Nifedipino Flashcards

1
Q

Mecanismo de acción

A

Bloqueador drihidropiridínico de los canales de calcio tipo L

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
2
Q

Indicaciones clínicas

A

Angina variante y de esfuerzo

Actualmente descontinuado por su absorción tan acelerada

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
3
Q

Farmacocinética relevante

A
A: Oral
    F: 90-100%
D: 
    PB: 98-100%
    VD: 54L
M: Hepático CYP3A4
E:  Renal/Heces
     V1/2e: 2-7h
How well did you know this?
1
Not at all
2
3
4
5
Perfectly
4
Q

Reacciones adversas

A
Hipotensión
Palpitaciones
Edema
Flushing
Mareo
Taquicardia importante
How well did you know this?
1
Not at all
2
3
4
5
Perfectly
5
Q

Interacciones relevantes

A

Inhibidores de CYP3A4

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
6
Q

Clasificación en el embarazo

A

C

Viable durante la lactancia

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
7
Q

Precauciones y contrainidicaciones

A

Shock Cardiogénico

How well did you know this?
1
Not at all
2
3
4
5
Perfectly