Acetylcholinesterase inhibitors Flashcards
(4 cards)
1
Q
Drugs
A
Donepezil (Aricept)
Galantamine (Razadyne)
Rivastigmine (Exelon)
Neostigmine
Pyridostigmine
Physostigmine
2
Q
MOA
A
inhibit acetylcholinesterase from destroying ACh, increasing ACh levels
3
Q
AE/SE
A
GI, bradycardia
Cholinergic crisis (SLUDGE and Killer Bs)
4
Q
Indication
A
Alzheimer’s
Neo/pyrido are also used for MG
Physostigmine also treats anticholinergic toxicity, MG, neuromuscular blocker reversal