Pharmacodynamics Pt. II Flashcards Preview

Fundamentals of Molecular Medicine > Pharmacodynamics Pt. II > Flashcards

Flashcards in Pharmacodynamics Pt. II Deck (24)
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1
Q
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2
Q

Agonist vs. Anatgonist vs. Antagonist 10X

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3
Q

Eqn for Agonist Alone

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4
Q

Eqn for Agonist + Competitive Antagonist

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5
Q

Competitive antagonist and the Schild Eqn

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6
Q

Applying the Schlid Eqn

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7
Q

Irreversible Antagonists

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8
Q

Irreversible Antagonists with Spare Receptors

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9
Q

Clinical Implications of Irreversible Antagonists

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10
Q

Overdoses

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11
Q

Reversible Competitive Antagonism

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12
Q

Reversible vs. Irreversible Antagonists

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13
Q

Spare Receptors and Physiological Response

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14
Q

Response time vs. Absolute Sensitivity

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15
Q

Transmembrane signaling Mechanisms

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16
Q

G-Protein Coupled Receptors

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17
Q

Two Common Signaling Pathways

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18
Q

Pharmacodynamics and regulating agonists and receptors

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19
Q

Allosteric Modulation of Receptors

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20
Q

Biased Agonists

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21
Q

Receptor Subtypes

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22
Q

Alpha 1 Receptor

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23
Q

Beta 1 Receptors

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24
Q

Beta II Receptors

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