lecture 9 Flashcards
(20 cards)
adrenaline
hormone, binds all alpha and beta receptors
noradrenaline
neurotransmitter, mostly is retaken up, binds mostly alpha receptors
alpha adrenoreceptor
everything to do with calming down the body, vasodilation/constriction
beta adrenoreceptor
have to do with metabolism, also cardiac arrest and allergies
alpha 2 receptor
presynaptic autoreceptor, inhibition of AC, noradrenaline release
isoprenaline
binds all beta receptors
alpha 1/2 receptor
smooth muscles, glands
beta 1 receptor
heart (metabolism)
beta 2 receptor
smooth muscles, metabolism, bronchial dilation
beta 3 receptor
lipolysis
clonidine, oxymetazoline
bind alpha 2 receptor
phenylephrine
binds alpha 1 receptor
fenoterol, salbutamol
bind beta 2 receptor, short acting inhalation drugs
PLC is activated by which subunits of which proteins
beta gamma of Gi and alpha of Gq, causing vasoconstriction
positive chronotrope
Na+, increases heart rate, SA node
positive inotrope
Ca2+, increases heart contractility, cardiac muscles
arrythmia
permanent change in heart rate or heartbeat
adams stoke attack
too much ACh can activate a too active vagus causing fainting
renin (kidneys)
alpha 2 decreases renin, beta 1 increases renin
tyramine
helps sodium and NA get into presynaptic area and NA also in vesicles once its there