l16 Flashcards
first synapse release what to what receptors
Acetylcholine to nicotinic receptors
Nicotine is agonists or antagonists nicotinic receptors are what channel
agonist
- ligand gated channel
- direct
cholinergic receptors
receive acetycholine
can b g coupled or ligand gated
parasympathetic second synapse release what to what
acetycholyne to muscurania receptors
muscarinic receptors
muscarine is agonist
- receptor is g coupled channels
- activate second messenger
sympathetic second synapse release what to what
noradrenaline to adrenergic receptors
adrenergic receptors
a class of g coupled
- receive norepinephrine (noradrenaline) and epinephrine (adrenaline).
a1 adrenoreceptor excitatory
Smooth muscle:
vascular
genitunary (sphincter, urinary bladder)
heart
liver
eyes
CNS post synaptic neuron
saliva
a1 adrenoreceptor inhibitory
smooth muscle intestinal
a2 adreno receptor inhibitory
pre + post synaptic neuron, cns and
-> pancreas platelets
b1 excitatory adreno
cns post synaptic
intestinal
heart
rena juxtaglomarular (regulate blood pressure - blood vessel)
b2 excitatory adreno
cns post-synaptic, intestinal, bronchial, skeletal mus vascula bed + skeletal mus liver eyes (cililary muscle) mast cell, blood vessel, detrusor muscle (urinary)
b3 excitatory adreno
adipose tissue
sympathetic innervation: tissue influenced by a1 + effects:
eye iris (contract radial muscle)
saliva gland (release k+)
blood vessel (contraction constriction of vascular muscle in skin, mucosa, abdominal)
gastrointestinal (contraction - sphincter)
urinary bladder (contraction - sphincter)
sympathetic innervation: tissue influenced by b1 + effects:
salivary (amylase secretion)
heart (increase contraction sa node, automaticity av node)
sympathetic innervation: tissue influenced by b2 + effects:
eye ciliary muscle (relax far vision)
bronchi (relax/dilation smooth muscle)
blood vessel (dilation coronary vessel, vasculature in skeletal muscle bed)
gastrointestinal tract (relax sphincter)
urinary bladder (relax detrusor)
skeletal muscle (tremor, glycogenolysis)
mast cell (inhibition of histamine release)
sympathomemtic
insomnia
restlestness
tremor
palpitation
tachyrcardia
adrenergic agonist