4.5 pharm cholinergic Flashcards
(37 cards)
Reversible short acting AChE inhibitor
Donezepil
Edrophonium
Degrades SNARE proteins & prevents transmitter release
Botulinum toxin
Intermediate acting covalent / reversible inhibitor in myasthenia gravis
Neostigmine
Pyridostigmine
Long acting AChE inhibitor
Causes contraction of ciliary muscle to increase aqueous humor outflow
Ecothiophate
Irreversible organophosphate AChE inhibitor
Malathion
Sarin
Non depolarizing / competitive nicotinic receptor blocker
Atracurium
Depolarizing nicotinic receptor blocker
Succinylcholine
Muscarinic receptor agonist
Bethanechol
Muscarinic receptor antagonist
Atropine
Scopolamine
Tiotropium
Darifenacin
Palliative for Alzheimer’s
Donezepil
Open angle glaucoma
Ecothiophate
Bethanechol
Treats dry mouth
Bethanechol
Transdermal patch for motion sickness
Scopolamine
Inhaled for asthma and COPD
Tiotropium
Used for urinary incontinence (leak urine)
Botulinum toxin
Darifenacin
To increase urination
Bethanechol
Used for head lice
Malathion
Used for insecticide
Malathion
For skeletal muscle relaxation
Atracurium
Succinylcholine
Treats post operative pain
Bethanechol
Therapy for organophosphate poisoning
Atropine
Can cause skeletal muscle toxicity
Botulinum toxin
Causes Bradycardia as a side effect
Sarin
Atropine
Causes miosis ADR
Sarin