Drug card quiz 3 Flashcards
(45 cards)
Urinary bladder modifier
Solifenacin Succinate
Oxybutynin Chloride
Tolterodine Tartrate
Solifenacin Succinate
Oxybutynin Chloride
Tolterodine Tartrate
Vesicare
Ditropan, Ditropan XL
Deltrol, Deltrol XR
Urinary bladder modifier
Dosage
Solifenacin Succinate
5 mg, 10 mg
Oxybutynin Chloride
Tablet : 5 mg, 10mg, 15 mg
Syrup : 5mg/ 5mL
(available in topical patch)
Tolteridone : 1 and 2
2,4
Urinary bladder modifier indications
- overactive bladder
Vesicare,ditropan =5mg
Detrol = 4
Urinary bladder modifier
MOA
Solifenacin, Tolterodone :
competitive muscarinic receptor antagonist
Oxybutynin Chloride :
inhibits muscarinic action of ACH on smooth muscle
Urinary bladder modifier
contraindications
- urinary retention
-gastric retention - uncontrolled narrow angle glaucoma
Detrol, Vesicare :
-nursing mothers
Urinary bladder modifier
adverse effects
dry mouth, constipation, blurred vision,dizziness
Solifinacin : UTI, abdominal pain
Urinary bladder modifier
PC
- avoid hot weather
- care operating heavy machinery/mental alertness
Oxybutinin, Solifenacin : - swallow whole
Tolteridone :
No alcohol
Cephalosporin
Sulfonamide Antiobiotics
Antibacterial
Cephalexin Monohydrate
Nitrofurantoin
Sulfamethoxazole w/ Trimethoprim
Cephalexin Monohydrate
Nitrofurantoin
Sulfamethoxazole w/ Trimethoprim
Keflex
Macrodantin, Macrobid, Furadantin
Bactrim, Septra
Antibacterial
dosage
Cephalexin :250 mg, 500mg , 750mg
powder
Nitrofuran : 25,50,100
suspension
Sulfamethoxazole : T80,S400
suspension, injection
250mg to 1 g every six hours
Antibacterial
indications
Nitrofuran, Cephalexin, Sulfamethoxazole:
UTI, bacterial infection
Sulfamethoxazole :
travelers diarrhea, pneumonities (PCP)
Antibacterial
MOA
Cephalexin : acylation of transpeptidase enzyme
Nitrofuran : inhibition of acetyl co-enzyme A
Sulfamethoxazole : inhibiting enzyme dihydrfolate reductase
Antibacterial
interactions
Keflex : oral contraceptives
false positive for tests
Macrobid : Mg
Bactrim : Cyclosporine
Antibacterial
contraindications
Impaired renal fxn
Septra, Keflex : sulfa drug allergy,
Septra, Macrodantin : pregnancy, infants,
Macrodantin : anuria,oliguria,
Keflex : penicillin,
Septra: magaloblastic anemia
Antibacterial
adverse effects
Nitrofuran, Cephalexin, Sulfomethoxazole : nausea , vomiting , diarrhea , hives, itching, rash
Sulfamethoxazole : stevens Johnsons syndrome, sunlight sensitivity
Antibacterial PC
Nitrofuran : urine discoloration
Cephalexin, Sulfomethoxazole : empty stomach 2 hours
Sulfamethoxazole : sunlight sensitivity
COPD
Ipratropium Bromide
Ipratropium Bromide w/ Albuterol Sulfate
Tiotropium Bromide
Ipratropium Bromide
Ipratropium Bromide w/ Albuterol Sulfate
Tiotropium Bromide
Atrovent
Combivent, DuoNeb
Spirivia
(inhalers )
COPD Indications
bronchospasm w/ COPD
Tiotropium : asthma
Ipratropium Bromide : Rhinorrhea
COPD MOA
ipratropium sulfate : stimulates adenyl cyclase to form c-AMP
Tiotropium : long acting antagonist of ACH @ M3
Ipratropium bromide : anticholinergic agent
COPD
contraindications
renal impaired,
Ipatropium Bromide, Tiotropium : glaucoma
Ipratropium Sulfate : peanut allergy
COPD adverse effects
Iprotropium Sulfate : chest pain,abdominal pain, constipation
Iprotropium Bromide :oropharynx, GI distress, epistaxis, pharyngitis
Tiotropium : moniliasis, epistaxis, constipation
GI antiplasmodics
Hyoscyamine sulfate
Dicyclomine Hydrochloride
Beers list