Drug Discovery And Design Flashcards

(10 cards)

1
Q

Target-based fasi
MOLECULAR DOCKING

A
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2
Q

Ligand-based fasi
QSAR
PHARMACOPHORE MODELLING
FRAGMENT BASED DRUG DISCOVERY

A
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3
Q

Regola di lipinski o del 5, come la uso

A
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4
Q

Definizione di QSAR e workflow

A
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5
Q

3D QSAR
COMFA APPROCCIO

A
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6
Q

Molecular docking

A
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7
Q

Fragment based
Differenze tra growing e linking

A
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8
Q

Fasi del fragment based

A
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9
Q

Confronto HTS e Fragment based

A
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10
Q

LE ligand efficiency

A
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