Exam 1 Flashcards
(32 cards)
Cholinomimetics: Direct acting- choline esters
ACh
bethanechol
methacholine
carbechol
Cholinomimetics: Direct acting- naturally occurring
nicotine
muscarine
pilocarpine
Cholinomimetics: Indirect acting: Reversible AChE inhibitors
physostigmine neostigmine pyridostigmine ambenonium edrophonium tacrine and donepezil carbaryl
Cholinomimetics: Indirect acting: Irreversible AChE inhibitors
echotiophate dyflos/fluostigmine parathion malathion sarin and soman
Anticholinergics: Antimuscarinics
atropine scopolamine tropicamide cyclopentolate ipratropium tiotropium benzotropine trihexphenidyl
Ganglionic blocker
hexamethonium, nicotine (high doses)
Neuromuscular blockers- non-depolarizing/competetive
tubocurarine doxacurium pancuronium atracurium cistacurium vecuronium rocuronium mivacuronium
Anticholinergics: neuromuscular blockers: depolarizing
succinylcholine
Block ACh synthesis w/
hemicholinium
Block ACh storage w/
vesamicol
Block ACh release w/
botulinum toxin
Sympathomimetics: Direct acting: Endogenous
epi
norepi
dopamine
Sympathomimetics: Direct acting: alpha1 selective agonists
phenylephrine
methoxamine
midodrine
Sympathomimetics: Direct acting: alpha2 selective agonists
clonidine a-methyldopa apraclonidine and brimonidine guanfacine tizanidine
Sympathomimetics: Direct acting: Non selective Beta agonists
isoproterenol
ephedrine
pseudoephedrine
Sympathomimetics: Direct acting: Beta1 agonist
dobutamine
Sympathomimetics: Direct acting: Beta3 agonists
mirabegron
Sympathomimetics: Indirect acting
tyramine amphetamine methamphetamine methylphenidate cocaine TCAs
Adrenergic Blockers: Alpha blockers-nonselective
phentolamine
phenoxybenzamine
Adrenergic Blockers: Alpha1 blockers
prazosin
terazosin
doxazosin
Adrenergic Blockers: Alpha2 blockers
yohimbine
Adrenergic Blockers: Beta blockers-nonselective
propranolol
pindolol
timolol
nadolol
Adrenergic Blockers: Beta1 blockers- selective
metoprolol
atenolol
betaxolol
esmolol
Adrenergic Blockers: Beta2 blockers- selective
butoxamine