHIBITORS (-PRAZOLE)
``` LANSOPRAZOLE PANTOPRAZOLE ESOMEPRAZOLE OMEPRAZOLE RABEPRAZOLE ```
136
DICYCLOMINE
ANTICHOLINERGIC
137
ANATACIDS | ALUM, CALCIUM, MAG, SODIUM)
ALUMINUM HYDROXIDE MAGNESIUM HYDROXIDE SODIUM BICARBONATE CALCIUM CARBONATE
138
MISOPROSTOL
PROSTAGLANDIN
139
SODIUM CITRATE
ANTACID (NON PARTICULATE ANTACID THERAPY)
140
CISAPRIDE | DOPERIDONE
PROKINETIC
141
SEROTONIN
5HT pro kinetic drug
142
5ht3 antagonists - prokinetic (-setron)
ondasetron granisetron dolasetron tropisetron
143
DEXAMETHASONE
STEROID
144
FUROSEMIDE
LOOP DIURETIC
145
HYDROCHLOROTHIAZIDE
THIAZIDE DIURETIC
146
MANNITOL (6 CARBON HEXOSE SUGAR)
OSMOTIC DIURETIC
147
ALBUTEROL
``` RESPIRATORY AGENT, B2 AGONIST SHORT ACTING, 2 ISOMERS (R & S) ```
148
TERBUTALINE
RESPIRATORY AGENT, BE AGONIST, SHORT ACTING
149
IPRATROPIUM
RESPIRATORY AGENT, ANTICHOLINERGIC, QUATERNARY AMINE, SALT DERIVATIVE OF ATROPINE
150
TETRACAINE
LOCAL ANESTHETIC: ESTER. PKA 8.5, LS: 80, PB: 85% DOSE: 3MG/KG SPINAL (0.23-1.0%): 5-20 MG DOA~90-200MIN
151
BUPIVICAINE
LOCAL ANESTHETIC: AMIDE PKA 8.1, LS: 30, PB 90% DOSE 2.5MG/KG EPIDURAL (0.25-0.75%): 40-225MG DOA~ 180-350MIN SPINAL (0.5-0.75%: 15-20MG DOA~90-200 MIN PNB (0.25-0.5%) MAJOR: 225MG MAX. MINOR: 12.5-100 MG DOA~240-420MIN
152
LIDOCAINE
``` LOCAL ANESTHETIC: AMIDE PKA, 7.9, LS: 4, PB: 65% DOSE 4MG/KG, 7MG/KG* ACLS: 1MG/KG EPIDURAL (1-2%) 150-500MG SPINAL (1.5, 5.0%) 30-100MG DOA~60 MIN PNB: MAJOR (1-2%)500MG MAX. MINOR(1%)50-200 MG DOA~60MINUTES ```
153
MEPIVICAINE
``` LOCAL ANESTHETIC: AMIDE PKA. 7.6, LS: 1, PB: 75% DOSE: EPIDURAL (1-2%) 150-500MG DOA~120 MIN SPINAL (4%) 40-80 MG DOA~60 MIN PNB: MAJOR (1-1.5%) 500MG MAX. MINOR (1%) 50-200MG DOA~180 MINUTES ```
154
ETIDOCAINE
LOCAL ANESTHETIC: AMIDE PKA 7.7, LS: 140 PB: 95% DOSE: 4MG/KG, 7MG/KG*
155
CHLOROPROCAINE
``` LOCAL ANESTHETIC: ESTER PKA: 8.7, LS: 1, PB: 7% DOSE 12MG/KG EPIDURAL (2-3%) 300-900 DOA~60 MIN PNB: MINOR (2%) 100-400MG DOA~30 MINUTES ```
156
COCAINE
LOCAL ANESTHETIC: ESTER. MET IN LIVER. | DOSE: 3MG/KG
157
LEVOBUPIVICAINE
``` LOCAL ANESTHETIC: ESTER. DOSE: EPIDRUAL (0.25-0.75%) 40-250MG DOA~240 min spinal (0.5-0.75%) 15-20MG DOA~120 min PNB: MAJOR (0.25-0.5%) 225MG MAX. ```
158
ROPIVACAINE
``` LOCAL ANESTHETIC: AMIDE DOSE EPIDURAL (0.25-0.7%) 40-250MG DOA~240 MIN SPINAL (0.5-0.75%) 15-20MG DOA~120 MIN PNB MAJOR (0.2-0.5%) 250MG MAX. MINOR (0.2-0.5%) 10-100MG DOA~240 MIN ```
159
PRILOCAINE
``` LOCAL ANESTHETIC: AMIDE DOSE EPIDURAL (1-3%) 150-600MG PNB MAJOR(1-2%) 600MG DOA ~ 240 MIN MINOR (1%) 50-200MG DOA~120 MIN ```