Gliptins/DPP4i DI Flashcards Preview

PHM 602- Diabetes > Gliptins/DPP4i DI > Flashcards

Flashcards in Gliptins/DPP4i DI Deck (20)
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1
Q

DPP4i MoA

A

potentiate effects of incretin hormones

2
Q

DPP4i drugs

A

Sitagliptin (Januvia)
Saxagliptin (Onglyza)
Linagliptin (Tradjenta)
Alogliptin (Nesina)

3
Q

Brand name for sitagliptin

A

Januvia

4
Q

Brand name for saxagliptin

A

Onglyza

5
Q

Brand name for linagliptin

A

Tradjenta

6
Q

Brand name for alogliptin

A

Nesina

7
Q

DPP4i side effects

A

nasopharyngitis, URI

8
Q

DPP4i precaution

A

HF, use with GLP-1RA

9
Q

DPP4i counseling

A

Take once a day at the same time each day, can be taken with or without food, avoid alcohol

10
Q

What should you ask about at DPP4i refills?

A

URI and nasopharyngitis

11
Q

DPP4i clinical pearls

A

Intermediate A1C lowering, neutral weight gain, neutral ASCVD and CKD effects, increased HF risk with saxagliptin and alogliptin

12
Q

Renal dosing in DPP4is

A

All require renal dosing except for linagliptin

13
Q

DPP4i monitoring

A

A1C, FBG/PPG, URI, GI disturbances

14
Q

DPP4i peak effect

A

6-8 weeks

15
Q

DPP4is in ADA guidelines

A

Used to minimize hypoglycemia

16
Q

DPP4is in AACE guidelines

A

4th-line option after metformin, GLP-1 RA, SGLT2is

17
Q

Sitagliptin dosing

A

100mg QD

18
Q

Linagliptin dosing

A

5mg QD

19
Q

Saxagliptin dosing

A

5mg QD

20
Q

Alogliptin dosing

A

25mg QD