random Flashcards
(10 cards)
1
Q
Cyproheptadine
A
serotonin receptor antagonist Tx for seratonin syndrome
2
Q
aluminum antidote
A
deferoxamine
3
Q
DNA pol 3
A
Initiates replication in prokaryotes. Has primate activity. Analogous to pol alpha in eu
4
Q
-navirs
A
Protease inhibitors, depend on hiv protease (pol gene)
5
Q
NNRTIs
A
Delavirdine
Efavirenz
Nevirapine
Non comp inhibitors of RT. Don’t require phosphorylation.
6
Q
NRTI
A
All require activation except tenofovir.
Zidovudine used in ppx for preggers
7
Q
Raltegravir
A
Inhibits integrase in hiv
8
Q
Hiv fusion inhibitors
A
Enfuvirtide (gp41)
Maraviroc (ccr5 )
9
Q
Cidofovir
A
Inhibits viral DNA pol, doesn’t require activation.
10
Q
Foscarnet
A
Viral DNA/rna pol inhibitors and hiv RT.
Pyro phosphate analog. Doesn’t require activation.