Pharm - ANS Drugs Flashcards
(35 cards)
Neostigmine
Anti-AChE; bowel & bladder, mysethenia gravis
a-methyldopa
Hypertension in pregnancy
Rivastigmine
Anti-AChE; Alzheimer
Isoproterenol
B1 = B2 agonist; Tachyarrhythmia evaluation
Phyostigmine
Anti-AChE; Anticholinergic toxicity (crosses blood-brain border)
Pilocarpine
Cholinomimetic; Glaucoma
Amphetamine
General SNS agonist; narcolepsy, obesity, ADD
Epinephrine
B > a agonist; Anaphylaxis, open-angle glaucoma, asthma
Methacholine
Cholinomimetic; asthma challenge test
Carbachol
Cholinomimetic; Glaucoma
Pyridostigmine
Anti-AChE (long-acting); Myesthenia gravis
Oxybutynin, darifenacin, solifenacin
Muscarinic antagonists; Reduce bladder spasms
Norepinephrine
a1 > a2 > B1 agonist; hypotention
Dobutamine
B1 > B2, a agonist; Heart failure
Benztropine
Muscarinic antagonist; Parkinson disease
Phenoxybenzamine
a antagonist; pheochromocytoma
Carvedilol
Nonselective a/B antagonist
Dopamine
D1 = D2 > B > a agonist; Unstable bradycardia, heart failure, shock
Cocaine
General SNS agonist
Edrophonium
Anti-AChE (short-acting); myasthenia gravis diagnosis
Atropine
Muscarinic antagonist; bradycardia, pupil dilation
Ipratropium, tiotropium
Muscarinic antagonist; COPD/asthma
Labetalol
Nonselective a/B antagonist
Phenylephrine
a1 > a2; Hypotention, ocular procedures, rhinitis