CYP450s inhibitors, inducers and sulfas Flashcards

(35 cards)

1
Q

AAA RACKS IN GQ M

CCGPPRNSN

A

yep

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
2
Q

acute alcohol abuse

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
3
Q

chronic alcohol abuse

A

inducer

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
4
Q

ritonavir

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
5
Q

amiodarone

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
6
Q

cimetidine

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
7
Q

ketoconazole

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
8
Q

sulfonamides

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
9
Q

isoniazid

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
10
Q

grapefruit juice

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
11
Q

quinidine

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
12
Q

macrolides

A

inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
13
Q

st johns wort

A

inducer

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
14
Q

phenytoin

A

inducer

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
15
Q

phenobarbital

A

inducer

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
16
Q

nevirapine

17
Q

rifampin

18
Q

griseofulvin

19
Q

carbamazepine

20
Q

list all inhibitors

A

acute alcohol abuse, ritonavir, amiodarone, cimetidine, ketoconazole, sulfomamides, isoniazid, grapefruit guice, quinidine, macrolides

21
Q

list all inducers

A

chonic alchol abuse, ste johns ort, phenytoin, phenobarbital, nevirapine, rifampin, grisefulvin, carbamazepine

22
Q

list all substrates

A

A TWO

antipsychotics, theophylline, warfarin, OCP

23
Q

antipsychotics

24
Q

theophylline

25
warfarin
substrate
26
OCP
substrate
27
list all the sulfa drugs
PFACTSSS: probenecid, furosemide, acetazolamide, celecoxib, thiazides, sulfonamide antibiotics, sulfasalazine, sulfonylureas
28
probenecid
sulfa drug
29
furosemide
sulf drug
30
acetazolamide
sulfa drug
31
celecoxib
sulfa drug
32
thiazides
sulfa drug
33
sulfonamide antibiotics
sulfa drug
34
sulfasalazine
sulfa drug
35
sulfonylureas
sulfa drug