Anxiolytics and Hypnotic Drugs 1 (Benzos) Flashcards
(12 cards)
Benzodiazepines
What is the primary use of Alprazolam (Xanax)?
Anxiety, phobias
Alprazolam increases the binding of GABA and enhances chloride influx with an action duration of approximately 15 hours.
Benzodiazepines
What is the action duration of Diazepam (Valium)?
Approximately 36 hours
Diazepam is used for anxiety, phobias, and epilepsy, increasing GABA binding and chloride influx.
Benzodiazepines
What condition is Flurazepam (Dalmane) primarily used to treat?
Insomnia
Flurazepam enhances GABA binding and chloride influx, with an action duration of around 36 hours and does not cause rebound sleep.
Benzodiazepines
What is the action duration of Lorazepam (Ativan)?
Approximately 15 hours
Lorazepam is used for anxiety and phobias, increasing GABA binding and chloride influx.
Benzodiazepines
What is Midazolam (Versed) used for?
Anxiety, preanesthetic, IV anesthetic
Midazolam increases GABA binding and chloride influx with an action duration of about 5 hours.
Benzodiazepines
What is the primary indication for Temazepam (Restoril)?
Insomnia
Temazepam enhances GABA binding and chloride influx, with an action duration of approximately 15 hours.
Benzodiazepines
What is the action duration of Triazolam (Halcion)?
Approximately 5.5 hours
Triazolam is used for insomnia and increases GABA binding and chloride influx.
Benzodiazepines
Fill in the blank: _______ is used to treat anxiety and phobias, with an action duration of about 15 hours.
Lorazepam (Ativan)
Benzodiazepines
True or False: Flurazepam (Dalmane) causes rebound sleep.
False
Flurazepam is noted for not causing rebound sleep despite its use in treating insomnia.
Benzodiazepines
List three uses of Diazepam (Valium).
- Anxiety
- Phobias
- Epilepsy
Benzodiazepines
What is the mechanism of action for benzodiazepines?
Increases binding of GABA and chloride influx
name: 7 Benzodiazepines
Alprazolam (Xanax)
Diazepam (Valium)
Flurazepam (Dalmane)
Lorazepam (Ativan)
Midazolam (Versed)
Temazepam (Restoril)
Triazolam (Halcion)