04 - Cardiovascular Flashcards
ezetimibe (EZ)
dyslipidaemic drug
increase intestinal cholesterol absorption
only dyslipidaemic drug without increase HDL
fenofibrate (ff)
dyslipidaemic drug
1) increase muscle LPL
2) increase HDL
niacin
dyslipidaemic drug
1) decrease hormone-sensitive lipase
2) increase HDL
colestyramine
dyslipidaemic drug
1) decrease bile reabsorption
2) increase HDL
statin
dyslipidaemic drug
1) inhibit HMG-CoA reductase
2) increase HDL
ticagrelor
anti-platelet drug
inhibit ADP receptor
eptifibatide (tiff)
anti-platelet drug
inhibit GPIIa/IIIb
aspirin
anti-platelet drug
inhibit PG release
warfarin
anti-coagulant
inhibit VKOR –> inhibit factor X and factor II
heparin
anti-coagulant
inhibit factor Xa and IIa via ATIII
enoxaparin (enoch)
anti-coagulant
inhibit factor Xa selectively via ATIII
dabigatran
anti-coagulant
inhibit factor IIa directly
streptokinase
thrombolytic
activates fibrin-bound and circulating PLG non-selectively
tenecteplase
thrombolytic
activates fibrin-bound PLG selectively
ivabradine (brad)
drugs for IHD
decrease funny current