Muscarinic receptor agonist or antagonist Flashcards
(101 cards)
1
Q
Carbachol
A
Muscarinic receptor agonist
2
Q
Bethanechol
A
muscarinic receptor agonist
3
Q
Pilocarpine
A
Vuity - muscarinic receptor agonist
4
Q
Cevimeline
A
Evoxac - muscarinic receptor agonist
5
Q
Botox
A
Botulinum toxin -indirect acting parasympatholytics
6
Q
Daxxify
A
Botulinum toxin -indirect acting parasympatholytics
7
Q
Atropine
A
Muscarinic receptor antagonist
8
Q
Glycopyrrolate
A
Muscarinic receptor antagonist
9
Q
Dicyclomine
A
Muscarinic receptor antagonist
10
Q
Hyoscyamine
A
Muscarinic receptor antagonist
11
Q
Scopolamine
A
Muscarinic receptor antagonist
12
Q
Belladonna
A
Muscarinic receptor antagonist
13
Q
Ipratropium
A
Atrovent Muscarinic receptor antagonist
14
Q
Tiotropium
A
Spiriva Muscarinic receptor antagonist
15
Q
Tolterodine (De-)
A
Detrol Muscarinic receptor antagonist
16
Q
Fesoterodine
A
Toviaz Muscarinic receptor antagonist
17
Q
Oxybutynin
A
Ditropan Muscarinic receptor antagonist
18
Q
Darifenacin (ena-
A
Enablex Muscarinic receptor antagonist
19
Q
Solifenacin (vesi)
A
Vesicare Muscarinic receptor antagonist
20
Q
Trospium
A
Sanctura Muscarinic receptor antagonist
21
Q
Revefenacin
A
Yupelri Muscarinic receptor antagonist
22
Q
Neostigme
A
Reversible cholinesterase inhibitor
23
Q
Physostigmine
A
reversible cholinesterase inhibitor
24
Q
Pyridostigmine
A
reversible cholinesterase inhibitor
25
Ambenonium
reversible cholinesterase inhibitor
26
edrophonium
reversible cholinesterase inhibitor
27
Malathione
| ovide
irreversible cholinesterase inhibitor
28
Parathion
Is a insecticide is a irreversible cholinesterase inhibitor
When the pt inhales it is going to go in cholinergic crisis state
29
Sarin
Is a nerve gas that is irreversible cholinesterase inhibitor and when the pt inhales it the pt will go into cholinergic crisis and cause bronchioconstriction and dies
30
Pralidoxime
| 2-Pam
is a antidote of intoxication of irreversable cholinesterase inhibitors
If is administer before the complex between the irriversible cholinesterase inhibitor and the enzyme cholinesterase form Pralodixime will reactivate the acetyl cholinesterase
31
Nicotine
| Explain the physical dependence
32
Varenicline
| Chantix
Central nicotinic partial agonist
33
Vecuronium
Muscle nicotinic receptor antagonist
34
Atracurium
Muscle nicotinic receptor antagonist
35
Doxacurium
Muscle nictonic receptor antagonist
36
Cisatracurium
Muscle nicotinic receptor antagonist
37
Rocuronium
Muscle nicotinic receptor antagonist
38
Pipecuronium
Muscle nictonic receptor antagonis
39
Pancuronium
Muscle nicotinic receptor antagonist
40
Succinylcholine
Muscle nicotinic receptor agonist
41
Sugammadex
Reverse the effects of vecuronium and rocuronium
42
Rivastigmine
Reversible cholinesterase inhibitor
43
Donezepil
Reversible cholinesterase inhibitor
44
DFP
| Diisopropyl flurophosphate
Irreversible cholinesterase inhibitor use as eye drops
45
Echothiophate
Irreversible cholinesterase inhibitor
46
Dobutamine
B1 Selective Receptor Agonist
47
Atenolol
B1 antagonist
48
Acebutolol
B1 antagonist
49
Betaxolol
b 1 receptor antagonist
50
Bisoprolol
B1 Antagonist
51
Metoprolol
| Tropol XR
B1 receptor antagonist
52
nebivolol
B1 receptor antagonist
53
Esmolol
| brevibloc
B1 receptor antagonist
54
Ivabradine
| Corlanor
affects the cardiac currents
55
Albuterol
B2 agonist
56
Levalbuterol
| xopenex
Xopenex
B2 agonist
57
Salmeterol
B2 agonist
58
Formoterol
B2 agonist
59
Alformoterol
b2 agonist
60
Indacaterol
B2 receptor agonist
61
Olodaterol
B2 agonist
62
Pirbuterol
B2 agonist
63
Vilanterol
B2 agonist
64
Terbutaline
B2 agonist
65
Roflumilast
| Daliresp
PDE4 inhibitor
66
Theophylline
Non selective Phosphodiesterase inhibitor
67
Aminophylline
Non Selective Phosphodiesterase inhibitor
68
Norepinephrine
Has more affinity to the Alpha subtypes
Can be metabolize by MOA and COMT
69
Epinephrine
Has better affinity to beta receptors
Metabolize by N-demethylation or COMT
70
Isoproterenol
Non selective Beta-adrenergic agonist
71
Propranolol
| Inderal
Non Selective B-adrenergic Antagonist
72
Nadolol
Non selective Beta-adrenergic antagonist
73
Pindolol
Non Selective beta-adrenergic antagonist
74
Sotalol
Non selective Beta-adrenergic antagonist
75
Timolol
Non selective Beta-adrenergic antagonist
76
Levobunalol
Non selective Beta adrenergic antagonist
77
Mirabegron
| Myrbetriq
B3 Receptor Agonist
78
Vibegron
| Gemtesa
B3 Selective agonist
79
Midodrine
Alpha 1 selective receptor agonist
80
Phenylephrine
Alpha 1 selective agonist
| Neo-Synephrine
81
Pseudoephrine
Alpha 1 selective agonist
| Sudafed
82
Oxymetazoline
Alpha 1 selective agonist
| Afrin
83
Northera
Inderect sympathomimetic
| Droxidopa
84
Prazosin
Non Selective Alpha 1 antagonist
Block A1B- Blood vessels
Block A1A- Prostate and bladder
85
Terazosin
Non selective Alpha 1 antagonist
Block A1B-blood vessel
Block A1A- Prostate and bladder
86
Doxazosin
Non selective Alpha 1 antagonist
Blocks A1A- prostate and bladder
Blocks A1B- Blood vessels
87
Alfuzosin
Selective Alpha a1a antagonist
88
Tamsulosin
Selective Alpha 1 antagonist
A1A antagonist
89
Labetalol
Non selective Alpha 1, Beta 1 and Beta 2 antagonist
90
Carvedilol
Non selective alpha 1, Beta 1, Beta 2 antagonist
91
Clonidine
Alpha 2 agonist
92
Lofexidine
Alpha 2 agonist
93
Methyldopa
Alpha 2 agonist
94
Guanfacine
Alpha 2 agonist
95
Dexmedetomidine
Alpha 2 agonist
96
Brimonidine
| Alphagan, mirvaso
Alpha 2 agonist
97
Apraclonidine
Alpha 2 agonist
98
Phentolamine
Non selective alpha adrenergic antagonist
| Oraverse
99
Phenoxybenzamine
irreversible non selective alpha adrenergic antagonist
100
Metyrosine
Indirect acting sympatholytic
| Inhibit tyrosine hydroxylase
101
Reserpine
Indirect acting sympatholytics
| Inhibit VMAT
