ACETAMINOPHEN (TYENOL) Flashcards
(10 cards)
CLASS
ANALGESIC, ANTIPYERETIC
DESCRIPTION
ACTS PRIMARILY ON CNS INCREASING THE PAIN THRESHOLD BY INHIBITING THE ISOFORMS OF CYCLOOXYGENASE, ENZYMES THAT ARE INVOLVED IN PROSTAGLANDIN SYNTHESIS.
ONSET & DURATION
ONSET- ORALLY: 10- 30 MINUTES
IV- 3-5 MINUTES
DURATION- PO: 3-4 HOURS
IV: 4-6 HOURS
INDICATIONS
TEMPORARY RELIEF OF FEVER, MILD OR MODERATE PAIN
CONTRAINDICATIONS
HYPERSENSITIVITY
HEPATIC IMPAIRMENT
RENAL IMPAIRMENT
HYPOVOLEMIA, SEVERE
CHRONIC ALCOHOL USE
ADVERSE REATIONS
NAUSEA/VOMITING
RASH
HEADACHE
ANEMIA
THROMBOCYTOPENIA
DRUG INTERACTIONS
VOID WITH CONCURRENT USE OF ETHANOL, ISOIAZID, AND OVER-THE-COUNTER DRUGS THAT CONTAIN ACETAMINOPHEN.
HOW ACETAMINOPHEN IS SUPPLIED
325MG, 500MG,(CAPSULES)
DOSAGE AND ADMINISTRATION
MILD PAIN AND FEVER: 325- 1000 MG PO EVERY 4-6 HOURS AS NEEDED
SPECIAL CONSIDERATIONS
PREGNANCY SAFTEY- CATEGORY B
HARMLESS AT LOW DOSES, MAY CAUSE ACUTE LIVER FAILURE IF TAKEN IN EXCESS