03 - Synaptic Flashcards
(25 cards)
pilocarpine
muscarinic agonist
atropine
muscarinic antagonist
scopolamine
muscarinic antagonist
anaesthetic pre-med
pancuronium (-onium)
nicotinic antagonist (competitive blocker) non-depolarising block
nicotinic agonist
duh..
depolarising block
acts on NMJ and autonomic ganglia
trimetaphan
ganglia blocker
hexamethonium
ganglia channel
via channel block
bromopyruvate
Drugs acting pre-synaptically
target: pyruvate
hemicholinium
Drugs acting pre-synaptically
target: choline transport
vesamicol
Drugs acting pre-synaptically
target: vesicle transport
botulinum toxin
Drugs acting pre-synaptically
target: exocytosis
edrophonium
anti-AChE
short-acting for M.S. diagnosis
neostigmine
anti-AChE
medium-acting for M.S. treatment
dyflos
anti-AChE
long-acting / irreversible
clonidine
(1) alpha(2) autoreceptor agonist
doubutamine (-buta-)
beta(1) agonist
salbutamol (-buta-)
beta(2) agonist
phenoxybenzamine
alpha(1) blocker
2) NRI (NET inhibitor
tamsulosin (-osin)
alpha(1) blocker
propanolol (-olol)
beta blocker
atenolol (-lol)
beta blocker
tyramine
(3) indirectly-acting sympathomimetic
alpha-methyl DOPA
(4) false transmitter
lidocaine / lignocaine
(5) local anaesthetic