Respiratory (Asthma) drugs Drug 1 Flashcards
(39 cards)
β-Adrenergic Agonists
What are β-Adrenergic Agonists used for?
Asthma, Anaphylactic shock
They cause bronchodilation.
β-Adrenergic Agonists
What is the effect of Epinephrine on adenylyl cyclase?
↑ adenylyl cyclase
β-Adrenergic Agonists
What does Epinephrine increase in cells?
↑ cAMP
β-Adrenergic Agonists
True or False: Epinephrine causes bronchodilation.
True
Methylxanthines
What are Methylxanthines used for?
Asthma
Methylxanthines
What is the effect of Theophylline on phosphodiesterase?
↓ cAMP phosphodiesterase
Methylxanthines
What is the result of increased cAMP due to Theophylline?
Bronchodilation
Methylxanthines
Fill in the blank: Theophylline increases _______ leading to bronchodilation.
cAMP
Anticholinergics
What are Anticholinergics?
A class of drugs that block the action of acetylcholine in the body.
Anticholinergics
What is Ipratropium?
An anticholinergic drug used for asthma.
Anticholinergics
How does Ipratropium compare to β2-agonists in terms of bronchodilation?
Produces less bronchodilation than β2-agonists.
Corticosteroids
What is Beclomethasone also known as?
Vanceril
Beclomethasone is a corticosteroid used as a bronchodilator and steroid inhaler.
Corticosteroids
What is the primary function of Budesonide?
Bronchodilator, steroid inhaler, ↓ Prostaglandin synthesis
Budesonide is marketed as Rhinocort Aqua.
Corticosteroids
Which corticosteroid is known as Flovent?
Fluticasone propionate
Fluticasone propionate functions as a bronchodilator and steroid inhaler.
Corticosteroids
What type of medication is Methylprednisolone?
Respiratory, steroid IV or oral, anti-inflammatory
Methylprednisolone can be administered intravenously or orally.
Corticosteroids
What is Mometasone used for?
Corticosteroid, ↓ action of inflammation mediators
Mometasone is marketed as Nasonex.
Corticosteroids
What is the main action of Prednisone?
Bronchodilator, anti-inflammatory, ↓ Prostaglandin synth.
Prednisone is a commonly prescribed corticosteroid.
Corticosteroids
Fill in the blank: Fluticasone propionate is a __________.
Bronchodilator, steroid inhaler, ↓ Prostaglandin synthesis
Corticosteroids
True or False: Mometasone is a bronchodilator.
False
Mometasone is a corticosteroid, not a bronchodilator.
Corticosteroids
Which corticosteroid can be administered both IV and orally?
Methylprednisolone
Corticosteroids
Fill in the blank: Budesonide is marketed as __________.
Rhinocort Aqua
Corticosteroids
What is the mechanism of action for corticosteroids like Beclomethasone?
↓ Prostaglandin synthesis
Name a corticosteroid used for asthma management
Beclomethasone (Vanceril)
Beclomethasone is commonly used as an inhaled corticosteroid for asthma treatment.
What is Budesonide also known as?
Rhinocort Aqua
Budesonide is often prescribed for allergic rhinitis and asthma.