Pharma Final Drug Names Flashcards

(231 cards)

1
Q

Direct Parasympathomimetics

A
ACh
Carbachol
Pilocarpine 
Bethanacol (Hu)
Methacoline (Hu)
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2
Q

Indirect Parasympathomimetics

A
Physostigmine 
Neostigmine 
Pyridostigmine 
Edrophonium (Tensilon)
Organophosphates: Diazinon (ectoparasiticide) and Echothiophate
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3
Q

Parasympatholytics

A
Atropine!
Tropicamide
Homatropine 
Ipratropium
Glycopyrrolate
Benzethimide
Butyl scopalamine
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4
Q

Non-specific sympathomimetics

A

Adrenaline/ Epinephrine
Noradrenaline/ Norepinephrine
Dopamine

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5
Q

Specific Sympathomimetics: Beta1 Adrenoreceptor agonists

A

Dobutamine

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6
Q

Specific Sympathomimetics: Beta2 Adrenoreceptor Agonists

A
Clenbutarole
Salbutamole
Terbutarole
Salmeterole 
Isoxsuprine
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7
Q

Specific Sympathomimetics: Alpha1 Adrenoreceptor Agonists

A

Phenylephrine
Xylometazoline, Oxymetazoline, Naphazoline, Tetrazoline
Phenylpropanolamine
Ephedrine

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8
Q

Specific Sympathomimetics: Alpha2 Adrenoreceptor Agonists

A

Xylazine
Detomidine
Medetomidine

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9
Q

Sympatholytics: Alpha

A

Phenoxybenzamine (non-specific)
Prazosine, Doxasosine (specific alpha1)
Atipamezole, Yohimbine (specific alpha2)

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10
Q

Sympatholytics: Beta

A

Propanole, Timolol (non-specific)

Atenolole, Metapronole (specific beta1)

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11
Q

Tranquilizer Sedatives

A

Phenothiazine and Butyrophenone derivatives

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12
Q

Phenothiazine Derivatives

A
Chlorpromazine 
Propionyl-promazine
Acepromazine 
Promethazine 
Trifluorperazine 
Proquamezine
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13
Q

Butyrophenone Derivatives

A

Azaperone
Droperidol
Haloperidol
Fluanison

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14
Q

Alpha-2-agonists

A
Xylazine
Detomidine 
Medetomidine 
Dexmedetomidine
Romifidine
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15
Q

Alpha-2-Antagonists

A

Atipamezole

Yohimbine

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16
Q

Benzodiazepines

A

Diazepam
Midazolam
Clonazepam

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17
Q

Barbiturates

A

Long: Phenobarbital
Short: Pentobarbital
Ultra-short: Thiopental, Thiomylal, Methohexital

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18
Q

Proprandiol derivatives

A

Meprobamate

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19
Q

The sedato-hypnotics

A

Alpha-2-agonists
Benzodiazepines
Proprandiol derivs
Barbiturates

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20
Q

Endogenous Opioids:

A

Opiopeptins!
Encephalins
Endorphins

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21
Q

Semisynth Opioids

A
Azidomorphine 
Ethylmorphine 
Etorphine 
Heroin
Burenorphine 
Hydro- and Oxycodone 
Hydro- and Oxymorphone
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22
Q

Synth Opioids

A
Morphinanes: Butorphanol
Diphenyl heptanes: Methadone 
Phenylpiperidines: Pethidine, Fentanyl, Diphenoxylate, Loperamide
Benzomorphanes: Pentazocine
Cyclohexanols: Tramadol
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23
Q

Opioid Active substances:

A
Morphine
Fentanyl
Sulfetanyl and Remifentanyl
Tramadol
Buprenorphine 
Butorphanol
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24
Q

Neuroleptanalgesia

A

Tranquilizer and opiate

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25
Ataranalgesia
BZD and opiate
26
Inhalational Anaesthetics
``` Halothane Isoflurane Sevoflurane Desflurane N2O ```
27
Injectable Anaesthetics
``` Barbiturates Propofol Imidazoles Dissociative Anaesthetics Steroid Anaesthetics ```
28
Imidazoles
Etomidate | Metomidate
29
Dissociative Anaesthetics
Ketamine | Tiletamine
30
Steroid Anaesthetics
Alfaxlon | Alfadolon
31
Anticonvulsants: Barbiturates
Phenobarbital Pentobarbital Primidone
32
Anticonvulsants: Benzodiazepines
Diazepam Clonazepam Carbamazepin
33
Anticonvulsants: Others
Phenytoin | Valproic acid
34
Treatment of status epilepticus
Diazepam Phenobarbital (pentobarbital) Propofol
35
Prevention of seizures: Maintenance
``` Phenobarbital Phenytoin Valproic acid Bromide salts (Na, K) Clonazepam Clorazepate Felbamate Gabapentin Primidone ```
36
Active sunstances: Anticonvulsants
``` Phenobarbital Diazepam Clonazepam Sodium potassium bromide Phenytoin Carbamazepine Sodium Valproate Gabapentin ```
37
Antidepressants
Tricyclic Antidepressants (TCA's) Serotonin Reuptake Inhibitors (SRI's) Monoamine Oxidase Inhibitors (MAOI's) Lithium
38
Tricyclic Antidepressants (TCA's)
Amitryptiline Clomipramine Doxepin Imipramine
39
Serotonin Reuptake Inhibitors (SRI's)
Fluoxetine Fluvoxamine Sertraline
40
Monoamine Oxidase Inhibitors (MAOI's)
Selegiline
41
Behaviour Modifying Drugs
Sedatives: Neuroleptics, BZD Beta-adrenoceptor antagonists: Propranolol Antiepileptics:Carbamezipine, Phenobarbital Opioid antagonists: Naloxone, Naltrexone CNS stimulants: Dexamphetamine Antihistamines: Chlorphenamine, Diphenhydramine Hormones: Megastrol, Cabergoline, Dalmadinon Cerebral VasoD: Nicergoline, Propenfophylline Artificial Pheromones: Feliway, Felifriend, DAP Feed supplements: Alpha casozepine, Tryptophan
42
Depolarizing NM Blocking Agents:
Succinylcholine/ Succinylcholine Chloride/ Suxamethonium
43
Non-depolarizing/ Competitive NM Blocking Agents class acc to structure
Benzylisoquinolin group Aminosteroid group Others (Gallamine)
44
Non-depolarizing/ Competitive NM Blocking Agents class acc to duration of action
Ultra-short: Gentacurium Short: Mivacurium, Chandonium Intermediate: Atracurium, Cistracurium, Rocuronium, Vecuronium Long....
45
Benzyl Isoqiunolin group NM blocking agents
d- Tobobcurarine Atracurium Cisatracurium Mivacurium
46
Aminosteroid group NM Blocking agents
Pancuronium Vecuronium Rocuronium
47
Non-depolarizing/ Competitive NM Blocking Agents to discuss in the exam
``` d- Tobocurarine Gallamine Atracurium Cisatracurium Vecuronium Rocuronium Mivacurium ```
48
Local Anaesthetics: Esters
Procaine Tetracaine Benzocaine Cocaine
49
Local Anaesthetics: Amides
Prilocaine Lignocaine Mepivacaine/ Ropivacaine Bupivacaine
50
Cardiac Rhythm Drugs
Antiarrhythmic drugs
51
Cardiac Contractility
Cardiac Glycosides Beta-adrenergic receptor Agonists PDE Inhibitors Calcium-sensitizing Agents
52
Volume Regulators (caridac)
Inhibs of RAS B-type Natriuretic Peptide ADH antagonists Agents that decrease Na reabs
53
Agents that modify vasc tone (cardiac)
Vasoldilators
54
Inhibs of RAS
ACE inhibs | Angiotensin Receptor Antagonists
55
ACE Inhibitors
``` Captopril Enalopril Lisinopril Benazepril Ramipril ```
56
Angiotensin Receptor Antagonists
Valsartan Losartan Tilmisartan
57
Vasodilators: Organic Nitrates
Nitroglycerine (NO) | Nitroprusside Na
58
Vasodilators: Ca Channel Blockers
Dihydropyridines | Non-dihydropyridines
59
Dihydropyridines
Amlodipine | Nifedipine
60
Non-dihydropyridines
Verpamil | Diltiazem
61
I A Class Antiarrhythmic Drugs
Quinidine | Procainamide
62
I B Class Antiarrhythmic Drugs
Lidocaine | Mexiletine
63
II Class Antiarrhythmic Drugs
Beta Blockers!!
64
First gen Beta blocker
Propranolol
65
2nd gen beta blocker
Metoprolol Atenolol Esmolol
66
3rd gen beta blocker
Carvedilol
67
III Class Antiarrhythmic Drugs
Sotalol | Amiodarone
68
IV Class Atiarrhythmic Drugs
Dihydropyridine: Amlodipine, Nifedipine | Non-Dihdropyridine: Verapamil, Diltiazem
69
Emetics
Apomorfin Xylazine Peripheral: Syrup of Ipecacuanha, 3-4% H2O2
70
Antiemetics: Local
Local anaesthetics- Lidocaine, Vit B6
71
Antiemetics: Systemic
``` Phenothiazines Dopamine antagonists Antihistamines Serotonin antagonists NK-1 receptor antagonists Parasympathomimetics ```
72
Antiemetics: Phenothiazines
Tiethylperazine Acepromazine Chlorpromazine Promethazine
73
Antiemetics: Dopamine antagonists
Metoclopramide | Domperidone
74
Antiemetics: Serotonin Antagonists
Ondansetron | Dolasetron
75
Antiemetics: Antihistamines
Dimenhydrinate | Diphenhydramine
76
Antiemetics: Neurokinin-1-Antagonists
Maropitant Citrate
77
Prokinetics/ Propulsive/ Modulators of gastric motility
``` Metoclopramide, Domperidone Cisapride Ranitidine, Nizatidine Parasympathomimetics: Neostigmin, Piridostigmin, Bethanecol Erythromycin ```
78
Laxatives
Stimulant Osmotic Colloidal Coating agents
79
Stimulant Laxatives
``` Phenophtalein Bisacodyl Emodin Aloe Docusate Atrakinone Derivs Castor Oil ```
80
Osmotic Laxatives
Na2SO4 MgSO4 Na- Citrate Lactulose
81
Colloidal Laxatives
Psyllium, cornmeal, pumpkin
82
Coating agents
Liquid parrafin
83
Antidiarrheals
Adsorbents Adstringents Motility Modifiers Treatment of chronic colitis
84
Antidiarrheals : Adsorbents
Activated charcoal Kaolin Montomorillonit
85
Antidiarrheals: Adstringents
``` Bismuth Salts (subsalicylate, subgallate, subnitrate, carbonate) Tannic acid ```
86
Antidiarrheals: Motility Modifiers
Parasympatholytics (atropine) | Morphine Derivs: Diphenoxylate, Loperamide
87
Treatment of Chronic Colitis
Sulfasalazine: Sulfapyridin and Amino-salicylic acid Mesalazine Olsalazine
88
Appetite Stimulants
``` B-Vits Anabolic steroids: Nandrolone, Stanozolone BZD: Diazepam, oxazepam Cyproheptidine Propofol ```
89
Antiulcer Drugs
Acid Neutralizers (Antacids) Acid Secretion Inhibitors: H2 antagonists and PPI's Drugs increasing mucosal resistance: PGE analogues, coating agents
90
Antiulcer: Acid Neutralizers/ Antacids
Systemic: NaHCO3 | Non-systemic: Mg(OH)2 and Al(OH)3 combo, Al-Mg carbonate
91
Antiulcer: H2 antagonists
Cimetidine Ranitidine Famotidine
92
Antiulcer: Proton Pump Inhibitirs (PPI's)
Omeprazole
93
Antiulcer: Drugs increasing mucosal resistance: PGE analogues
Misoprostole
94
Antiulcer: Drugs increasing mucosal resistance: Coating agents
Sucralfate: Sucrose Octasulfate and Al(OH)3
95
Hepatoprotectives
Cholagogues: Cholekinetics and Cholerectics Hepatoprotectants Lipotopic Agents
96
Hepatoprotectives: Cholagogues: Cholekinetics
UDCA: ursodeoxycholic acid Menbuton Clanobutin
97
Hepatoprotectants
``` Silymarin D-Penicillamin Glucose, fructose NAC: N-acetyl-Cysteine Vit E Vit C Selenium ```
98
Hepatoprotectives: Lipotropic Agents
Choline SAMe (S-Adenosyl Methionine) Methionine
99
Diuretics
Cardiac Diuretics Osmotic diuretics Natriuretics
100
Cardiac Diuretics
Digoxin Xanthine derivs: Caffeine, Theophylline, Theobromine ACE inhibs
101
Osmotic Diuretics
Mannitol | Glycerine
102
Natriuretics
PCT: Carboanhydrase Inhibs LOOP: Furosemide DCT: Thiazides CT: Potassium sparing diuretics
103
Natriuretics: Carboanhydrase inhibs
Acetazolamide Dorsalamide Brinzolamide
104
Natriuretics : Loop diuretics
Furosemide | Turosemide
105
Natriuretics : Thiazides
Hydrochlorothiazide | Chlorothiazide
106
Natriuretics: Potassium Sparing diuretics
Spironolactone
107
Combined treatment of CHF in dogs
Pimobendan and Furosemide and Spironolactone or | ACE Inhibs and Furosemide and Spironolactone
108
Combined treatment of CHF in cats
Furosemide and Spironolactone
109
Treating Hypertension
Amlodipine AT-II-Antag ACE inhibitor
110
Gandotropin releasing hormones (GnRH)
Buserelin Gonadorelin Fertilin Dezlorelin
111
Hormones of the Anterior pituitary/ Adenohypophysis
``` GH TSH ACTH PRL FSH and LH ```
112
Hormones of the posterior pituitary/ Neurohypophysis
Oxytocin | Vasopressin/ ADH
113
Growth hormones
Pure hST (human) Bovine bST Porcine pST But all are banned in the EU
114
Corticotropin, ACTH
Tetracosactrin
115
The ergolides/ PRL antagonists
Bromocriptidine | Cabergoline
116
What are the analogues of FSH and LH? i.e the non-pituitary gonadotropins
hCG= human corionic gonadrotropin (LH activity) | PMSG/eCG (FSH activity)
117
Insulin formualtions
Regular crystalline zinc insulin Isophane insulin Lente insulin Protamine Zinc Insulin (PZI)
118
Drugs influencing glucose metab i.e oral antidiabetics
Acarbose Sulphonylurea substances Biguanides
119
The sulphonylurea substances
``` Tolbutamide Chlorpropramide Metahexamide Glipizide/ Glibenclamide Glinides e.g Nateglinide Glitazones e.g pioglitazone ```
120
Biguanides
Fenformine Buformine Methformine
121
Short acting GC drugs
Cortisol | Cortisone
122
Middle acting GC drugs
Prednisolone Prednisone Methylprednisolone Triamcinolone
123
Long acting GC drugs
Dexamethasone Betamethasone Flumethasone
124
Treatment of Hypoadrenocorticism/ Addison's
``` Aldosterone Deoxycorticosterone Pivalat (DOCP) Fludrocortisone Acetate ```
125
Treatment of Hyperadrenocorticism/ Cushing's
Pituitary dependent: Bromocriptidine, Cyproheptidine HCl | Pituitary and or adrenal dependent: Ketoconazole, Mitotane, Trilostane
126
Preparations for Hypothyroidism
Crude thyroid products Iodine containing products: Iodised salt, Lugol's soln Synth preps: Levothyroxine, Levothyroxine Na, L-triiodothyronine, Liothyronine
127
Preparations for Hyperthyroidism
Thiouracil Methimazol/ Tiamazol Propylthiouracil Iodine
128
Prostaglandin systemic analogues
Cloprostenol Dinoprost Luprostiol Etiproston
129
Anticoccidials
``` Ionophores Triazines Sulphonamides Pyridine deriv: Clopidol Pyrimidine deriv: Amprolium Quinazolin deriv: Halofuginon Carbanilide deriv: Nicarbazin Guanidine deriv: Robenidine Quinoline deriv: Decoquinate Purine deriv: Aprinocid ```
130
Ionophore antibiotics:
``` Monensin Narasin Salinomycin Lasalocid Maduramycin Semduramycin ```
131
Sulphonamide anticoccidials
Sulphaquinoxaline | Sulphachlorpyrazine
132
Triazines anticoccidials
Toltrazuril | Diclazuril
133
Drugs for extraintestinal coccidia: | Toxoplasmosis and canine neosporosis
Clindamycin | Sulfadiazine and Pyrimethamin
134
Drugs for extraintestinal coccidia: | Only toxoplasmosis
Doxycycline | Decoquinate
135
Classes of benzimidazoles
Thiazolil benzimidazoles Benzimidazole carbamates Probenzimidazoles
136
Thiazolil benzimidazoles
Thiabendazole | Cambendazole
137
Benzimidazole Carbamates
``` Albendazole Flubendazole Fenbendazole Mebendazole Oxfendazole Oxibendazole Ricobendazole Luxabendazole Triclabendazole ```
138
Probenzimidazoles= Prodrugs
Febantel- fenbendazole- oxfendazole Netobimin- albendazole- ricobendazole Thiophanate- lobendazole
139
Imidazothiazoles
Tetramisole | Levamisole
140
Tetrahydopyrimidines
Pyrantel Morantel Oxantel
141
Salicylanilides
``` Closantel Oxyclozanide Rafoxanide Brotianide Clioxanide Niclosamide ```
142
Substituted Phenols
``` Nitroxinil Bithionol Disophenol Dichlorophene Diamphenethide Nitroscanate ```
143
Isoquinolin and Benzazepin Derivs
Praziquantel | Epsiprantel
144
Macrocyclic Lactones
Avermectins | Milbemycins
145
Avermectins
``` Abamectin Ivermectin Doramectin Eprinomectin Selamectin ```
146
Milbemycins
Milbemycin oxime | Moxidectin
147
Chemical classes of ectoparasiticides
``` Organophosphates Carbamates Pyrethroids Formamidines Macrocyclic lactones Phenylpyrazoles Indoxacarb Neonicotinoids Isoxazolines IGR's ```
148
Organophosphates
Diazinon Coumaphos Phoxim Fenthion
149
Carbamates
Propoxur
150
Pyrethroids
Tetramethrin Permethrin Deltamethrin Flumethrin
151
Formamidines
Amitraz
152
Neonicotinoids
Imidacloprid Nitenpyramin Dinotefuran
153
Phenylpyrazoles
Fipronil | Pyriprol
154
Juvenile hormone analogues
Pyriproxyfen | Methoprene
155
Chitin inhibitors
Lufenuron | Novaluron
156
Progestagens/ Gestagens (synth)
``` Fluorogestone acetate Norgestomet Proligestone Medroxyprogesterone acetate Altrenogest Megestrol acetate ```
157
Progesterone antagonists
Aglepriston | Bromocriptidine and Cabergoline
158
Oestrogens (synth)
Estradiol benzoate Estradiol cypionate Estradiol valerate Estradiol incurin
159
Androgens (synth)
Testosterone undecanoate Testosterone phenylpropionate Methyltestosterone and etinyl-estradiol
160
Anabolic steroid
Stanazolole Metandienone Nandrolone
161
Anti-Androgens
Cyproterone | Delmadinon
162
Uterine Stimulants
Oxytocin Ergot alkaloids Prostaglandins
163
Oxytocin deriv
Carbetocin
164
Ergot alkaloids
Ergotoxin Ergotamine Erogometrine (maleate salt and methyl ergometrine)
165
Prostaglandins
Etiproston Luprostiol Dinoprost
166
Uterine relaxing agents
Antispasmodics | Beta adrenoceptor agonists
167
Antispasmodics (uterine)
Danaverin Vetrabutin/ Dimophebumine Proquamezine, Aminopromazin
168
Beta adrenoceptor agonists (uterine)
Clenbutarol Terbutaline Isoxsuprine lactate
169
Isoxazolines
Fluralaner Afoxolaner Sarolaner Lotilaner
170
Antifungal drugs
Poliene AB's Azoles (imidazoles and triazoles) Allylamines Inhibitor of fungal mitosis (griseofulvin) Inhibitor of fungal nucleic acid (flucytosine) Lufenuron Echinocandins
171
Poliene AB's
Natamycin Nystatin Amphotericin B
172
Azoles
``` Imidazoles: Thiabendazole Clotrimazole Enilconazole Miconazole Bifoconazole Ketoconazole ``` ``` Triazoles: Posaconazole Itraconazole Fluconazole Voriconazole ```
173
Allylamines
Terbinafin | Naftidine
174
Echinocandins
Caspofungin Micafungin Anidulafungin
175
Drugs acting on the respiratory system
Bronchodilators Resp anti-inflamm drugs Antitussives Mucolytics, expectorants
176
The groups of bronchodilators
Sympathomimetics Parasympatholytics Methylxanthine derivatives
177
Non-specific sympathomimetics
Adrenaline Ephedrin Isoproterenol
178
Specific Sympathomimetics (acting on beta2)
Short-acting: Salbutamol Long-acting: Terbutaline Clenbutarole Salmeterole
179
Parasympatholytics (resp)
Ipratropium Atropine Glycopyrrolate
180
Methylxanthine derivatives
Caffeine Theophylline Theobromine
181
The respiratory anti-inflammatories
Inhalational Glucocorticoids Chromones Leukotriene antagonists
182
Inhalational glucocorticoids
Inhalosol dosage form Beclomethasone Fluticasone
183
Chromones
Na-chromoglycate | Nedocromil
184
Leukotriene synthesis inhibitors
Zileuton | Fenleuton
185
Leukotriene antagonists
Zafirlukast | Montelukast
186
Central antitussives
``` Codeine (vs morphine) Dihydrocodeine, hydrocodon Butorphanol Tramadol Dextrometorphen ```
187
Mucolytics
N-acetylcysteine | Carbocysteine
188
Expectorants
Bromhexin Ambroxol Dembrexine Guaifenesin
189
Anaemia: Erythropoietin as a drug
``` Epoetin alpha (rhEPO-alpha) Darbepoetin-alpha ```
190
Iron deficiency anaemia: oral
Iron fumarate iron glutamate Fe2+
191
Iron deficiency anaemia: IM
Iron dextran Fe3+ 100mg elemental iron/kg
192
Classes of 1st generation antihistamines
Ethylenediamines Ethanolamines Phenothiazines Piperidines
193
AH: Ethylenediamines
Chloropyramine | Chlorpheniramine
194
AH: Ethanolamines
Diphenhydramine | Dimenhydrinate
195
AH: Phenothiazine
Promethazine
196
AH: Piperidine
Cyproheptadine
197
2nd generation antihistamines
Loratidine Cetirizine Levocetirizine
198
Leukotriene synth inhibitors
Zileuton Fenleuton Adenosine
199
Leukotriene receptor antagonists
Montelukast | Zafirlulast
200
Human JAK inhibitors
Ruxolitinib | Tofacitinib
201
Vet JAK inhibitors
Oclacitinib-apoquel
202
Monoclonal antibodies
Lokivetmab-cytopoint
203
NSAID's classification
Salicylates Acetic acid derivatives Arilpropionic acids Acidic substances: Heteroaryl acetic acids, butyl pyrazolidines, anthranilic acids Non-acid substances: Anilin derivs, pyrazoles
204
NSAID's acetic acid derivs
Diclofenac | Eltenac
205
NSAID's arilpropionic acid deriv's
``` Ketoprofen Vedaprofen Carprofen Ibuprofen Naproxen ```
206
NSAID's acidic substances
Heteroaryl acetic acids: Diclofenac, Indomethacin, Etoldolac Butyl pyrazolidines: Phenylbutazone Anthranilic acids: Flunixin meglumine, Tolfenamic acid, Meloxicam
207
NSAID's non-acidic substances
Anilin derivatives: paracetemol | Pyrazolones: Metrimidazole Na
208
NSAID's: Selective COX= COXIBs
``` Deracoxib Firocoxib Robendacoxib Cimicoxib Mevacoxib ```
209
Immunosuppression: classification of drugs
Inhibitors of gene expression Cytotoxic agents: antimetabolites and alkylating agents Specific lymphocyte-signalling inhibitors Cytokine inhibition: TNFalpha inhibs and IL-1 inhibs
210
Inhibitors of gene expression
Glucocorticoids
211
Cytotoxic agents: Antimetabolites
Purin analogues: Azathioprene, Mycophenolate mofetil Pyrimidine analogue: Leflunomide FA antag: Methotrexate
212
Cytotoxic agents: Alkylating agents
Cyclophosphamide
213
Specific lymphocyte-signalling inhibs (calcineurin inhibs)
Cyclosporin | Tacrolimus, Pimecrolimus
214
Cytokine inhibs: TNFalpha inhibs
Adalimumab Infiximab Etanercept
215
Cytokine inhibs: IL-1 inhibs
Anakira
216
Antiviral drugs: Pyrimidine analogues
Idoxuridin | Trifluridin
217
Antiviral drugs
``` Acyclovir Gancyclovir Famciclovir Vidarabin Zidovudin Oseltamavir ```
218
Neuramidinase and ion channel inhibitors against influenza virus
Amantadine | Rimantidine
219
Antineoplastic agents
``` Antimetabolites Agents that directly modify DNA structure Topoisomerase inhibitors Microtubule inhibitors GC's-- lymphoma and mastocytoma Other ```
220
Antineoplastic: antimetabolites
Methotrexate 5-FU Cytarabin
221
Antineoplastic: Agents that directly modify DNA structure
Alkylating: Cyclophosphamide Chlorambucil Lomustine Platinum compounds: Cisplatin Carboplatin
222
Antineoplastic: Topoisomerase inhibs
Anthracyclines- Topoisomerase II: Doxorubicin GZ Mitoxantrone
223
Antineoplastic: Microtubule inhibs
``` Inhibit microtubule polymerization: Vinblastine Vinchristine Inhibit microtubule depolymerization: Pacltaxel ```
224
Classes of drugs with analgesic activity
Narcotic analgesics: opioids Non-narcotic: antipyretics, NSAID's Antoconvulsive/ Antiepileptics: Gabapentin, Pregabalin, Iamotrigin, Carbamazepine Anti-arrythemic: Mexileting, Lidocaine NMDA receptor antagonists: Ketamine, Tiletamine, Dextrometorphan Alpha-2 agonists: Xylazine, Medetomidine Local anaesthetics General anaesthetics
225
Aminoquinolines
Chloroquine | Primaquine
226
Hydroxy (hakogenated) FQ's
Chlorquinaldole
227
Isoquinolone derivatives (FQ's)
Papaverine | Praziquantel
228
1st gen 4 Quinolones
Oxolinic acid Nalidixic acid Pipemedic acid
229
1st gen Fluoroquinolones 2
Flumequin | Norfloxacin
230
2nd gen Fluoroquinolones 2
``` Enrofloxacin Marbofloxacin Ibafloxacin Danofloxacin Orbifloxacin Difloxacin Ciprofloxacin ```
231
3rd and 4th gen fluoroquinolones
Moxifloxacin | Pradofloxacin