03 - Synaptic Flashcards
pilocarpine
muscarinic agonist
atropine
muscarinic antagonist
scopolamine
muscarinic antagonist
anaesthetic pre-med
pancuronium (-onium)
nicotinic antagonist (competitive blocker) non-depolarising block
nicotinic agonist
duh..
depolarising block
acts on NMJ and autonomic ganglia
trimetaphan
ganglia blocker
hexamethonium
ganglia channel
via channel block
bromopyruvate
Drugs acting pre-synaptically
target: pyruvate
hemicholinium
Drugs acting pre-synaptically
target: choline transport
vesamicol
Drugs acting pre-synaptically
target: vesicle transport
botulinum toxin
Drugs acting pre-synaptically
target: exocytosis
edrophonium
anti-AChE
short-acting for M.S. diagnosis
neostigmine
anti-AChE
medium-acting for M.S. treatment
dyflos
anti-AChE
long-acting / irreversible
clonidine
(1) alpha(2) autoreceptor agonist