Cholinergic Receptor Inhibitors Class/mechanism Flashcards Preview

Pharm Unit 2 MJC > Cholinergic Receptor Inhibitors Class/mechanism > Flashcards

Flashcards in Cholinergic Receptor Inhibitors Class/mechanism Deck (14)
1

Atropine

Tertiary amine antimuscarinic
blocks muscarinic receptors

2

scopolamine (transderm-scop)

Tertiary amine antimuscarinic
blocks muscarinic receptors

3

Dicyclomine (Bentyl)

Tertiary amine antimuscarinic
blocks muscarinic receptors

4

Tropicamide (mydriacyl)

Tertiary amine antimuscarinic
blocks muscarinic receptors

5

Tolterodine (detrol)

Tertiary amine antimuscarinic
blocks muscarinic receptors

6

Benztropine (Cogentin)

Tertiary amine antimuscarinic
blocks muscarinic receptors

7

Ipratropium (Atrovent)

Quaternary amine antimuscarinic
blocks muscarinic receptors

8

Tiotropium (spiriva)

Quaternary amine antimuscarinic
blocks muscarinic receptors

9

Hexamethonium (Methium)

Ganglionic blocker
blocks ganglionic Nn/N2 receptor and sympathetic tone

10

Mecamylamine

ganglionic blocker (Crosses BBB)
blocks ganglionic Nn/N2 receptor and sympathetic tone

11

Succinylcholine (Anectine)

Depolarizing blocker
overstimulation of nicotinic receptor, leading to desensitization of muscle unit to further ACh stimulation

12

Tubocurarine (Curare)

Nondepolarizing blocker
blocks nicotinic Nm/N1 receptor

13

Mivacurium (Mivacron)

Nondepolarizing blocker
blocks nicotinic Nm/N1 receptor

14

Botulinum toxin A (Botox)

Local paralytic
Blocks vesicle fusion and ACh release on presynaptic terminal by degrading SNAP-25