anti- arrhythmia drugs Flashcards
(8 cards)
PROCAIDENAMIDE
CLASS ONE DRUG (NA CHANNEL BLOCK)
FIRST LINE TX FOR V.A
ADMINISTER VIA IV
LIDOCAINE
CLASS ONE DRUG
GIVEN VIA IV FOR V.A
ALSO USED AS A TOPICAL ANAESTHETIC
IT CAN ALSO BE INJECTED BELOW THE DERMIS BEFORE INSERTION
OR INSTILLED DOWN ETT PRE-SUCTION TO PREVENT COUGHING
SIDE EFFECTS- CAN SLOW REFRACTORY PERIOD TOO MUCH CAUSING 2ND DEGREE HEART BLOCK OR EVEN CAUSE COMPLETE BLOCK ( ASYSTOLE)
METOPROPOL AND LABETALOL
BOTH DRUGS ARE CLASS 2 (BETA BLOCKER)
CAN BE TAKEN PO AS A MAINTENANCE DRUG AFTER MI AND VIA IV IN EMERGENCY SITUATIONS
SIDE EFFECTS
-BRONCHOSPASMS (DUE TO CROSS OVER EFFECT)
BRADYCARDIA
HYPOTENSION- ALSO USE AS AN ANTI- HYPERTENSION
AMIODARONE
CLASS THREE DRUG ( PROLONGS PHASE 3) USE AS A FIRTS LINE THERAPY FOR -A-FIB AND V-TACH BROAD SPECTRUM USAGE PO AND IV
SIDE EFFECTS
- BRADYCARDIA
- HYPOTENSION
- INTERSTITIAL PULMONARY FIBROSIS
DILTIAZEM (CARDIZEM)
VERAPAMIL
CLASS 4 DRUG (CA CHANNEL BLOCKER)
NEG DROMOTROPES
ALSO CAUSES VASODILATION
ANGINA RELIEVER
SIDE EFFECTS
HYPOTENTION (LOW BP)
PERIPHERAL EDEMA
ATROPINE
COMPETITIVE ANTAGONIST FOR MUSCARINIC RECEPTORS
HAS NO INOTROPIC EFFECT
ADENOSINE
CAUSES A COMPLETE DEPRESSION OF SA AND ACV NODE CONDUCTION FLAT LINE UNTIL DRUG WEARS OFF IV PUSH FOLLOWED BY SALINE ONLY USE ON ACUTE SITUATIONS ALSO A VASODILATOR SIDE EFFECTS CAN BE DETREMENTAL IF PT DONT RETURN TO S.R CHEST PAIN BRONCHOCONSTRICTION
DIGOXIN
NOT PART OF THE 4 CLASS DRUGS
SECOND LINE THERAPY AFTER BETA BLOCKERS
BLOCKS THE AV NODE, DECREASING CONDUCTION INTO VENTRICLES
HAS SOME (+) INOTROPIC EFFECTS- INCREASES CO
BUT SMALL THERAPEUTIC INDEX