20. Agonists Flashcards

1
Q

What is a ligand?

A

Chemical that specifically binds to a receptor

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2
Q

What is an agonist?

A

Ligand that binds and causes a biological response

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3
Q

What is the dose-response relationship?

A

Tissue response is generally directly proportional to the ratio of receptors occupied with the agonist

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4
Q

What is potency?

A

Measure of drug activity

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5
Q

What is a partial agonist?

A

One that never produces the max response

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6
Q

What does it mean to have spare receptors?

A

The maximum response has been reached but not all receptors used

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7
Q

Name two ways of studying drug interactions

A
  1. Functional studies

2. Binding studies

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