Semester 2 Exam II Drugs Flashcards
(110 cards)
Levodopa
Dopaminergic agent; precursor in dopamine synthesis, crossed BBB
Carbidopa
Decarboxylation inhibitor (never monotherapy)
Carbidopa/levodopa (Sinemet)
Preferred Parkinson’s treatment
Bromocriptine
Ergot dopamine agonist
Ropinirole
Non-ergot dopamine agonist (Parkinson’s or restless leg)
Pramipexole
Non-ergot dopamine agonist (Parkinson’s or restless leg)
Selegiline
Monoamine oxidase type B inhibitor (always use with sinemet)
Rasagiline
Monoamine oxidase type B inhibitor (always use with sinemet)
Amantadine
Alternative to MAO-B inhibitor
Entacapone
COMT inhibitor (always with sinemet)
Tolcapone
COMT inhibitor (always with sinemet)
Pimavanserin
Atypical antipsychotic (only for Parkinson’s associated psychosis)
Tetrabenazine
VMAT-2 inhibitor (for chorea management)
Propranolol
Beta blocker (for essential tremor)
Atenolol
Beta blocker (for essential tremor)
Nadolol
Beta blocker (for essential tremor)
Metoprolol
Beta blocker (for essential tremor)
Primidone
Anticonvulsant (best choice for essential tremor)
Gabapentin
Anticonvulsant (essential tremor)
Topiramate
Anticonvulsant (essential tremor)
Interferon beta-1a
Interferon (MS) (SC)
Interferon beta-1b
Interferon (MS) (SC)
Glatiramer acetate
Immunomodulator for MS (daily SC)
Fingolimod
Immunomodulator for MS (PO)